DK0708105T3 - 5-HT4-receptoragonister - Google Patents
5-HT4-receptoragonisterInfo
- Publication number
- DK0708105T3 DK0708105T3 DK95307480T DK95307480T DK0708105T3 DK 0708105 T3 DK0708105 T3 DK 0708105T3 DK 95307480 T DK95307480 T DK 95307480T DK 95307480 T DK95307480 T DK 95307480T DK 0708105 T3 DK0708105 T3 DK 0708105T3
- Authority
- DK
- Denmark
- Prior art keywords
- receptor agonists
- agonists
- receptor
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP25490794 | 1994-10-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
DK0708105T3 true DK0708105T3 (da) | 1999-08-23 |
Family
ID=17271511
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK95307480T DK0708105T3 (da) | 1994-10-20 | 1995-10-20 | 5-HT4-receptoragonister |
Country Status (8)
Country | Link |
---|---|
US (1) | US5684003A (da) |
EP (1) | EP0708105B1 (da) |
KR (1) | KR960014128A (da) |
CA (1) | CA2160420A1 (da) |
DE (1) | DE69506826T2 (da) |
DK (1) | DK0708105T3 (da) |
ES (1) | ES2128668T3 (da) |
TW (1) | TW403747B (da) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR19990022096A (ko) * | 1995-05-31 | 1999-03-25 | 쇼다 오사무 | 모노시클릭 아미노기를 갖는 인다졸 유도체 |
US5914405A (en) * | 1997-10-07 | 1999-06-22 | Eli Lilly And Company | Process for preparing 3-substituted indazoles |
US6069152A (en) * | 1997-10-07 | 2000-05-30 | Eli Lilly And Company | 5-HT4 agonists and antagonists |
FR2792318B1 (fr) * | 1999-04-16 | 2001-06-15 | Synthelabo | Derives d'indazole, leur preparation et leur application en therapeutique |
US7671097B2 (en) * | 2005-05-24 | 2010-03-02 | Georgia-Pacific Chemicals Llc | Stable phenolic resin polymer dispersions having low free aldehyde content |
WO2003035005A2 (en) | 2001-10-26 | 2003-05-01 | University Of Connecticut | Heteroindanes: a new class of potent cannabimimetic ligands |
TW200533348A (en) * | 2004-02-18 | 2005-10-16 | Theravance Inc | Indazole-carboxamide compounds as 5-ht4 receptor agonists |
US8309575B2 (en) | 2004-04-07 | 2012-11-13 | Theravance, Inc. | Quinolinone-carboxamide compounds as 5-HT4 receptor agonists |
US7728006B2 (en) * | 2004-04-07 | 2010-06-01 | Theravance, Inc. | Quinolinone-carboxamide compounds as 5-HT4 receptor agonists |
TWI351282B (en) | 2004-04-07 | 2011-11-01 | Theravance Inc | Quinolinone-carboxamide compounds as 5-ht4 recepto |
WO2006052640A1 (en) * | 2004-11-05 | 2006-05-18 | Theravance, Inc. | 5-ht4 receptor agonist compounds |
ES2327142T3 (es) * | 2004-11-05 | 2009-10-26 | Theravance, Inc. | Compuestos de quinolinona-carboxamida. |
NZ555180A (en) * | 2004-12-22 | 2010-09-30 | Theravance Inc | Indazole-carboxamide compounds useful as 5-HT4 receptor agonists |
NZ560828A (en) * | 2005-03-02 | 2011-01-28 | Theravance Inc | Quinolinone compounds as 5-HT4 receptor agonists |
JOP20130213B1 (ar) * | 2012-07-17 | 2021-08-17 | Takeda Pharmaceuticals Co | معارضات لمستقبلht3-5 |
PL3201203T3 (pl) | 2014-09-29 | 2021-11-22 | Takeda Pharmaceutical Company Limited | Krystaliczna postać 1-(1-metylo-1h-pirazol-4-ilo)-n-((1r,5s,7s)-9-metylo-3-oksa-9-azabicyklo[3.3.1]nonan-7-ylo)-1h-indolo-3-karboksyamidu |
GB201511382D0 (en) | 2015-06-29 | 2015-08-12 | Imp Innovations Ltd | Novel compounds and their use in therapy |
WO2023230540A2 (en) * | 2022-05-25 | 2023-11-30 | Katholieke Universiteit Leuven | Indazole derivatives for treating trpm3-mediated disorders |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8829079D0 (en) * | 1988-12-13 | 1989-01-25 | Beecham Group Plc | Novel compounds |
GB9009389D0 (en) * | 1990-04-26 | 1990-06-20 | Smith Kline French Lab | Treatment |
US5256656A (en) * | 1990-07-31 | 1993-10-26 | Nisshin Flour Milling Co., Ltd. | Azabicyclo derivatives |
US5187166A (en) * | 1990-07-31 | 1993-02-16 | Nisshin Flour Milling Co., Ltd. | Azabicyclo derivatives and their use as antiemetics |
TW251287B (da) * | 1993-04-30 | 1995-07-11 | Nissei Co Ltd |
-
1995
- 1995-10-12 US US08/543,853 patent/US5684003A/en not_active Expired - Lifetime
- 1995-10-12 CA CA002160420A patent/CA2160420A1/en not_active Abandoned
- 1995-10-20 TW TW084111089A patent/TW403747B/zh not_active IP Right Cessation
- 1995-10-20 DK DK95307480T patent/DK0708105T3/da active
- 1995-10-20 ES ES95307480T patent/ES2128668T3/es not_active Expired - Lifetime
- 1995-10-20 EP EP95307480A patent/EP0708105B1/en not_active Expired - Lifetime
- 1995-10-20 KR KR1019950036424A patent/KR960014128A/ko not_active Application Discontinuation
- 1995-10-20 DE DE69506826T patent/DE69506826T2/de not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
EP0708105B1 (en) | 1998-12-23 |
US5684003A (en) | 1997-11-04 |
KR960014128A (ko) | 1996-05-22 |
CA2160420A1 (en) | 1996-04-21 |
DE69506826D1 (de) | 1999-02-04 |
EP0708105A1 (en) | 1996-04-24 |
TW403747B (en) | 2000-09-01 |
DE69506826T2 (de) | 1999-08-05 |
ES2128668T3 (es) | 1999-05-16 |
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