DK1283838T3 - Piperazin- og piperidinforbindelser - Google Patents

Piperazin- og piperidinforbindelser

Info

Publication number
DK1283838T3
DK1283838T3 DK01938214T DK01938214T DK1283838T3 DK 1283838 T3 DK1283838 T3 DK 1283838T3 DK 01938214 T DK01938214 T DK 01938214T DK 01938214 T DK01938214 T DK 01938214T DK 1283838 T3 DK1283838 T3 DK 1283838T3
Authority
DK
Denmark
Prior art keywords
piperazine
piperidine compounds
piperidine
compounds
Prior art date
Application number
DK01938214T
Other languages
Danish (da)
English (en)
Inventor
Stephen K Long
Roelof W Feenstra
Der Heijden Johannes A M Van
Cornelis G Kruse
Scharrenburg Gustaaf J M Van
Original Assignee
Solvay Pharm Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharm Bv filed Critical Solvay Pharm Bv
Application granted granted Critical
Publication of DK1283838T3 publication Critical patent/DK1283838T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Hydrogenated Pyridines (AREA)
DK01938214T 2000-05-12 2001-05-10 Piperazin- og piperidinforbindelser DK1283838T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00201699 2000-05-12
PCT/EP2001/005320 WO2001085725A1 (en) 2000-05-12 2001-05-10 Piperazine and piperidine compounds

Publications (1)

Publication Number Publication Date
DK1283838T3 true DK1283838T3 (da) 2004-03-22

Family

ID=8171488

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01938214T DK1283838T3 (da) 2000-05-12 2001-05-10 Piperazin- og piperidinforbindelser

Country Status (27)

Country Link
US (2) US6911448B2 (cs)
EP (1) EP1283838B1 (cs)
JP (1) JP2003532729A (cs)
CN (1) CN1174979C (cs)
AR (1) AR028443A1 (cs)
AT (1) ATE255578T1 (cs)
AU (2) AU2001263927B2 (cs)
BR (1) BR0110592A (cs)
CA (1) CA2405971C (cs)
CZ (1) CZ301464B6 (cs)
DE (1) DE60101386T2 (cs)
DK (1) DK1283838T3 (cs)
DZ (1) DZ3370A1 (cs)
ES (1) ES2211809T3 (cs)
HU (1) HUP0302016A2 (cs)
IL (2) IL152177A0 (cs)
MX (1) MXPA02011084A (cs)
NO (1) NO323778B1 (cs)
NZ (1) NZ522116A (cs)
PL (1) PL198857B1 (cs)
PT (1) PT1283838E (cs)
RU (1) RU2261250C2 (cs)
SK (1) SK286778B6 (cs)
TR (1) TR200302294T4 (cs)
UA (1) UA72337C2 (cs)
WO (1) WO2001085725A1 (cs)
ZA (1) ZA200208537B (cs)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2211809T3 (es) * 2000-05-12 2004-07-16 Solvay Pharmaceuticals B.V. Compuesto de piperazina y piperidina.
ATE424825T1 (de) 2001-07-20 2009-03-15 Psychogenics Inc Behandlung von hyperaktivitätsstörungen und aufmerksamkeitsdefiziten
WO2004000837A1 (ja) * 2002-06-25 2003-12-31 Sumitomo Pharmaceuticals Co., Ltd. 新規なベンズオキサゾリノン誘導体
ES2232292B1 (es) * 2003-07-30 2006-11-01 Laboratorios Del Dr. Esteve, S.A. Compuestos sulfonamidicos derivados de benzoxazinona, su preparacion y uso como medicamentos.
US7596407B2 (en) 2004-03-26 2009-09-29 Solvay Pharmaceuticals, B.V. Transdermal iontophoretic delivery of piperazinyl-2(3H)-benzoxazolone compounds
EP1595542A1 (en) * 2004-03-26 2005-11-16 Solvay Pharmaceuticals B.V. Transdermal iontophoretic delivery of piperazinyl-2(3H)-benzoxazolone compounds
RU2394821C2 (ru) * 2005-08-22 2010-07-20 Солвей Фармасьютикал Б.В. N-оксиды как пролекарства производных пиперазина и пиперидина
AR058022A1 (es) * 2005-08-22 2008-01-23 Solvay Pharm Bv Derivados de benzooxazoles, composiciones farmaceuticas y su uso para el tratamiento de desordenes del sistema nervioso.
US7750013B2 (en) 2005-08-22 2010-07-06 Solvay Pharmaceuticals, B.V. N-oxides as prodrugs of piperazine and piperidine derivatives
US20070275977A1 (en) * 2006-05-02 2007-11-29 Van Aar Marcel P N-oxides of pyridylmethyl -piperazine and -piperidine derivatives
US8106056B2 (en) 2006-06-16 2012-01-31 Solvay Pharmaceuticals B.V. Combination preparations comprising bifeprunox and a dopamine agonist
KR101050568B1 (ko) 2006-12-07 2011-07-19 에프. 호프만-라 로슈 아게 V1a 수용체 길항제로서의 스피로-피페리딘 유도체
MX2009005507A (es) 2006-12-07 2009-06-03 Hoffmann La Roche Derivados de espiro-piperidina.
MX2009005544A (es) 2006-12-08 2009-06-05 Hoffmann La Roche Indoles.
DE602007007512D1 (de) 2006-12-08 2010-08-12 Hoffmann La Roche Als via-rezeptor-antagonisten verwendbare indole
US8084609B2 (en) 2006-12-22 2011-12-27 Hoffman-La Roche Inc. Spiropiperidine derivatives
CA2711520A1 (en) * 2008-01-15 2009-07-23 Abbott Healthcare Products B.V. Bifeprunox derivatives
RU2764716C2 (ru) 2016-08-26 2022-01-19 Экссива Уг (Хафтунгзбешрэнкт) Композиции и связанные с ними способы
SG11202100680WA (en) * 2018-07-27 2021-02-25 Chugoku Marine Paints Antifouling paint composition, antifouling coating, substrate with antifouling coating, production method thereof, and repair method

