DK1299389T3 - Fremgangsmåde til fremstilling af pyrazolpyrimidinonderivater til behandling af impotens - Google Patents

Fremgangsmåde til fremstilling af pyrazolpyrimidinonderivater til behandling af impotens

Info

Publication number
DK1299389T3
DK1299389T3 DK01932366T DK01932366T DK1299389T3 DK 1299389 T3 DK1299389 T3 DK 1299389T3 DK 01932366 T DK01932366 T DK 01932366T DK 01932366 T DK01932366 T DK 01932366T DK 1299389 T3 DK1299389 T3 DK 1299389T3
Authority
DK
Denmark
Prior art keywords
compound
impotence
treatment
pyrazole
preparation
Prior art date
Application number
DK01932366T
Other languages
English (en)
Inventor
Moo-Hi Yoo
Won-Bae Kim
Min-Sun Chang
Soon-Hoe Kim
Dong-Sung Kim
Chul-Jun Bae
Yong-Duck Kim
Eun-Ha Kim
Original Assignee
Dong A Pharm Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dong A Pharm Co Ltd filed Critical Dong A Pharm Co Ltd
Application granted granted Critical
Publication of DK1299389T3 publication Critical patent/DK1299389T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK01932366T 2000-06-23 2001-05-18 Fremgangsmåde til fremstilling af pyrazolpyrimidinonderivater til behandling af impotens DK1299389T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR10-2000-0034966A KR100377782B1 (ko) 2000-06-23 2000-06-23 발기부전 치료에 효과를 갖는 피라졸로피리미디논화합물의 제조방법
PCT/KR2001/000819 WO2001098304A1 (en) 2000-06-23 2001-05-18 A process for preparing pyrazolopyrimidinone derivatives for the treatment of impotence

Publications (1)

Publication Number Publication Date
DK1299389T3 true DK1299389T3 (da) 2007-02-05

Family

ID=36087864

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01932366T DK1299389T3 (da) 2000-06-23 2001-05-18 Fremgangsmåde til fremstilling af pyrazolpyrimidinonderivater til behandling af impotens

Country Status (19)

Country Link
US (1) US6844436B2 (da)
EP (1) EP1299389B1 (da)
JP (1) JP3939646B2 (da)
KR (1) KR100377782B1 (da)
CN (1) CN1217946C (da)
AT (1) ATE341549T1 (da)
AU (2) AU2001258896B2 (da)
BR (1) BRPI0111793B8 (da)
CA (1) CA2413761C (da)
CY (1) CY1105769T1 (da)
DE (1) DE60123616T2 (da)
DK (1) DK1299389T3 (da)
ES (1) ES2272475T3 (da)
HK (1) HK1055732A1 (da)
MX (1) MXPA02012420A (da)
NZ (1) NZ523238A (da)
PT (1) PT1299389E (da)
RU (1) RU2236410C2 (da)
WO (1) WO2001098304A1 (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100377782B1 (ko) * 2000-06-23 2003-03-29 동아제약 주식회사 발기부전 치료에 효과를 갖는 피라졸로피리미디논화합물의 제조방법
CN100374441C (zh) 2003-06-06 2008-03-12 天津倍方科技发展有限公司 二氢吡咯[2，3-d]嘧啶-4-酮衍生物，其制备方法及其制药用途
EP1888074B1 (en) 2005-06-10 2011-12-21 Dong-A Pharmaceutical Co., Ltd. Agent for the prevention and treatment of liver diseases containing pyrazolopyrimidine derivative
KR100963644B1 (ko) 2007-11-23 2010-06-15 한국과학기술연구원 피라졸로피리미딘온 유도체 및 그의 제조방법
WO2022123310A1 (en) 2020-12-11 2022-06-16 Ildong Pharmaceutical Co., Ltd. Novel compounds as androgen receptor and phosphodiesterase dual inhibitor

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9013750D0 (en) 1990-06-20 1990-08-08 Pfizer Ltd Therapeutic agents
GB9119704D0 (en) 1991-09-14 1991-10-30 Pfizer Ltd Therapeutic agents
NZ338075A (en) * 1997-04-25 2000-10-27 Pfizer Ltd Pyrazolopyrimidinones which inhibit type 5 cyclic guanosine 3',5'-monophosphate phosphodiesterase (cGMP PED5) for the treatment of sexual dysfunction
GB9708831D0 (en) 1997-04-30 1997-06-25 Unilever Plc Suspensions with high storage stability, comprising an aqueous silicate solution and filler material
DK1109814T3 (da) * 1998-09-04 2004-08-02 Ortho Mcneil Pharm Inc 5-Heterocyclylpyrazolo[4,3-d]pyrimidin-7-oner til behandling af mandlig erektil dysfunktion
KR100353014B1 (ko) * 1998-11-11 2002-09-18 동아제약 주식회사 발기부전 치료에 효과를 갖는 피라졸로피리미디논 화합물
EP1002798A1 (en) * 1998-11-20 2000-05-24 Orchid Chemicals & Pharmaceuticals Ltd. An improved process for preparing a therapeutically active pyrazolopyrimidinone derivative
KR100377782B1 (ko) * 2000-06-23 2003-03-29 동아제약 주식회사 발기부전 치료에 효과를 갖는 피라졸로피리미디논화합물의 제조방법

Also Published As

Publication number Publication date
AU2001258896B2 (en) 2005-12-08
AU5889601A (en) 2002-01-02
CA2413761C (en) 2007-09-04
DE60123616T2 (de) 2007-01-18
JP3939646B2 (ja) 2007-07-04
RU2236410C2 (ru) 2004-09-20
KR100377782B1 (ko) 2003-03-29
CN1441802A (zh) 2003-09-10
BR0111793A (pt) 2003-05-27
US6844436B2 (en) 2005-01-18
PT1299389E (pt) 2006-12-29
HK1055732A1 (en) 2004-01-21
MXPA02012420A (es) 2004-02-26
BRPI0111793B1 (pt) 2019-07-16
EP1299389A1 (en) 2003-04-09
BRPI0111793B8 (pt) 2021-05-25
JP2004501155A (ja) 2004-01-15
US20030176696A1 (en) 2003-09-18
EP1299389A4 (en) 2005-02-02
CY1105769T1 (el) 2011-02-02
CA2413761A1 (en) 2001-12-27
DE60123616D1 (de) 2006-11-16
NZ523238A (en) 2003-11-28
WO2001098304A1 (en) 2001-12-27
EP1299389B1 (en) 2006-10-04
ATE341549T1 (de) 2006-10-15
KR20020001041A (ko) 2002-01-09
CN1217946C (zh) 2005-09-07
ES2272475T3 (es) 2007-05-01

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