DK134161B - Analogifremgangsmåde til fremstilling af steroidketoner. - Google Patents

Analogifremgangsmåde til fremstilling af steroidketoner.

Info

Publication number
DK134161B
DK134161B DK400464A DK400464A DK134161B DK 134161 B DK134161 B DK 134161B DK 400464 A DK400464 A DK 400464A DK 400464 A DK400464 A DK 400464A DK 134161 B DK134161 B DK 134161B
Authority
DK
Denmark
Prior art keywords
production
analogous method
steroid ketones
steroid
ketones
Prior art date
Application number
DK400464A
Other languages
Danish (da)
English (en)
Other versions
DK134161C (enrdf_load_stackoverflow
Inventor
Gordon Alan Hughes
Herchel Smith
Original Assignee
Herchel Smith
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to BE651797D priority Critical patent/BE651797A/xx
Priority claimed from DK448162AA external-priority patent/DK113641B/da
Priority claimed from GB3206463A external-priority patent/GB1100441A/en
Priority to GB4001667A priority patent/GB1100443A/en
Priority to GB4001767A priority patent/GB1100444A/en
Priority to IL2182664A priority patent/IL21826A/en
Priority to IN95058A priority patent/IN95058B/en
Priority to NO15427664A priority patent/NO126016B/no
Priority to DE19641468988 priority patent/DE1468988B1/de
Priority to BR16164364A priority patent/BR6461643D0/pt
Priority to DE19641793641 priority patent/DE1793641C2/de
Priority to DE19641618872 priority patent/DE1618872C3/de
Priority to DE19641618871 priority patent/DE1618871C3/de
Priority to CH1387870A priority patent/CH507225A/de
Priority to CH1742068A priority patent/CH498820A/de
Priority to CH1742168A priority patent/CH498821A/de
Priority to CH1052964A priority patent/CH498819A/de
Priority to CH381370A priority patent/CH499510A/de
Application filed by Herchel Smith filed Critical Herchel Smith
Priority to AT227470A priority patent/AT301045B/de
Priority to FR1566154D priority patent/FR1566154A/fr
Priority to DK400464A priority patent/DK134161B/da
Priority to AT292768A priority patent/AT301039B/de
Priority to AT696964A priority patent/AT269376B/de
Priority to NL6409391A priority patent/NL139307B/xx
Priority to SE983464A priority patent/SE331470B/xx
Priority to SE843170A priority patent/SE350256B/xx
Priority to FR994684A priority patent/FR4915M/fr
Priority to NO16575366A priority patent/NO127193B/no
Priority to NO16575266A priority patent/NO132762C/no
Priority to SE04238/68A priority patent/SE335120B/xx
Priority to SE04237/68A priority patent/SE335119B/xx
Priority to SE04239/68A priority patent/SE334879B/xx
Priority to DK655269A priority patent/DK127598B/da
Priority to JP5758471A priority patent/JPS4837029B1/ja
Priority to DK395771A priority patent/DK132031C/da
Priority to NO495971A priority patent/NO129905B/no
Priority to DK220272A priority patent/DK127475B/da
Priority to DK38273A priority patent/DK131020B/da
Priority to DK84773A priority patent/DK131367B/da
Priority to DK286173A priority patent/DK134264B/da
Priority to NL7308508A priority patent/NL7308508A/xx
Priority to NL737308507A priority patent/NL145559B/xx
Priority to IN1000/CAL/74A priority patent/IN137556B/en
Priority to IN1001/CAL/74A priority patent/IN137557B/en
Priority to IN137555A priority patent/IN137555B/en
Publication of DK134161B publication Critical patent/DK134161B/da
Publication of DK134161C publication Critical patent/DK134161C/da
Application granted granted Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J75/00—Processes for the preparation of steroids in general

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pressure-Spray And Ultrasonic-Wave- Spray Burners (AREA)
DK400464A 1961-10-19 1964-08-13 Analogifremgangsmåde til fremstilling af steroidketoner. DK134161B (da)

