DK1483271T3 - Heterocykliske amidderivater, der har glycogenphosphorylaseinhiberende aktivetet - Google Patents

Heterocykliske amidderivater, der har glycogenphosphorylaseinhiberende aktivetet

Info

Publication number
DK1483271T3
DK1483271T3 DK03743418T DK03743418T DK1483271T3 DK 1483271 T3 DK1483271 T3 DK 1483271T3 DK 03743418 T DK03743418 T DK 03743418T DK 03743418 T DK03743418 T DK 03743418T DK 1483271 T3 DK1483271 T3 DK 1483271T3
Authority
DK
Denmark
Prior art keywords
inhibitory activity
amide derivatives
glycogen phosphorylase
heterocyclic amide
phosphorylase inhibitory
Prior art date
Application number
DK03743418T
Other languages
Danish (da)
English (en)
Inventor
Paul Robert Owen Whittamore
Stuart Norman Lile Bennett
Iain Simpson
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Application granted granted Critical
Publication of DK1483271T3 publication Critical patent/DK1483271T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK03743418T 2002-03-06 2003-03-04 Heterocykliske amidderivater, der har glycogenphosphorylaseinhiberende aktivetet DK1483271T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0205170.4A GB0205170D0 (en) 2002-03-06 2002-03-06 Chemical compounds
PCT/GB2003/000875 WO2003074531A1 (en) 2002-03-06 2003-03-04 Heterocyclic amide derivatives having glycogen phosphorylase inhibitory activity

Publications (1)

Publication Number Publication Date
DK1483271T3 true DK1483271T3 (da) 2007-02-19

Family

ID=9932334

Family Applications (1)

Application Number Title Priority Date Filing Date
DK03743418T DK1483271T3 (da) 2002-03-06 2003-03-04 Heterocykliske amidderivater, der har glycogenphosphorylaseinhiberende aktivetet

Country Status (26)

Country Link
US (1) US7122567B2 (es)
EP (1) EP1483271B1 (es)
JP (1) JP2005524669A (es)
KR (1) KR20040091101A (es)
CN (1) CN1307183C (es)
AR (1) AR038886A1 (es)
AT (1) ATE346072T1 (es)
AU (1) AU2003209445A1 (es)
BR (1) BR0308145A (es)
CA (1) CA2477125A1 (es)
DE (1) DE60309849T2 (es)
DK (1) DK1483271T3 (es)
ES (1) ES2276092T3 (es)
GB (1) GB0205170D0 (es)
HK (1) HK1070365A1 (es)
IL (1) IL163802A0 (es)
IS (1) IS7433A (es)
MX (1) MXPA04008611A (es)
NO (1) NO20044033L (es)
NZ (1) NZ534684A (es)
PL (1) PL372772A1 (es)
PT (1) PT1483271E (es)
RU (1) RU2004125145A (es)
TW (1) TW200306176A (es)
WO (1) WO2003074531A1 (es)
ZA (1) ZA200406685B (es)

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Also Published As

Publication number Publication date
IL163802A0 (en) 2005-12-18
WO2003074531A1 (en) 2003-09-12
GB0205170D0 (en) 2002-04-17
DE60309849D1 (de) 2007-01-04
DE60309849T2 (de) 2007-06-14
ZA200406685B (en) 2005-10-31
KR20040091101A (ko) 2004-10-27
PL372772A1 (en) 2005-08-08
TW200306176A (en) 2003-11-16
NO20044033L (no) 2004-11-25
PT1483271E (pt) 2007-02-28
MXPA04008611A (es) 2004-12-06
JP2005524669A (ja) 2005-08-18
EP1483271B1 (en) 2006-11-22
CN1639167A (zh) 2005-07-13
NZ534684A (en) 2006-02-24
EP1483271A1 (en) 2004-12-08
AU2003209445A1 (en) 2003-09-16
ATE346072T1 (de) 2006-12-15
US20050131052A1 (en) 2005-06-16
AR038886A1 (es) 2005-02-02
HK1070365A1 (en) 2005-06-17
ES2276092T3 (es) 2007-06-16
BR0308145A (pt) 2004-12-07
IS7433A (is) 2004-09-01
RU2004125145A (ru) 2005-06-10
CN1307183C (zh) 2007-03-28
US7122567B2 (en) 2006-10-17
CA2477125A1 (en) 2003-09-12

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