DK1427730T3 - Nye dihydropteridinoner, fremgangsmåde til fremstilling af disse og anvendelse af disse som lægemiddel - Google Patents

Nye dihydropteridinoner, fremgangsmåde til fremstilling af disse og anvendelse af disse som lægemiddel

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Publication number
DK1427730T3
DK1427730T3 DK02772249T DK02772249T DK1427730T3 DK 1427730 T3 DK1427730 T3 DK 1427730T3 DK 02772249 T DK02772249 T DK 02772249T DK 02772249 T DK02772249 T DK 02772249T DK 1427730 T3 DK1427730 T3 DK 1427730T3
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DK
Denmark
Prior art keywords
drug
processes
preparation
dihydropteridinones
new
Prior art date
Application number
DK02772249T
Other languages
Danish (da)
English (en)
Inventor
Matthias Hoffmann
Matthias Grauert
Steffen Breitfelder
Christian Eickmeier
Gerald Pohl
Gisela Schnapp
Martin Steegmaier
Eckhart Bauer
Jens Juergen Quant
Thorsten Lehmann-Lintz
Norbert Redemann
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
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Publication of DK1427730T3 publication Critical patent/DK1427730T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
DK02772249T 2001-09-04 2002-08-30 Nye dihydropteridinoner, fremgangsmåde til fremstilling af disse og anvendelse af disse som lægemiddel DK1427730T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10143272 2001-09-04

Publications (1)

Publication Number Publication Date
DK1427730T3 true DK1427730T3 (da) 2006-11-06

Family

ID=7697637

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02772249T DK1427730T3 (da) 2001-09-04 2002-08-30 Nye dihydropteridinoner, fremgangsmåde til fremstilling af disse og anvendelse af disse som lægemiddel

Country Status (30)

Country Link
EP (1) EP1427730B1 (ru)
JP (1) JP3876254B2 (ru)
KR (1) KR100955589B1 (ru)
CN (1) CN1551881A (ru)
AR (1) AR036586A1 (ru)
AT (1) ATE332898T1 (ru)
AU (1) AU2002337047B2 (ru)
BR (1) BRPI0212137A2 (ru)
CA (1) CA2458699C (ru)
CO (1) CO5560575A2 (ru)
CY (1) CY1105337T1 (ru)
DE (1) DE50207522D1 (ru)
DK (1) DK1427730T3 (ru)
EA (1) EA007062B1 (ru)
EC (1) ECSP045003A (ru)
ES (1) ES2268093T3 (ru)
HR (1) HRP20040213A2 (ru)
HU (1) HUP0401293A3 (ru)
IL (2) IL160440A0 (ru)
MX (1) MXPA04002067A (ru)
MY (1) MY129751A (ru)
NO (1) NO328804B1 (ru)
NZ (1) NZ531928A (ru)
PL (1) PL369740A1 (ru)
PT (1) PT1427730E (ru)
RS (1) RS51012B (ru)
UA (1) UA76512C2 (ru)
UY (1) UY27427A1 (ru)
WO (1) WO2003020722A1 (ru)
ZA (1) ZA200401365B (ru)

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CN111039944B (zh) * 2018-10-12 2021-11-23 中国科学院合肥物质科学研究院 Mst1激酶抑制剂及其用途
CN113637017B (zh) * 2021-08-12 2024-03-26 中国药科大学 含二氢喋呤结构的化合物及其制备方法与用途

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ATE332898T1 (de) 2006-08-15
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