DK1131292T3 - Acycliske og cycliske guanidin- og acetamidinderivater, deres fremstilling og deres anvendelse som pesticider, især som parasiticider - Google Patents

Acycliske og cycliske guanidin- og acetamidinderivater, deres fremstilling og deres anvendelse som pesticider, især som parasiticider

Info

Publication number
DK1131292T3
DK1131292T3 DK99958038T DK99958038T DK1131292T3 DK 1131292 T3 DK1131292 T3 DK 1131292T3 DK 99958038 T DK99958038 T DK 99958038T DK 99958038 T DK99958038 T DK 99958038T DK 1131292 T3 DK1131292 T3 DK 1131292T3
Authority
DK
Denmark
Prior art keywords
parasiticides
pesticides
acyclic
preparation
cyclic guanidine
Prior art date
Application number
DK99958038T
Other languages
English (en)
Inventor
Thomas Goebel
Eliane Humbert-Droz
Maurizio Schwarzenbach
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Application granted granted Critical
Publication of DK1131292T3 publication Critical patent/DK1131292T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/12—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing a —O—CO—N< group, or a thio analogue thereof, neither directly attached to a ring nor the nitrogen atom being a member of a heterocyclic ring
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/16—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/40—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides
    • A01N47/42—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides containing —N=CX2 groups, e.g. isothiourea
    • A01N47/44—Guanidine; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
DK99958038T 1998-11-17 1999-11-15 Acycliske og cycliske guanidin- og acetamidinderivater, deres fremstilling og deres anvendelse som pesticider, især som parasiticider DK1131292T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH229898 1998-11-17
CH79799 1999-04-29

Publications (1)

Publication Number Publication Date
DK1131292T3 true DK1131292T3 (da) 2006-04-18

Family

ID=25685711

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99958038T DK1131292T3 (da) 1998-11-17 1999-11-15 Acycliske og cycliske guanidin- og acetamidinderivater, deres fremstilling og deres anvendelse som pesticider, især som parasiticider

Country Status (22)

Country Link
US (3) US6538013B2 (da)
EP (1) EP1131292B1 (da)
JP (1) JP2002529532A (da)
KR (1) KR100620470B1 (da)
CN (1) CN1177823C (da)
AR (1) AR023703A1 (da)
AT (1) ATE317385T1 (da)
AU (1) AU762529B2 (da)
BR (1) BR9915430A (da)
CA (1) CA2350742A1 (da)
CO (1) CO5210925A1 (da)
CY (1) CY1106083T1 (da)
DE (1) DE69929820T2 (da)
DK (1) DK1131292T3 (da)
ES (1) ES2255766T3 (da)
HK (1) HK1038563B (da)
IL (2) IL142687A0 (da)
NZ (1) NZ511380A (da)
PT (1) PT1131292E (da)
RU (1) RU2245877C2 (da)
TW (1) TW561149B (da)
WO (1) WO2000029378A2 (da)