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS60126275A (ja) * 1983-12-13 1985-07-05 Otsuka Pharmaceut Co Ltd ベンゾチアゾ−ル誘導体
FR2567884B1 (fr) 1984-07-19 1987-03-06 Roussel Uclaf Nouveaux derives de l'indole, leur preparation, leur application comme medicaments et les compositions les renfermant
EP0189612B1 (en) * 1984-12-21 1992-11-04 Duphar International Research B.V New pharmaceutical compositions having a psychotropic activity
EP0185429A1 (en) 1984-12-21 1986-06-25 Duphar International Research B.V New bicyclic heteroaryl piperazines
DE4127849A1 (de) * 1991-08-22 1993-02-25 Merck Patent Gmbh Benzodioxanderivate
NZ331860A (en) * 1996-03-29 2000-04-28 Duphar Int Res Piperazine and piperidine compounds with affinity for both dopamine D2 and seratonin 5-HT1A receptors
TW530054B (en) * 1997-09-24 2003-05-01 Duphar Int Res New piperazine and piperidine compounds
GB9811879D0 (en) * 1998-06-03 1998-07-29 Knoll Ag Therapeutic agents
UA71590C2 (en) * 1998-11-13 2004-12-15 Duphar Int Res Piperazine and piperidine derivatives
EP1284731A1 (en) * 2000-05-12 2003-02-26 Solvay Pharmaceuticals B.V. Use of compounds having combined dopamine d2, 5-ht1a and alpha adrenoreceptor agonistic action for treating cns disorders
ES2211809T3 (es) * 2000-05-12 2004-07-16 Solvay Pharmaceuticals B.V. Compuesto de piperazina y piperidina.

Also Published As

Publication number Publication date
US20060089366A1 (en) 2006-04-27
CA2405971A1 (en) 2001-11-15
DZ3370A1 (fr) 2001-11-15
WO2001085725A1 (en) 2001-11-15
NO20025365L (no) 2002-11-08
IL152177A (en) 2009-08-03
RU2261250C2 (ru) 2005-09-27
HK1055952A1 (en) 2004-01-30
NO323778B1 (no) 2007-07-02
PL198857B1 (pl) 2008-07-31
UA72337C2 (uk) 2005-02-15
AU2001263927B2 (en) 2004-09-30
CZ301464B6 (cs) 2010-03-10
PT1283838E (pt) 2004-04-30
PL358201A1 (en) 2004-08-09
CN1174979C (zh) 2004-11-10
US20030119849A1 (en) 2003-06-26
TR200302294T4 (tr) 2004-02-23
IL152177A0 (en) 2003-05-29
AU6392701A (en) 2001-11-20
DE60101386T2 (de) 2004-05-27
US6911448B2 (en) 2005-06-28
AR028443A1 (es) 2003-05-07
BR0110592A (pt) 2003-04-01
ZA200208537B (en) 2004-01-22
SK15872002A3 (sk) 2003-04-01
CA2405971C (en) 2010-03-30
DE60101386D1 (de) 2004-01-15
MXPA02011084A (es) 2003-03-10
CN1429226A (zh) 2003-07-09
HUP0302016A2 (hu) 2003-09-29
NZ522116A (en) 2004-04-30
SK286778B6 (sk) 2009-05-07
US7297699B2 (en) 2007-11-20
NO20025365D0 (no) 2002-11-08
ES2211809T3 (es) 2004-07-16
JP2003532729A (ja) 2003-11-05
ATE255578T1 (de) 2003-12-15
EP1283838A1 (en) 2003-02-19
CZ20023721A3 (cs) 2003-02-12
EP1283838B1 (en) 2003-12-03

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