DK152211C - Analogifremgangsmaade til fremstilling af n-phenyl-n-(4-piperidinyl)-amider eller farmaceutisk acceptable syreadditionssalte deraf. - Google Patents

Analogifremgangsmaade til fremstilling af n-phenyl-n-(4-piperidinyl)-amider eller farmaceutisk acceptable syreadditionssalte deraf.

Info

Publication number
DK152211C
DK152211C DK193778A DK193778A DK152211C DK 152211 C DK152211 C DK 152211C DK 193778 A DK193778 A DK 193778A DK 193778 A DK193778 A DK 193778A DK 152211 C DK152211 C DK 152211C
Authority
DK
Denmark
Prior art keywords
amids
piperidinyl
analogue
phenyl
preparation
Prior art date
Application number
DK193778A
Other languages
Danish (da)
English (en)
Other versions
DK193778A (da
DK152211B (da
Inventor
Frans Eduard Janssens
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of DK193778A publication Critical patent/DK193778A/da
Publication of DK152211B publication Critical patent/DK152211B/da
Application granted granted Critical
Publication of DK152211C publication Critical patent/DK152211C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D257/00Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04Five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DK193778A 1977-05-05 1978-05-03 Analogifremgangsmaade til fremstilling af n-phenyl-n-(4-piperidinyl)-amider eller farmaceutisk acceptable syreadditionssalte deraf. DK152211C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US79381477A 1977-05-05 1977-05-05
US79381477 1977-05-05
US88618878A 1978-03-13 1978-03-13
US88618878 1978-03-13

Publications (3)

Publication Number Publication Date
DK193778A DK193778A (da) 1978-11-06
DK152211B DK152211B (da) 1988-02-08
DK152211C true DK152211C (da) 1988-08-08

Family

ID=27121432

Family Applications (1)

Application Number Title Priority Date Filing Date
DK193778A DK152211C (da) 1977-05-05 1978-05-03 Analogifremgangsmaade til fremstilling af n-phenyl-n-(4-piperidinyl)-amider eller farmaceutisk acceptable syreadditionssalte deraf.

Country Status (26)

Country Link
JP (1) JPS53149980A (ja)
AT (1) AT368994B (ja)
AU (1) AU514360B2 (ja)
CA (1) CA1105464A (ja)
CH (1) CH635585A5 (ja)
CY (1) CY1253A (ja)
DE (1) DE2819873A1 (ja)
DK (1) DK152211C (ja)
ES (1) ES469473A1 (ja)
FI (1) FI64364C (ja)
FR (1) FR2389622B1 (ja)
GB (1) GB1598872A (ja)
HK (1) HK72585A (ja)
HU (1) HU179204B (ja)
IE (1) IE46836B1 (ja)
IL (1) IL54639A (ja)
IT (1) IT1105288B (ja)
KE (1) KE3429A (ja)
LU (1) LU79575A1 (ja)
NL (1) NL186861C (ja)
NO (1) NO148747C (ja)
NZ (1) NZ187164A (ja)
PH (1) PH12831A (ja)
SE (1) SE437516B (ja)
SU (1) SU867304A3 (ja)
YU (1) YU40703B (ja)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6144294A (ja) * 1984-08-07 1986-03-03 Nippon Denso Co Ltd 熱交換器
USRE34201E (en) * 1989-04-20 1993-03-23 Anaquest, Inc. N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds
US5053411A (en) * 1989-04-20 1991-10-01 Anaquest, Inc. N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds
JPH08193074A (ja) * 1994-11-18 1996-07-30 Nippon Bayeragrochem Kk 除草性1−シクロプロピルテトラゾリノン類
JP2000327668A (ja) 1999-05-21 2000-11-28 Nippon Bayer Agrochem Co Ltd テトラゾリノン誘導体
JP2003515588A (ja) 1999-12-06 2003-05-07 マリンクロッド・インコーポレイテッド アルフェンタニル、スフェンタニルおよびレミフェンタニルの新合成法
JPWO2006030931A1 (ja) * 2004-09-14 2008-05-15 日本ケミファ株式会社 N−置換−n−(4−ピペリジニル)アミド誘導体

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3998834A (en) * 1975-03-14 1976-12-21 Janssen Pharmaceutica N.V. N-(4-piperidinyl)-n-phenylamides and -carbamates

Also Published As

Publication number Publication date
LU79575A1 (fr) 1978-11-03
PH12831A (en) 1979-09-05
ATA322078A (de) 1982-04-15
AT368994B (de) 1982-11-25
NZ187164A (en) 1981-03-16
CY1253A (en) 1984-08-31
IT1105288B (it) 1985-10-28
DK193778A (da) 1978-11-06
YU108578A (en) 1983-01-21
KE3429A (en) 1984-08-10
IE780901L (en) 1978-11-05
IT7849203A0 (it) 1978-05-04
SE437516B (sv) 1985-03-04
CA1105464A (en) 1981-07-21
IL54639A0 (en) 1978-07-31
SU867304A3 (ru) 1981-09-23
NO148747B (no) 1983-08-29
NL186861C (nl) 1991-03-18
FI781398A (fi) 1978-11-06
YU40703B (en) 1986-04-30
NL7804844A (nl) 1978-11-07
FR2389622B1 (ja) 1982-05-21
NL186861B (nl) 1990-10-16
GB1598872A (en) 1981-09-23
DE2819873C2 (ja) 1989-05-03
FI64364C (fi) 1983-11-10
HU179204B (en) 1982-09-28
JPS53149980A (en) 1978-12-27
FR2389622A1 (ja) 1978-12-01
IE46836B1 (en) 1983-10-05
AU3552278A (en) 1979-11-01
FI64364B (fi) 1983-07-29
NO148747C (no) 1983-12-07
IL54639A (en) 1982-02-28
NO781559L (no) 1978-11-07
DK152211B (da) 1988-02-08
DE2819873A1 (de) 1978-11-09
SE7805110L (sv) 1978-11-06
JPS6324995B2 (ja) 1988-05-23
ES469473A1 (es) 1979-09-16
CH635585A5 (en) 1983-04-15
AU514360B2 (en) 1981-02-05
HK72585A (en) 1985-10-04

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