NO20053726D0 - Forbindelser med prolyloligopeptidase-hemmende aktivitet - Google Patents
Forbindelser med prolyloligopeptidase-hemmende aktivitetInfo
- Publication number
- NO20053726D0 NO20053726D0 NO20053726A NO20053726A NO20053726D0 NO 20053726 D0 NO20053726 D0 NO 20053726D0 NO 20053726 A NO20053726 A NO 20053726A NO 20053726 A NO20053726 A NO 20053726A NO 20053726 D0 NO20053726 D0 NO 20053726D0
- Authority
- NO
- Norway
- Prior art keywords
- compounds
- inhibitory activity
- prolyl oligopeptidase
- oligopeptidase inhibitory
- prolyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FI20030014A FI20030014A0 (fi) | 2003-01-03 | 2003-01-03 | Prolyylioligopeptidaasia inhiboivaa aktiivisuutta omaavia yhdisteitä |
| PCT/FI2004/000001 WO2004060862A2 (en) | 2003-01-03 | 2004-01-02 | Compounds having prolyl oligopeptidase inhibitory activity |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20053726D0 true NO20053726D0 (no) | 2005-08-03 |
| NO20053726L NO20053726L (no) | 2005-09-28 |
Family
ID=8565256
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20053726A NO20053726L (no) | 2003-01-03 | 2005-08-03 | Forbindelser med prolyloligopeptidase-hemmende aktivitet |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US20060229254A1 (no) |
| EP (1) | EP1581489A2 (no) |
| JP (1) | JP2006516557A (no) |
| KR (1) | KR20060027789A (no) |
| CN (1) | CN1747930A (no) |
| AU (1) | AU2004203788A1 (no) |
| BR (1) | BRPI0406618A (no) |
| CA (1) | CA2511856A1 (no) |
| EA (1) | EA010022B1 (no) |
| FI (1) | FI20030014A0 (no) |
| HR (1) | HRP20050693A2 (no) |
| IS (1) | IS7963A (no) |
| MX (1) | MXPA05007262A (no) |
| NO (1) | NO20053726L (no) |
| PL (1) | PL378329A1 (no) |
| RS (1) | RS20050514A (no) |
| WO (1) | WO2004060862A2 (no) |
| ZA (1) | ZA200505183B (no) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL2513053T3 (pl) | 2009-12-18 | 2018-03-30 | Ogeda Sa | Pochodne kwasu pirolidyno-karboksylowego jako agoniści receptora 43 sprzężonego z białkiem G (GPR43), kompozycja farmaceutyczna i sposoby do zastosowania w leczeniu zaburzeń metabolicznych |
| EP2730571A1 (en) | 2012-11-12 | 2014-05-14 | Universitat De Barcelona | 1-[1-(benzoyl)-pyrrolidine-2-carbonyl]-pyrrolidine-2-carbonitrile derivatives |
| EP3610872A1 (en) * | 2013-11-27 | 2020-02-19 | Epics Therapeutics | Compounds, pharmaceutical composition and methods for use in treating inflammatory diseases |
| KR101913506B1 (ko) * | 2017-07-18 | 2018-10-30 | 경상대학교산학협력단 | 프롤릴 올리고펩티다아제 억제제를 유효성분으로 함유하는 퇴행성 뇌질환 예방 또는 치료용 조성물 |
| CN117545738A (zh) | 2020-07-07 | 2024-02-09 | 安克瑞治疗公司 | 1-[1-(4-苄氧基-3,5-二氟-苯甲酰基)-4-氟-吡咯烷-2-羰基]吡咯烷-2-腈 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4483991A (en) * | 1983-01-17 | 1984-11-20 | American Home Products Corporation | Hypotensive agents |
| CA1309805C (en) * | 1985-04-16 | 1992-11-03 | Naoki Higuchi | Dipeptide derivative and synthesis and use thereof |
| JPH0696563B2 (ja) * | 1986-02-04 | 1994-11-30 | サントリー株式会社 | アシルアミノ酸誘導体、その製法並びに用途 |
| CA1320734C (en) * | 1986-02-04 | 1993-07-27 | Suntory Limited | Pyrrolidineamide derivative of acylamino acid and pharmaceutical composition containing the same |
| CA2084412C (en) * | 1990-06-04 | 2000-05-09 | W. Stephen Faraci | Pyrrolidine and thiazolidine amides |
| AU643300B2 (en) * | 1990-06-07 | 1993-11-11 | Zeria Pharmaceutical Co., Ltd. | Novel arylalkanoylamine derivative and drug containing the same |
| ES2182203T3 (es) * | 1997-10-31 | 2003-03-01 | Hoffmann La Roche | Derivados de d-prolina. |
-
2003
- 2003-01-03 FI FI20030014A patent/FI20030014A0/fi unknown
-
2004
- 2004-01-02 MX MXPA05007262A patent/MXPA05007262A/es not_active Application Discontinuation
- 2004-01-02 EA EA200501083A patent/EA010022B1/ru not_active IP Right Cessation
- 2004-01-02 WO PCT/FI2004/000001 patent/WO2004060862A2/en active Application Filing
- 2004-01-02 CA CA002511856A patent/CA2511856A1/en not_active Abandoned
- 2004-01-02 BR BR0406618-9A patent/BRPI0406618A/pt not_active IP Right Cessation
- 2004-01-02 JP JP2006500146A patent/JP2006516557A/ja active Pending
- 2004-01-02 EP EP04700047A patent/EP1581489A2/en not_active Withdrawn
- 2004-01-02 RS YUP-2005/0514A patent/RS20050514A/sr unknown
- 2004-01-02 CN CNA2004800034680A patent/CN1747930A/zh active Pending
- 2004-01-02 US US10/541,387 patent/US20060229254A1/en not_active Abandoned
- 2004-01-02 KR KR1020057012201A patent/KR20060027789A/ko not_active Application Discontinuation
- 2004-01-02 PL PL378329A patent/PL378329A1/pl unknown
- 2004-01-02 AU AU2004203788A patent/AU2004203788A1/en not_active Abandoned
-
2005
- 2005-06-27 ZA ZA200505183A patent/ZA200505183B/en unknown
- 2005-07-28 IS IS7963A patent/IS7963A/is unknown
- 2005-08-02 HR HR20050693A patent/HRP20050693A2/hr not_active Application Discontinuation
- 2005-08-03 NO NO20053726A patent/NO20053726L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| FI20030014A0 (fi) | 2003-01-03 |
| IS7963A (is) | 2005-07-28 |
| JP2006516557A (ja) | 2006-07-06 |
| ZA200505183B (en) | 2006-04-26 |
| BRPI0406618A (pt) | 2005-12-06 |
| US20060229254A1 (en) | 2006-10-12 |
| NO20053726L (no) | 2005-09-28 |
| EP1581489A2 (en) | 2005-10-05 |
| CN1747930A (zh) | 2006-03-15 |
| WO2004060862A2 (en) | 2004-07-22 |
| CA2511856A1 (en) | 2004-07-22 |
| WO2004060862A3 (en) | 2004-11-25 |
| EA200501083A1 (ru) | 2006-02-24 |
| MXPA05007262A (es) | 2005-09-08 |
| EA010022B1 (ru) | 2008-06-30 |
| PL378329A1 (pl) | 2006-03-20 |
| RS20050514A (en) | 2007-12-31 |
| AU2004203788A1 (en) | 2004-07-22 |
| KR20060027789A (ko) | 2006-03-28 |
| HRP20050693A2 (en) | 2005-10-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |