DK1283838T3 - Piperazin- og piperidinforbindelser - Google Patents

Piperazin- og piperidinforbindelser

Info

Publication number
DK1283838T3
DK1283838T3 DK01938214T DK01938214T DK1283838T3 DK 1283838 T3 DK1283838 T3 DK 1283838T3 DK 01938214 T DK01938214 T DK 01938214T DK 01938214 T DK01938214 T DK 01938214T DK 1283838 T3 DK1283838 T3 DK 1283838T3
Authority
DK
Denmark
Prior art keywords
piperazine
piperidine compounds
piperidine
compounds
Prior art date
Application number
DK01938214T
Other languages
Danish (da)
English (en)
Inventor
Stephen K Long
Roelof W Feenstra
Der Heijden Johannes A M Van
Cornelis G Kruse
Scharrenburg Gustaaf J M Van
Original Assignee
Solvay Pharm Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharm Bv filed Critical Solvay Pharm Bv
Application granted granted Critical
Publication of DK1283838T3 publication Critical patent/DK1283838T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurosurgery (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Addiction (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
DK01938214T 2000-05-12 2001-05-10 Piperazin- og piperidinforbindelser DK1283838T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00201699 2000-05-12
PCT/EP2001/005320 WO2001085725A1 (en) 2000-05-12 2001-05-10 Piperazine and piperidine compounds

Publications (1)

Publication Number Publication Date
DK1283838T3 true DK1283838T3 (da) 2004-03-22

Family

ID=8171488

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01938214T DK1283838T3 (da) 2000-05-12 2001-05-10 Piperazin- og piperidinforbindelser

Country Status (27)

Country Link
US (2) US6911448B2 (cs)
EP (1) EP1283838B1 (cs)
JP (1) JP2003532729A (cs)
CN (1) CN1174979C (cs)
AR (1) AR028443A1 (cs)
AT (1) ATE255578T1 (cs)
AU (2) AU2001263927B2 (cs)
BR (1) BR0110592A (cs)
CA (1) CA2405971C (cs)
CZ (1) CZ301464B6 (cs)
DE (1) DE60101386T2 (cs)
DK (1) DK1283838T3 (cs)
DZ (1) DZ3370A1 (cs)
ES (1) ES2211809T3 (cs)
HU (1) HUP0302016A2 (cs)
IL (2) IL152177A0 (cs)
MX (1) MXPA02011084A (cs)
NO (1) NO323778B1 (cs)
NZ (1) NZ522116A (cs)
PL (1) PL198857B1 (cs)
PT (1) PT1283838E (cs)
RU (1) RU2261250C2 (cs)
SK (1) SK286778B6 (cs)
TR (1) TR200302294T4 (cs)
UA (1) UA72337C2 (cs)
WO (1) WO2001085725A1 (cs)
ZA (1) ZA200208537B (cs)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL152177A0 (en) * 2000-05-12 2003-05-29 Solvay Pharm Bv Piperazine and piperidine compounds
DK1408976T5 (da) 2001-07-20 2011-01-10 Psychogenics Inc Behandling af ADHD (Attention deficit hyperactivity disorder)
WO2004000837A1 (ja) * 2002-06-25 2003-12-31 Sumitomo Pharmaceuticals Co., Ltd. 新規なベンズオキサゾリノン誘導体
ES2232292B1 (es) * 2003-07-30 2006-11-01 Laboratorios Del Dr. Esteve, S.A. Compuestos sulfonamidicos derivados de benzoxazinona, su preparacion y uso como medicamentos.
EP1595542A1 (en) * 2004-03-26 2005-11-16 Solvay Pharmaceuticals B.V. Transdermal iontophoretic delivery of piperazinyl-2(3H)-benzoxazolone compounds
US7596407B2 (en) 2004-03-26 2009-09-29 Solvay Pharmaceuticals, B.V. Transdermal iontophoretic delivery of piperazinyl-2(3H)-benzoxazolone compounds
AR058022A1 (es) * 2005-08-22 2008-01-23 Solvay Pharm Bv Derivados de benzooxazoles, composiciones farmaceuticas y su uso para el tratamiento de desordenes del sistema nervioso.
US7750013B2 (en) 2005-08-22 2010-07-06 Solvay Pharmaceuticals, B.V. N-oxides as prodrugs of piperazine and piperidine derivatives
ATE417834T1 (de) * 2005-08-22 2009-01-15 Solvay Pharm Bv N-oxide als prodrugs von piperazin- und piperidinderivaten
US20070275977A1 (en) * 2006-05-02 2007-11-29 Van Aar Marcel P N-oxides of pyridylmethyl -piperazine and -piperidine derivatives
US8106056B2 (en) 2006-06-16 2012-01-31 Solvay Pharmaceuticals B.V. Combination preparations comprising bifeprunox and a dopamine agonist
CN101547923A (zh) 2006-12-07 2009-09-30 弗·哈夫曼-拉罗切有限公司 作为via受体拮抗剂的螺环-哌啶衍生物
CN101541797A (zh) 2006-12-07 2009-09-23 弗·哈夫曼-拉罗切有限公司 螺-哌啶衍生物
WO2008068184A1 (en) 2006-12-08 2008-06-12 F. Hoffmann-La Roche Ag Indoles which act as via receptor antagonists
KR20090078367A (ko) 2006-12-08 2009-07-17 에프. 호프만-라 로슈 아게 인돌
EP2097376A2 (en) 2006-12-22 2009-09-09 F. Hoffmann-Roche AG Spiro-piperidine derivatives
CN101918382A (zh) * 2008-01-15 2010-12-15 雅培卫生保健产品有限责任公司 联苯芦诺衍生物
BR112019003811A2 (pt) 2016-08-26 2019-05-21 Exciva Ug (Haftungsbeschränkt) composição farmacêutica, método para aumentar os níveis plasmáticos de antagonista do receptor de nmda em um sujeito que precisa do mesmo, método para tratar uma doença ou transtorno em um sujeito que precisa do mesmo e uso da composição
CN112513207B (zh) * 2018-07-27 2022-06-17 中国涂料株式会社 防污涂料组合物、防污涂膜、带有防污涂膜的基材及其制造方法以及修补方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS60126275A (ja) * 1983-12-13 1985-07-05 Otsuka Pharmaceut Co Ltd ベンゾチアゾ−ル誘導体
FR2567884B1 (fr) 1984-07-19 1987-03-06 Roussel Uclaf Nouveaux derives de l'indole, leur preparation, leur application comme medicaments et les compositions les renfermant
EP0189612B1 (en) * 1984-12-21 1992-11-04 Duphar International Research B.V New pharmaceutical compositions having a psychotropic activity
ATE44528T1 (de) 1984-12-21 1989-07-15 Duphar Int Res Arzneimittel mit antipsychotischer wirkung.
DE4127849A1 (de) * 1991-08-22 1993-02-25 Merck Patent Gmbh Benzodioxanderivate
RU2178414C2 (ru) 1996-03-29 2002-01-20 Дюфар Интернэшнл Рисерч Б.В. Производные пиперазина и пиперидина и способ их получения
TW530054B (en) * 1997-09-24 2003-05-01 Duphar Int Res New piperazine and piperidine compounds
GB9811879D0 (en) * 1998-06-03 1998-07-29 Knoll Ag Therapeutic agents
UA71590C2 (en) * 1998-11-13 2004-12-15 Duphar Int Res Piperazine and piperidine derivatives
IL152177A0 (en) * 2000-05-12 2003-05-29 Solvay Pharm Bv Piperazine and piperidine compounds
EP1284731A1 (en) * 2000-05-12 2003-02-26 Solvay Pharmaceuticals B.V. Use of compounds having combined dopamine d2, 5-ht1a and alpha adrenoreceptor agonistic action for treating cns disorders

