DK152207C - Analogifremgangsmaade til fremstilling af sulfinylacetamid- eller malonamid-derivater eller syreadditionssalte deraf - Google Patents

Analogifremgangsmaade til fremstilling af sulfinylacetamid- eller malonamid-derivater eller syreadditionssalte deraf

Info

Publication number
DK152207C
DK152207C DK140878A DK140878A DK152207C DK 152207 C DK152207 C DK 152207C DK 140878 A DK140878 A DK 140878A DK 140878 A DK140878 A DK 140878A DK 152207 C DK152207 C DK 152207C
Authority
DK
Denmark
Prior art keywords
analogue
preparation
acid addition
addition salts
malonamide derivatives
Prior art date
Application number
DK140878A
Other languages
English (en)
Other versions
DK152207B (da
DK140878A (da
Inventor
Louis Lafon
Original Assignee
Lafon Labor
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lafon Labor filed Critical Lafon Labor
Publication of DK140878A publication Critical patent/DK140878A/da
Publication of DK152207B publication Critical patent/DK152207B/da
Application granted granted Critical
Publication of DK152207C publication Critical patent/DK152207C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C321/00—Thiols, sulfides, hydropolysulfides or polysulfides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK140878A 1977-03-31 1978-03-30 Analogifremgangsmaade til fremstilling af sulfinylacetamid- eller malonamid-derivater eller syreadditionssalte deraf DK152207C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB13579/77A GB1584462A (en) 1977-03-31 1977-03-31 N-diaryl-malonamide and diarylmethyl-sulphinyl-acetamide derivatives and pharmaceutical compositions containing them
GB1357977 1977-03-31

Publications (3)

Publication Number Publication Date
DK140878A DK140878A (da) 1978-10-01
DK152207B DK152207B (da) 1988-02-08
DK152207C true DK152207C (da) 1988-07-11

Family

ID=10025527

Family Applications (1)

Application Number Title Priority Date Filing Date
DK140878A DK152207C (da) 1977-03-31 1978-03-30 Analogifremgangsmaade til fremstilling af sulfinylacetamid- eller malonamid-derivater eller syreadditionssalte deraf

Country Status (14)

Country Link
US (1) US4177290A (da)
JP (1) JPS53121724A (da)
BE (1) BE865468A (da)
CA (1) CA1091679A (da)
CH (1) CH628026A5 (da)
DE (2) DE19875010I2 (da)
DK (1) DK152207C (da)
ES (1) ES468378A1 (da)
FR (1) FR2385693A1 (da)
GB (1) GB1584462A (da)
IE (1) IE46566B1 (da)
IT (1) IT1094041B (da)
LU (2) LU79335A1 (da)
NL (2) NL188692C (da)

Families Citing this family (101)

* Cited by examiner, † Cited by third party
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US4393026A (en) * 1980-06-19 1983-07-12 Petrolite Corporation Compounds containing sulfur and amino groups
US4616085A (en) * 1980-06-19 1986-10-07 Petrolite Corporation Thioethers of imidazolines
US4332967A (en) * 1980-06-19 1982-06-01 Petrolite Corporation Compounds containing sulfur and amino groups
US4450137A (en) * 1981-11-10 1984-05-22 Petrolite Corporation Processes for inhibiting corrosion using compounds containing sulfur and amino groups
US4450138A (en) * 1981-11-10 1984-05-22 Petrolite Corporation Processes for inhibiting corrosion using compounds containing sulfur and amino groups
US4684507A (en) * 1981-11-10 1987-08-04 Petrolite Corporation Process of corrosion inhibition using compounds containing sulfur and amino groups
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FR2528038B2 (fr) * 1982-06-04 1985-08-09 Lafon Labor Derives de benzhydrylsulfinylacetamide et leur utilisation en therapeutique
FR2528039A1 (fr) * 1982-06-04 1983-12-09 Lafon Labor Nouveaux derives de benzylsulfinylacetamide, utilisation en therapeutique et procede de preparation
FR2561646B1 (fr) * 1984-03-23 1987-10-09 Lafon Labor Derives d'acide (a-(alkylaminomethyl)-benzyl)-thioacetique, procede de preparation et utilisation en therapeutique
FR2584666B1 (fr) * 1985-07-10 1989-06-16 Champion Spark Plug Europ Bras moteur pour balai d'essuie-glace avec capuchon coulissant
FR2593809B1 (fr) * 1986-01-31 1988-07-22 Lafon Labor Benzhydrylsulfinylacetamide, procede de preparation et utilisation en therapeutique
FR2606015B1 (fr) * 1986-08-13 1989-05-19 Lafon Labor Derives du benzhydrylthiomethane, leurs procedes de preparation et leurs applications en therapeutique
FR2611709B1 (fr) * 1987-02-26 1989-06-09 Lafon Labor 2-(benzhydrylsulfonyl)acetamide, son procede de preparation et son application en therapeutique
FR2663225B1 (fr) * 1990-06-14 1994-11-04 Lafon Labor Nouvelle utilisation du modafinil.
JPH0421903U (da) * 1990-06-18 1992-02-24
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FR2697162B1 (fr) * 1992-10-23 1995-01-13 Lafon Labor Utilisation du modafinil pour la fabrication d'un médicament pour le traitement de l'incontinence urinaire et des troubles sphinctériens urétro vésicaux.
FR2706767B1 (da) * 1993-06-22 1995-09-08 Lafon Labor
FR2707637B1 (fr) * 1993-06-30 1995-10-06 Lafon Labor Nouveaux dérivés d'acétamide, leur procédé de préparation et leur utilisation en thérapeutique.
FR2708201B1 (fr) * 1993-06-30 1995-10-20 Lafon Labor Utilisation de dérivés d'acétamide pour la fabrication de médicaments.
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KR102126389B1 (ko) 2018-09-14 2020-06-25 셀라이온바이오메드 주식회사 벤즈히드릴티오 아세트아미드 화합물을 유효성분으로 포함하는 간 질환의 예방 또는 치료용 조성물
EP3863619A1 (en) 2018-10-11 2021-08-18 Novartis AG The use of a h3r inverse agonist for the treatment of excessive daytime sleepiness associated with parkinson's disease (pd)
KR102277739B1 (ko) 2019-12-11 2021-07-15 셀라이온바이오메드 주식회사 벤즈히드릴 티오 아세트아미드 화합물을 유효성분으로 포함하는 섬유화 질환의 치료용 조성물

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Also Published As

Publication number Publication date
IT1094041B (it) 1985-07-26
DK152207B (da) 1988-02-08
LU90153I2 (fr) 1998-02-16
DE2809625C2 (de) 1985-05-09
IE780433L (en) 1978-09-30
NL980003I2 (nl) 1998-05-06
DE19875010I2 (de) 2001-06-13
FR2385693A1 (fr) 1978-10-27
JPS629103B2 (da) 1987-02-26
BE865468A (fr) 1978-10-02
CH628026A5 (fr) 1982-02-15
NL7803432A (nl) 1978-10-03
CA1091679A (en) 1980-12-16
FR2385693B1 (da) 1980-04-11
JPS53121724A (en) 1978-10-24
GB1584462A (en) 1981-02-11
DE2809625A1 (de) 1978-10-05
IE46566B1 (en) 1983-07-27
ES468378A1 (es) 1978-12-16
LU79335A1 (fr) 1978-09-28
NL980003I1 (nl) 1998-03-02
NL188692C (nl) 1992-09-01
IT7821872A0 (it) 1978-03-31
DK140878A (da) 1978-10-01
US4177290A (en) 1979-12-04

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