Priority Applications (43)

Application Number Priority Date Filing Date Title
BE651797D BE651797A (enrdf_load_stackoverflow) 1962-10-17
GB4001667A GB1100443A (en) 1962-10-17 1963-08-14 17ª‡-chloroethynyl-13ª‰-ethylgonenolone
GB4001767A GB1100444A (en) 1962-10-17 1963-08-14 13-alkyl 17-halogenoalkynyl steroid 3-alcohols and their esters
IL2182664A IL21826A (en) 1962-10-17 1964-08-03 Steroid ketones and their derivatives
IN95058A IN95058B (enrdf_load_stackoverflow) 1962-10-17 1964-08-05
NO15427664A NO126016B (enrdf_load_stackoverflow) 1962-10-17 1964-08-05
BR16164364A BR6461643D0 (pt) 1962-10-17 1964-08-10 Processo de preparacao de cetonas esteroides e seus derivados
DE19641618871 DE1618871C3 (de) 1962-10-17 1964-08-10 Verfahren zur Herstellung eines Steroidketonderivates. Ausscheidung aus: 1468988
DE19641793641 DE1793641C2 (de) 1962-10-17 1964-08-10 Verfahren zur Herstellung von 17-Halogenalkinyl 3-ketogonen und deren Verwendung. Ausscheidung aus: 1468988
DE19641618872 DE1618872C3 (de) 1962-10-17 1964-08-10 Verfahren zur Herstellung von 13-Äthylgonanverbindungen und gewisse 13-Äthylgonanverbindungen. Ausscheidung aus: 1468988
DE19641468988 DE1468988B1 (de) 1962-10-17 1964-08-10 17alpha-Chloraethinyl-13beta-aethyl-4- oder -5(10)-gonen-3-ketone
CH1387870A CH507225A (de) 1962-10-17 1964-08-12 Verfahren zur Herstellung von Steroidketonen mit 17- oder 17a-Halogenalkinylgruppen
CH1742068A CH498820A (de) 1961-10-19 1964-08-12 Verfahren zur Herstellung von Steroidketonderivaten mit 17- oder 17a-Halogenalkinylgruppen
CH1742168A CH498821A (de) 1962-10-17 1964-08-12 Verfahren zur Herstellung von Steroidketonderivaten mit 17- und 17a-Halogenalkinylgruppen
CH1052964A CH498819A (de) 1962-10-17 1964-08-12 Verfahren zur Herstellung von Steroidketonen mit 17- oder 17a-Halogenalkinylgruppen
CH381370A CH499510A (de) 1962-10-17 1964-08-12 Verfahren zur Herstellung von Steroidketonderivaten mit 17-oder 17a-Halogenalkinylgruppen
AT696964A AT269376B (de) 1962-10-17 1964-08-13 Verfahren zur Herstellung von neuen Steroidketonen
AT227470A AT301045B (de) 1962-10-17 1964-08-13 Verfahren zur Herstellung von neuen Steroiden
FR1566154D FR1566154A (enrdf_load_stackoverflow) 1962-10-17 1964-08-13
DK400464A DK134161B (da) 1962-10-17 1964-08-13 Analogifremgangsmåde til fremstilling af steroidketoner.
AT292768A AT301039B (de) 1962-10-17 1964-08-13 Verfahren zur Herstellung von neuen Steroiden
SE983464A SE331470B (enrdf_load_stackoverflow) 1962-10-17 1964-08-14
NL6409391A NL139307B (nl) 1962-10-17 1964-08-14 Werkwijze voor het bereiden van een geneesmiddel met een hormoonactiviteit.
SE843170A SE350256B (enrdf_load_stackoverflow) 1962-10-17 1964-08-14
FR994684A FR4915M (enrdf_load_stackoverflow) 1962-10-17 1964-11-12
NO16575366A NO127193B (enrdf_load_stackoverflow) 1962-10-17 1966-11-25
NO16575266A NO132762C (enrdf_load_stackoverflow) 1962-10-17 1966-11-25
SE04239/68A SE334879B (enrdf_load_stackoverflow) 1962-10-17 1968-03-29
SE04237/68A SE335119B (enrdf_load_stackoverflow) 1962-10-17 1968-03-29
SE04238/68A SE335120B (enrdf_load_stackoverflow) 1962-10-17 1968-03-29
DK655269A DK127598B (da) 1962-10-17 1969-12-10 Analogifremgangsmåde til fremstilling af 17-halogenalkynyl-3,17-dihydroxy-13-ethylgonener eller -D-homogener eller estere eller ethere deraf.
JP5758471A JPS4837029B1 (enrdf_load_stackoverflow) 1962-10-17 1971-08-02
DK395771A DK132031C (da) 1962-10-17 1971-08-12 Analogifremgangsmade til fremstilling af 17-haloalkynyl-17-hydroxy-13-ethyl-gonen-3-oner eller de tilsvarende d-homo-forbindelser
NO495971A NO129905B (enrdf_load_stackoverflow) 1962-10-17 1971-12-30
DK220272A DK127475B (da) 1962-10-17 1972-05-03 Analogifremgangsmåde til fremstilling af17-halogenalkynyl-17-hydroxy-13-ethylgonener eller -D-homogonener eller estere eller ethere deraf.
DK38273A DK131020B (da) 1962-10-17 1973-01-24 Antikonceptionelt middel.
DK84773A DK131367B (da) 1962-10-17 1973-02-16 Antikonceptionelt middel.
DK286173A DK134264B (da) 1962-10-17 1973-05-24 Antikonceptionelt middel.
NL7308508A NL7308508A (enrdf_load_stackoverflow) 1962-10-17 1973-06-19
NL737308507A NL145559B (nl) 1962-10-17 1973-06-19 Werkwijze voor het bereiden van een preparaat met progestatieve en anti-oestrogene activiteit, gevormd geneesmiddel en werkwijze voor het bereiden van progestatieve en anti-oestrogeen actieve verbindingen.
IN1000/CAL/74A IN137556B (enrdf_load_stackoverflow) 1962-10-17 1974-05-03
IN1001/CAL/74A IN137557B (enrdf_load_stackoverflow) 1962-10-17 1974-05-03
IN137555A IN137555B (enrdf_load_stackoverflow) 1962-10-17 1974-05-03

