DK1440709T3 - Kombinationer, der omfatter cGMP PDE5 inhibitorer - Google Patents

Kombinationer, der omfatter cGMP PDE5 inhibitorer

Info

Publication number
DK1440709T3
DK1440709T3 DK04010436T DK04010436T DK1440709T3 DK 1440709 T3 DK1440709 T3 DK 1440709T3 DK 04010436 T DK04010436 T DK 04010436T DK 04010436 T DK04010436 T DK 04010436T DK 1440709 T3 DK1440709 T3 DK 1440709T3
Authority
DK
Denmark
Prior art keywords
combinations
pde5 inhibitors
cgmp pde5
cgmp
inhibitors
Prior art date
Application number
DK04010436T
Other languages
Danish (da)
English (en)
Inventor
Eliot Richard Forster
Nandan Parmanand Koppiker
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9924958.3A external-priority patent/GB9924958D0/en
Priority claimed from GB0021520A external-priority patent/GB0021520D0/en
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of DK1440709T3 publication Critical patent/DK1440709T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • A61K31/522Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
DK04010436T 1999-10-21 2000-10-17 Kombinationer, der omfatter cGMP PDE5 inhibitorer DK1440709T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9924958.3A GB9924958D0 (en) 1999-10-21 1999-10-21 Treatment of neuropathy
GB0021520A GB0021520D0 (en) 2000-09-01 2000-09-01 Treatment of neuropathy

Publications (1)

Publication Number Publication Date
DK1440709T3 true DK1440709T3 (da) 2008-03-17

Family

ID=26244947

Family Applications (1)

Application Number Title Priority Date Filing Date
DK04010436T DK1440709T3 (da) 1999-10-21 2000-10-17 Kombinationer, der omfatter cGMP PDE5 inhibitorer

Country Status (16)

Country Link
US (2) US20030162782A1 (fr)
EP (2) EP1129706A3 (fr)
JP (2) JP2001122803A (fr)
KR (1) KR20010051181A (fr)
AT (1) ATE380049T1 (fr)
AU (1) AU781550B2 (fr)
CA (1) CA2323839C (fr)
CO (1) CO5271711A1 (fr)
CY (1) CY1107285T1 (fr)
DE (1) DE60037347T2 (fr)
DK (1) DK1440709T3 (fr)
ES (1) ES2295726T3 (fr)
HU (1) HUP0004120A3 (fr)
IL (2) IL152925A (fr)
PE (1) PE20010754A1 (fr)
PT (1) PT1440709E (fr)

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Also Published As

Publication number Publication date
EP1440709A3 (fr) 2004-12-08
US20030162782A1 (en) 2003-08-28
JP2001122803A (ja) 2001-05-08
PE20010754A1 (es) 2001-07-18
ATE380049T1 (de) 2007-12-15
EP1129706A3 (fr) 2002-01-02
EP1440709A2 (fr) 2004-07-28
AU781550B2 (en) 2005-05-26
DE60037347T2 (de) 2008-11-27
AU6665000A (en) 2001-04-26
PT1440709E (pt) 2008-02-06
IL139073A0 (en) 2001-11-25
JP2003119131A (ja) 2003-04-23
EP1440709B1 (fr) 2007-12-05
IL152925A (en) 2010-04-15
CA2323839C (fr) 2008-03-18
HUP0004120A3 (en) 2003-11-28
CO5271711A1 (es) 2003-04-30
CY1107285T1 (el) 2012-11-21
KR20010051181A (ko) 2001-06-25
ES2295726T3 (es) 2008-04-16
HU0004120D0 (fr) 2001-01-29
US20040122010A1 (en) 2004-06-24
CA2323839A1 (fr) 2001-04-21
HUP0004120A2 (hu) 2002-11-28
EP1129706A2 (fr) 2001-09-05
DE60037347D1 (de) 2008-01-17

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