DK0836606T3 - Kondenserede thiazolderivater, der har 5-HT-receptoraffinitet - Google Patents

Kondenserede thiazolderivater, der har 5-HT-receptoraffinitet

Info

Publication number
DK0836606T3
DK0836606T3 DK96922862T DK96922862T DK0836606T3 DK 0836606 T3 DK0836606 T3 DK 0836606T3 DK 96922862 T DK96922862 T DK 96922862T DK 96922862 T DK96922862 T DK 96922862T DK 0836606 T3 DK0836606 T3 DK 0836606T3
Authority
DK
Denmark
Prior art keywords
receptor affinity
thiazole derivatives
condensed thiazole
condensed
derivatives
Prior art date
Application number
DK96922862T
Other languages
Danish (da)
English (en)
Inventor
Roy Victor Davies
Frank Kerrigan
Sharon Crawford Cheetham
Original Assignee
Knoll Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Knoll Ag filed Critical Knoll Ag
Application granted granted Critical
Publication of DK0836606T3 publication Critical patent/DK0836606T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/10—Expectorants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Anesthesiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
DK96922862T 1995-07-01 1996-06-20 Kondenserede thiazolderivater, der har 5-HT-receptoraffinitet DK0836606T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9513467.2A GB9513467D0 (en) 1995-07-01 1995-07-01 Therapeutic agents
PCT/EP1996/002676 WO1997002269A1 (fr) 1995-07-01 1996-06-20 Derives thiazoles condenses possedant une affinite pour les recepteurs 5-ht

Publications (1)

Publication Number Publication Date
DK0836606T3 true DK0836606T3 (da) 2000-11-20

Family

ID=10777016

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96922862T DK0836606T3 (da) 1995-07-01 1996-06-20 Kondenserede thiazolderivater, der har 5-HT-receptoraffinitet

Country Status (30)

Country Link
US (1) US5869492A (fr)
EP (1) EP0836606B1 (fr)
JP (1) JPH11508568A (fr)
KR (1) KR19990028619A (fr)
CN (1) CN1064966C (fr)
AR (1) AR003963A1 (fr)
AT (1) ATE195942T1 (fr)
AU (1) AU708789B2 (fr)
BG (1) BG63206B1 (fr)
BR (1) BR9609525A (fr)
CA (1) CA2222725A1 (fr)
CO (1) CO4700463A1 (fr)
CZ (1) CZ376297A3 (fr)
DE (1) DE69610104T2 (fr)
DK (1) DK0836606T3 (fr)
ES (1) ES2151175T3 (fr)
GB (1) GB9513467D0 (fr)
GR (1) GR3034397T3 (fr)
HR (1) HRP960306B1 (fr)
HU (1) HUP9901258A3 (fr)
IL (1) IL122158A (fr)
NO (1) NO310660B1 (fr)
NZ (1) NZ312130A (fr)
PL (1) PL324337A1 (fr)
PT (1) PT836606E (fr)
SK (1) SK179297A3 (fr)
TR (1) TR199701756T1 (fr)
TW (1) TW474939B (fr)
WO (1) WO1997002269A1 (fr)
ZA (1) ZA965494B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9705428D0 (en) 1997-03-15 1997-04-30 Knoll Ag Therapeutic agents
ES2244179T3 (es) * 1998-03-31 2005-12-01 SHIONOGI & CO., LTD. Proceso para la preparacion de derivados de acido 5-hidroxibenzo(b)tiofen-3-carboxilico.
DE19908536A1 (de) 1999-02-26 2000-08-31 Aventis Pharma Gmbh Polycyclische Thiazol-2-yliden Amine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
GB9911881D0 (en) * 1999-05-21 1999-07-21 Knoll Ag Therapeutic agents
GB9911863D0 (en) * 1999-05-21 1999-07-21 Knoll Ag Therapeutic agents
GB0005789D0 (en) 2000-03-11 2000-05-03 Knoll Ag Therapeutic agents
GB0023610D0 (en) * 2000-09-27 2000-11-08 Knoll Ag Therapeutic agents
DE10112197A1 (de) * 2001-03-14 2002-09-19 Gruenenthal Gmbh Substituierte Pyrazolo- und Thiazolopyrimidine
US8106074B2 (en) 2001-07-13 2012-01-31 Pierre Fabre Medicament Pyridin-2-yl-methylamine derivatives for treating opiate dependence

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0002400A1 (fr) * 1977-11-24 1979-06-13 Synthelabo Dérivés de thiazole, leur préparation, intermédiaires et leur application en thérapeutique
ES2159526T3 (es) * 1992-07-13 2001-10-16 Janssen Pharmaceutica Nv Nuevos derivados de 4-(3-benzofuranil)piperidinilo y 4-(3-benzotienil)piperidinilo y composiciones farmaceuticas que los contienen.

Also Published As

Publication number Publication date
GB9513467D0 (en) 1995-09-06
DE69610104T2 (de) 2001-01-18
AU6358996A (en) 1997-02-05
BG63206B1 (bg) 2001-06-29
HRP960306B1 (en) 2001-08-31
ES2151175T3 (es) 2000-12-16
ZA965494B (en) 1997-12-29
IL122158A0 (en) 1998-04-05
BG102084A (en) 1998-08-31
AU708789B2 (en) 1999-08-12
AR003963A1 (es) 1998-09-30
PL324337A1 (en) 1998-05-25
WO1997002269A1 (fr) 1997-01-23
TR199701756T1 (xx) 1998-04-21
HRP960306A2 (en) 1998-04-30
CZ376297A3 (cs) 1998-06-17
HUP9901258A2 (hu) 1999-08-30
NO976157D0 (no) 1997-12-30
NO976157L (no) 1997-12-30
JPH11508568A (ja) 1999-07-27
CA2222725A1 (fr) 1997-01-23
BR9609525A (pt) 1999-02-23
GR3034397T3 (en) 2000-12-29
KR19990028619A (ko) 1999-04-15
SK179297A3 (en) 1998-07-08
ATE195942T1 (de) 2000-09-15
NZ312130A (en) 1999-08-30
CN1189834A (zh) 1998-08-05
HUP9901258A3 (en) 2000-08-28
CN1064966C (zh) 2001-04-25
CO4700463A1 (es) 1998-12-29
NO310660B1 (no) 2001-08-06
MX9709509A (es) 1998-03-29
US5869492A (en) 1999-02-09
DE69610104D1 (de) 2000-10-05
TW474939B (en) 2002-02-01
PT836606E (pt) 2001-02-28
EP0836606B1 (fr) 2000-08-30
IL122158A (en) 2000-01-31
EP0836606A1 (fr) 1998-04-22

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