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DK448162AA DK113641B (da) 1961-10-19 1962-10-17 Fremgangsmåde til fremstilling af steroidketoner.
GB3206463A GB1100441A (en) 1963-08-14 1963-08-14 13-alkyl 17-halogenoalkynyl-steroid 3-ketones and their derivatives
DK400464A DK134161B (da) 1962-10-17 1964-08-13 Analogifremgangsmåde til fremstilling af steroidketoner.

Publications (2)

Publication Number Publication Date
DK134161B true DK134161B (da) 1976-09-20
DK134161C DK134161C (enrdf_load_stackoverflow) 1977-02-21

Family

ID=27221920

Family Applications (3)

Application Number Title Priority Date Filing Date
DK400464A DK134161B (da) 1961-10-19 1964-08-13 Analogifremgangsmåde til fremstilling af steroidketoner.
DK655269A DK127598B (da) 1962-10-17 1969-12-10 Analogifremgangsmåde til fremstilling af 17-halogenalkynyl-3,17-dihydroxy-13-ethylgonener eller -D-homogener eller estere eller ethere deraf.
DK220272A DK127475B (da) 1962-10-17 1972-05-03 Analogifremgangsmåde til fremstilling af17-halogenalkynyl-17-hydroxy-13-ethylgonener eller -D-homogonener eller estere eller ethere deraf.