Also Published As

Publication number Publication date
EP1283838B1 (en) 2003-12-03
US7297699B2 (en) 2007-11-20
ZA200208537B (en) 2004-01-22
EP1283838A1 (en) 2003-02-19
PL198857B1 (pl) 2008-07-31
AR028443A1 (es) 2003-05-07
DZ3370A1 (fr) 2001-11-15
CN1429226A (zh) 2003-07-09
MXPA02011084A (es) 2003-03-10
ATE255578T1 (de) 2003-12-15
NO20025365D0 (no) 2002-11-08
SK15872002A3 (sk) 2003-04-01
SK286778B6 (sk) 2009-05-07
IL152177A (en) 2009-08-03
NO20025365L (no) 2002-11-08
NO323778B1 (no) 2007-07-02
RU2261250C2 (ru) 2005-09-27
ES2211809T3 (es) 2004-07-16
NZ522116A (en) 2004-04-30
HK1055952A1 (en) 2004-01-30
AU6392701A (en) 2001-11-20
TR200302294T4 (tr) 2004-02-23
PL358201A1 (en) 2004-08-09
IL152177A0 (en) 2003-05-29
CZ20023721A3 (cs) 2003-02-12
US20060089366A1 (en) 2006-04-27
PT1283838E (pt) 2004-04-30
UA72337C2 (uk) 2005-02-15
AU2001263927B2 (en) 2004-09-30
US20030119849A1 (en) 2003-06-26
DE60101386D1 (de) 2004-01-15
CA2405971A1 (en) 2001-11-15
CA2405971C (en) 2010-03-30
BR0110592A (pt) 2003-04-01
CN1174979C (zh) 2004-11-10
JP2003532729A (ja) 2003-11-05
WO2001085725A1 (en) 2001-11-15
CZ301464B6 (cs) 2010-03-10
HUP0302016A2 (hu) 2003-09-29
US6911448B2 (en) 2005-06-28
DE60101386T2 (de) 2004-05-27

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