DK0708105T3 - 5-HT4-receptoragonister - Google Patents

5-HT4-receptoragonister

Info

Publication number
DK0708105T3
DK0708105T3 DK95307480T DK95307480T DK0708105T3 DK 0708105 T3 DK0708105 T3 DK 0708105T3 DK 95307480 T DK95307480 T DK 95307480T DK 95307480 T DK95307480 T DK 95307480T DK 0708105 T3 DK0708105 T3 DK 0708105T3
Authority
DK
Denmark
Prior art keywords
receptor agonists
agonists
receptor
Prior art date
Application number
DK95307480T
Other languages
English (en)
Inventor
Hiroaki Satoh
Masashi Suzuki
Ruta Fukutomi
Masahiro Ueno
Koichiro Hagihara
Takeo Arai
Setsuko Mino
Yumiko Noguchi
Haruhiko Kikuchi
Original Assignee
Nisshin Flour Milling Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nisshin Flour Milling Co filed Critical Nisshin Flour Milling Co
Application granted granted Critical
Publication of DK0708105T3 publication Critical patent/DK0708105T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK95307480T 1994-10-20 1995-10-20 5-HT4-receptoragonister DK0708105T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP25490794 1994-10-20

Publications (1)

Publication Number Publication Date
DK0708105T3 true DK0708105T3 (da) 1999-08-23

Family

ID=17271511

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95307480T DK0708105T3 (da) 1994-10-20 1995-10-20 5-HT4-receptoragonister

Country Status (8)

Country Link
US (1) US5684003A (da)
EP (1) EP0708105B1 (da)
KR (1) KR960014128A (da)
CA (1) CA2160420A1 (da)
DE (1) DE69506826T2 (da)
DK (1) DK0708105T3 (da)
ES (1) ES2128668T3 (da)
TW (1) TW403747B (da)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR19990022096A (ko) * 1995-05-31 1999-03-25 쇼다 오사무 모노시클릭 아미노기를 갖는 인다졸 유도체
US5914405A (en) * 1997-10-07 1999-06-22 Eli Lilly And Company Process for preparing 3-substituted indazoles
US6069152A (en) * 1997-10-07 2000-05-30 Eli Lilly And Company 5-HT4 agonists and antagonists
FR2792318B1 (fr) * 1999-04-16 2001-06-15 Synthelabo Derives d'indazole, leur preparation et leur application en therapeutique
US7671097B2 (en) * 2005-05-24 2010-03-02 Georgia-Pacific Chemicals Llc Stable phenolic resin polymer dispersions having low free aldehyde content
WO2003035005A2 (en) 2001-10-26 2003-05-01 University Of Connecticut Heteroindanes: a new class of potent cannabimimetic ligands
TW200533348A (en) * 2004-02-18 2005-10-16 Theravance Inc Indazole-carboxamide compounds as 5-ht4 receptor agonists
US8309575B2 (en) 2004-04-07 2012-11-13 Theravance, Inc. Quinolinone-carboxamide compounds as 5-HT4 receptor agonists
US7728006B2 (en) * 2004-04-07 2010-06-01 Theravance, Inc. Quinolinone-carboxamide compounds as 5-HT4 receptor agonists
TWI351282B (en) 2004-04-07 2011-11-01 Theravance Inc Quinolinone-carboxamide compounds as 5-ht4 recepto
WO2006052640A1 (en) * 2004-11-05 2006-05-18 Theravance, Inc. 5-ht4 receptor agonist compounds
ES2327142T3 (es) * 2004-11-05 2009-10-26 Theravance, Inc. Compuestos de quinolinona-carboxamida.
NZ555180A (en) * 2004-12-22 2010-09-30 Theravance Inc Indazole-carboxamide compounds useful as 5-HT4 receptor agonists
NZ560828A (en) * 2005-03-02 2011-01-28 Theravance Inc Quinolinone compounds as 5-HT4 receptor agonists
JOP20130213B1 (ar) * 2012-07-17 2021-08-17 Takeda Pharmaceuticals Co معارضات لمستقبلht3-5
PL3201203T3 (pl) 2014-09-29 2021-11-22 Takeda Pharmaceutical Company Limited Krystaliczna postać 1-(1-metylo-1h-pirazol-4-ilo)-n-((1r,5s,7s)-9-metylo-3-oksa-9-azabicyklo[3.3.1]nonan-7-ylo)-1h-indolo-3-karboksyamidu
GB201511382D0 (en) 2015-06-29 2015-08-12 Imp Innovations Ltd Novel compounds and their use in therapy
WO2023230540A2 (en) * 2022-05-25 2023-11-30 Katholieke Universiteit Leuven Indazole derivatives for treating trpm3-mediated disorders

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8829079D0 (en) * 1988-12-13 1989-01-25 Beecham Group Plc Novel compounds
GB9009389D0 (en) * 1990-04-26 1990-06-20 Smith Kline French Lab Treatment
US5256656A (en) * 1990-07-31 1993-10-26 Nisshin Flour Milling Co., Ltd. Azabicyclo derivatives
US5187166A (en) * 1990-07-31 1993-02-16 Nisshin Flour Milling Co., Ltd. Azabicyclo derivatives and their use as antiemetics
TW251287B (da) * 1993-04-30 1995-07-11 Nissei Co Ltd

Also Published As

Publication number Publication date
EP0708105B1 (en) 1998-12-23
US5684003A (en) 1997-11-04
KR960014128A (ko) 1996-05-22
CA2160420A1 (en) 1996-04-21
DE69506826D1 (de) 1999-02-04
EP0708105A1 (en) 1996-04-24
TW403747B (en) 2000-09-01
DE69506826T2 (de) 1999-08-05
ES2128668T3 (es) 1999-05-16

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