Family Applications After (2)

Application Number Title Priority Date Filing Date
DK655269A DK127598B (da) 1962-10-17 1969-12-10 Analogifremgangsmåde til fremstilling af 17-halogenalkynyl-3,17-dihydroxy-13-ethylgonener eller -D-homogener eller estere eller ethere deraf.
DK220272A DK127475B (da) 1962-10-17 1972-05-03 Analogifremgangsmåde til fremstilling af17-halogenalkynyl-17-hydroxy-13-ethylgonener eller -D-homogonener eller estere eller ethere deraf.

Country Status (14)

Country Link
JP (1) JPS4837029B1 (enrdf_load_stackoverflow)
AT (3) AT301039B (enrdf_load_stackoverflow)
BE (1) BE651797A (enrdf_load_stackoverflow)
BR (1) BR6461643D0 (enrdf_load_stackoverflow)
CH (1) CH498819A (enrdf_load_stackoverflow)
DE (4) DE1618872C3 (enrdf_load_stackoverflow)
DK (3) DK134161B (enrdf_load_stackoverflow)
FR (2) FR1566154A (enrdf_load_stackoverflow)
GB (2) GB1100443A (enrdf_load_stackoverflow)
IL (1) IL21826A (enrdf_load_stackoverflow)
IN (2) IN95058B (enrdf_load_stackoverflow)
NL (2) NL139307B (enrdf_load_stackoverflow)
NO (3) NO126016B (enrdf_load_stackoverflow)
SE (5) SE331470B (enrdf_load_stackoverflow)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2913381A1 (de) * 1979-03-30 1980-10-16 Schering Ag 11-methylensteroide, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
JPS57106714U (enrdf_load_stackoverflow) * 1980-12-23 1982-07-01
DE3214689A1 (de) * 1982-04-16 1983-10-27 Schering AG, 1000 Berlin und 4709 Bergkamen 11ss-chlor-steroide, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
JP2014505721A (ja) * 2011-02-17 2014-03-06 ルピン・リミテッド レボノルゲストレルを調製するための改良された方法

Also Published As

Publication number Publication date
DE1618872A1 (de) 1972-06-15
AT301039B (de) 1972-08-25
BE651797A (enrdf_load_stackoverflow)
IL21826A (en) 1968-12-26
DE1618872B2 (de) 1974-03-07
DE1618871A1 (de) 1972-08-10
DE1618871B2 (de) 1973-07-26
SE335119B (enrdf_load_stackoverflow) 1971-05-17
NO129905B (enrdf_load_stackoverflow) 1974-06-10
IN95058B (enrdf_load_stackoverflow) 1975-08-16
AT301045B (de) 1972-08-25
DE1618872C3 (de) 1974-10-24
GB1100444A (en) 1968-01-24
DE1793641C2 (de) 1973-12-20
NO126016B (enrdf_load_stackoverflow) 1972-12-11
IN137555B (enrdf_load_stackoverflow) 1975-08-16
GB1100443A (en) 1968-01-24
NL139307B (nl) 1973-07-16
DK127475B (da) 1973-11-12
DK134161C (enrdf_load_stackoverflow) 1977-02-21
SE335120B (enrdf_load_stackoverflow) 1971-05-17
AT269376B (de) 1969-03-10
NL6409391A (enrdf_load_stackoverflow) 1965-02-15
DK127598B (da) 1973-12-03
BR6461643D0 (pt) 1973-08-09
FR4915M (enrdf_load_stackoverflow) 1967-03-20
CH498819A (de) 1970-11-15
SE350256B (enrdf_load_stackoverflow) 1972-10-23
DE1468988B1 (de) 1971-11-25
NO127193B (enrdf_load_stackoverflow) 1973-05-21
DE1618871C3 (de) 1974-02-21
SE331470B (enrdf_load_stackoverflow) 1971-01-04
FR1566154A (enrdf_load_stackoverflow) 1969-05-09
SE334879B (enrdf_load_stackoverflow) 1971-05-10
DE1793641B1 (de) 1973-05-24
NL7308508A (enrdf_load_stackoverflow) 1973-09-25
JPS4837029B1 (enrdf_load_stackoverflow) 1973-11-08

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