ITMI20031298A1 - Processo di preparazione di modafinil forma polimorfa(i). - Google Patents
Processo di preparazione di modafinil forma polimorfa(i).Info
- Publication number
- ITMI20031298A1 ITMI20031298A1 IT001298A ITMI20031298A ITMI20031298A1 IT MI20031298 A1 ITMI20031298 A1 IT MI20031298A1 IT 001298 A IT001298 A IT 001298A IT MI20031298 A ITMI20031298 A IT MI20031298A IT MI20031298 A1 ITMI20031298 A1 IT MI20031298A1
- Authority
- IT
- Italy
- Prior art keywords
- preparation process
- polymorphic form
- modafinil polymorphic
- modafinil
- preparation
- Prior art date
Links
- YFGHCGITMMYXAQ-UHFFFAOYSA-N 2-[(diphenylmethyl)sulfinyl]acetamide Chemical compound C=1C=CC=CC=1C(S(=O)CC(=O)N)C1=CC=CC=C1 YFGHCGITMMYXAQ-UHFFFAOYSA-N 0.000 title 1
- 229960001165 modafinil Drugs 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
- C07C315/02—Preparation of sulfones; Preparation of sulfoxides by formation of sulfone or sulfoxide groups by oxidation of sulfides, or by formation of sulfone groups by oxidation of sulfoxides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
- C07C315/04—Preparation of sulfones; Preparation of sulfoxides by reactions not involving the formation of sulfone or sulfoxide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
- C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
- C07C319/20—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides by reactions not involving the formation of sulfide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT001298A ITMI20031298A1 (it) | 2003-06-26 | 2003-06-26 | Processo di preparazione di modafinil forma polimorfa(i). |
| PCT/EP2004/051227 WO2005000799A1 (en) | 2003-06-26 | 2004-06-24 | Process for preparing polymorphic form (i) of modafinil |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT001298A ITMI20031298A1 (it) | 2003-06-26 | 2003-06-26 | Processo di preparazione di modafinil forma polimorfa(i). |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ITMI20031298A0 ITMI20031298A0 (it) | 2003-06-26 |
| ITMI20031298A1 true ITMI20031298A1 (it) | 2004-12-27 |
Family
ID=30131297
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT001298A ITMI20031298A1 (it) | 2003-06-26 | 2003-06-26 | Processo di preparazione di modafinil forma polimorfa(i). |
Country Status (2)
| Country | Link |
|---|---|
| IT (1) | ITMI20031298A1 (it) |
| WO (1) | WO2005000799A1 (it) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20060024028A (ko) | 2000-07-27 | 2006-03-15 | 테바 파마슈티컬 인더스트리즈 리미티드 | 결정질의 순수한 모다피닐 및 이의 제조 방법 |
| US7960586B2 (en) | 2007-08-16 | 2011-06-14 | Teva Pharmaceutical Industries Ltd. | Purification of armodafinil |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1520812A (en) * | 1975-10-02 | 1978-08-09 | Lafon Labor | Benzhydrylsulphinyl derivatives |
| GB1584462A (en) * | 1977-03-31 | 1981-02-11 | Lafon Labor | N-diaryl-malonamide and diarylmethyl-sulphinyl-acetamide derivatives and pharmaceutical compositions containing them |
| FR2593809B1 (fr) * | 1986-01-31 | 1988-07-22 | Lafon Labor | Benzhydrylsulfinylacetamide, procede de preparation et utilisation en therapeutique |
| KR20060024028A (ko) * | 2000-07-27 | 2006-03-15 | 테바 파마슈티컬 인더스트리즈 리미티드 | 결정질의 순수한 모다피닐 및 이의 제조 방법 |
-
2003
- 2003-06-26 IT IT001298A patent/ITMI20031298A1/it unknown
-
2004
- 2004-06-24 WO PCT/EP2004/051227 patent/WO2005000799A1/en active Application Filing
Also Published As
| Publication number | Publication date |
|---|---|
| ITMI20031298A0 (it) | 2003-06-26 |
| WO2005000799A1 (en) | 2005-01-06 |
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