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US20050026811A1 (en) * 2003-05-20 2005-02-03 Mjalli Adnan M. M. Rage antagonists as agents to reverse amyloidosis and diseases associated therewith
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US7186855B2 (en) * 2001-06-11 2007-03-06 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
US6818787B2 (en) * 2001-06-11 2004-11-16 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
US8048917B2 (en) 2005-04-06 2011-11-01 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
US7232924B2 (en) * 2001-06-11 2007-06-19 Xenoport, Inc. Methods for synthesis of acyloxyalkyl derivatives of GABA analogs
JP2003026603A (ja) * 2001-07-17 2003-01-29 Sumika Life Tech Co Ltd コンパニオンアニマルの外部寄生虫駆除用水性滴下剤
US7011837B2 (en) * 2001-08-29 2006-03-14 Rutgers, The State University Of New Jersey Isolated species of steinernematid nematode and methods of white grub control therewith
MXPA04002477A (es) 2001-09-17 2004-05-31 Lilly Co Eli Formulaciones pesticidas.
CN101597262A (zh) * 2002-03-05 2009-12-09 特兰斯泰克制药公司 抑制配体与高级糖化终产物受体相互作用的单和双环吡咯衍生物
US7396819B2 (en) * 2003-08-08 2008-07-08 Virbac Corporation Anthelmintic formulations
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AR054849A1 (es) * 2005-07-26 2007-07-18 Wyeth Corp Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlas
TW200734334A (en) * 2006-01-13 2007-09-16 Wyeth Corp Treatment of substance abuse
CA2645099A1 (en) * 2006-03-24 2007-10-04 Wyeth Methods for modulating bladder function
WO2007112000A2 (en) * 2006-03-24 2007-10-04 Wyeth Treatment of pain
PE20080126A1 (es) * 2006-03-24 2008-04-07 Wyeth Corp Metodos para tratar trastornos cognitivos y otros afines
US20070225279A1 (en) * 2006-03-24 2007-09-27 Wyeth Therapeutic combinations for the treatment of depression
CL2008002777A1 (es) * 2007-09-21 2010-01-22 Wyeth Corp Metodo de preparacion de compuestos diazepinoquinolinicos quirales por recristalizacion en un sistema de solvente ternario.
FR2922108A1 (fr) * 2007-10-11 2009-04-17 Virbac Sa Utilisation d'un derive de 1-n-(halo-3-pyridylmethyle)-n-methylamino-1-alkylamino -2- nitroethylene pour la preparation d'une composition pharmaceutique veterinaire pour lutter contre les puces
US20100267662A1 (en) * 2007-11-08 2010-10-21 Ceapro, Inc. Avenanthramide-containing compositions
AU2009316899B2 (en) * 2008-11-19 2015-08-20 Boehringer Ingelheim Animal Health USA Inc. Compositions comprising 1-arylpyrazole alone or in combination with formamidine for the treatment of parasitic infection
US9173728B2 (en) 2008-11-19 2015-11-03 Merial Inc. Multi-cavity container having offset indentures for dispensing fluids
TWI517850B (zh) 2009-09-30 2016-01-21 Ｖｔｖ治療有限責任公司 經取代之咪唑衍生物及其使用方法
BR112013017305B1 (pt) 2011-01-04 2021-08-17 The Climate Corporation Métodos de gerar mapa de dados de solo
WO2012138320A1 (en) * 2011-04-04 2012-10-11 Carro, A Ingestible insect repellent composition and system
NZ722096A (en) 2011-12-15 2016-11-25 Alkermes Pharma Ireland Ltd Prodrugs of secondary amine compounds
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CN111978244B (zh) * 2019-05-24 2022-09-06 南开大学 一类烯啶虫胺酰基衍生物的合成及其应用
CN111978243B (zh) * 2019-05-24 2022-09-06 南开大学 草酸单酯类衍生物的合成及其应用
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Also Published As

Publication number Publication date
PT1131292E (pt) 2006-06-30
NZ511380A (en) 2003-10-31
HK1038563B (zh) 2006-11-24
BR9915430A (pt) 2001-08-07
ES2255766T3 (es) 2006-07-01
HK1038563A1 (en) 2002-03-22
WO2000029378A2 (en) 2000-05-25
US7271184B2 (en) 2007-09-18
CA2350742A1 (en) 2000-05-25
WO2000029378A3 (en) 2000-12-14
US6538013B2 (en) 2003-03-25
AU762529B2 (en) 2003-06-26
DE69929820D1 (de) 2006-04-20
US6759407B2 (en) 2004-07-06
CY1106083T1 (el) 2011-06-08
JP2002529532A (ja) 2002-09-10
US20040162283A1 (en) 2004-08-19
EP1131292B1 (en) 2006-02-08
AU1553100A (en) 2000-06-05
KR20010086445A (ko) 2001-09-12
US20020028806A1 (en) 2002-03-07
ATE317385T1 (de) 2006-02-15
EP1131292A2 (en) 2001-09-12
DE69929820T2 (de) 2006-07-27
CO5210925A1 (es) 2002-10-30
AR023703A1 (es) 2002-09-04
RU2245877C2 (ru) 2005-02-10
CN1177823C (zh) 2004-12-01
CN1326442A (zh) 2001-12-12
TW561149B (en) 2003-11-11
IL142687A0 (en) 2002-03-10
IL142687A (en) 2006-10-05
KR100620470B1 (ko) 2006-09-13
US20030203891A1 (en) 2003-10-30

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