HRP960306B1 - Condensed thiazole derivatives having 5-ht receptor affinity - Google Patents

Condensed thiazole derivatives having 5-ht receptor affinity

Info

Publication number
HRP960306B1
HRP960306B1 HR960306A HRP960306A HRP960306B1 HR P960306 B1 HRP960306 B1 HR P960306B1 HR 960306 A HR960306 A HR 960306A HR P960306 A HRP960306 A HR P960306A HR P960306 B1 HRP960306 B1 HR P960306B1
Authority
HR
Croatia
Prior art keywords
receptor affinity
thiazole derivatives
condensed thiazole
condensed
derivatives
Prior art date
Application number
HR960306A
Other languages
English (en)
Inventor
Frank Kerrigan
Sharon Crawford Cheetham
Roy Victor Davies
Original Assignee
Knoll Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Knoll Ag filed Critical Knoll Ag
Publication of HRP960306A2 publication Critical patent/HRP960306A2/hr
Publication of HRP960306B1 publication Critical patent/HRP960306B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/10—Expectorants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Anesthesiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
HR960306A 1995-07-01 1996-07-01 Condensed thiazole derivatives having 5-ht receptor affinity HRP960306B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9513467.2A GB9513467D0 (en) 1995-07-01 1995-07-01 Therapeutic agents

Publications (2)

Publication Number Publication Date
HRP960306A2 HRP960306A2 (en) 1998-04-30
HRP960306B1 true HRP960306B1 (en) 2001-08-31

Family

ID=10777016

Family Applications (1)

Application Number Title Priority Date Filing Date
HR960306A HRP960306B1 (en) 1995-07-01 1996-07-01 Condensed thiazole derivatives having 5-ht receptor affinity

Country Status (30)

Country Link
US (1) US5869492A (xx)
EP (1) EP0836606B1 (xx)
JP (1) JPH11508568A (xx)
KR (1) KR19990028619A (xx)
CN (1) CN1064966C (xx)
AR (1) AR003963A1 (xx)
AT (1) ATE195942T1 (xx)
AU (1) AU708789B2 (xx)
BG (1) BG63206B1 (xx)
BR (1) BR9609525A (xx)
CA (1) CA2222725A1 (xx)
CO (1) CO4700463A1 (xx)
CZ (1) CZ376297A3 (xx)
DE (1) DE69610104T2 (xx)
DK (1) DK0836606T3 (xx)
ES (1) ES2151175T3 (xx)
GB (1) GB9513467D0 (xx)
GR (1) GR3034397T3 (xx)
HR (1) HRP960306B1 (xx)
HU (1) HUP9901258A3 (xx)
IL (1) IL122158A (xx)
NO (1) NO310660B1 (xx)
NZ (1) NZ312130A (xx)
PL (1) PL324337A1 (xx)
PT (1) PT836606E (xx)
SK (1) SK179297A3 (xx)
TR (1) TR199701756T1 (xx)
TW (1) TW474939B (xx)
WO (1) WO1997002269A1 (xx)
ZA (1) ZA965494B (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9705428D0 (en) * 1997-03-15 1997-04-30 Knoll Ag Therapeutic agents
US6320060B1 (en) 1998-03-31 2001-11-20 Shionogi & Co., Ltd. Process for producing 5-hydroxybenzo[b] thiophene-3-carboxylic acid derivatives
DE19908536A1 (de) * 1999-02-26 2000-08-31 Aventis Pharma Gmbh Polycyclische Thiazol-2-yliden Amine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
GB9911881D0 (en) * 1999-05-21 1999-07-21 Knoll Ag Therapeutic agents
GB9911863D0 (en) * 1999-05-21 1999-07-21 Knoll Ag Therapeutic agents
GB0005789D0 (en) * 2000-03-11 2000-05-03 Knoll Ag Therapeutic agents
GB0023610D0 (en) * 2000-09-27 2000-11-08 Knoll Ag Therapeutic agents
DE10112197A1 (de) * 2001-03-14 2002-09-19 Gruenenthal Gmbh Substituierte Pyrazolo- und Thiazolopyrimidine
US8106074B2 (en) 2001-07-13 2012-01-31 Pierre Fabre Medicament Pyridin-2-yl-methylamine derivatives for treating opiate dependence

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0002400A1 (fr) * 1977-11-24 1979-06-13 Synthelabo Dérivés de thiazole, leur préparation, intermédiaires et leur application en thérapeutique
PT672043E (pt) * 1992-07-13 2001-11-30 Janssen Pharmaceutica Nv Novos derivados de 4-(3-benzofuranil)piperidinilo e 4-(3-benzotienil)piperidinilo e composicoes farmaceuticas que os contem

Also Published As

Publication number Publication date
IL122158A (en) 2000-01-31
MX9709509A (es) 1998-03-29
GR3034397T3 (en) 2000-12-29
NO976157D0 (no) 1997-12-30
HUP9901258A3 (en) 2000-08-28
CA2222725A1 (en) 1997-01-23
PL324337A1 (en) 1998-05-25
IL122158A0 (en) 1998-04-05
CO4700463A1 (es) 1998-12-29
KR19990028619A (ko) 1999-04-15
EP0836606B1 (en) 2000-08-30
BR9609525A (pt) 1999-02-23
AR003963A1 (es) 1998-09-30
NO976157L (no) 1997-12-30
CN1064966C (zh) 2001-04-25
JPH11508568A (ja) 1999-07-27
DE69610104D1 (de) 2000-10-05
CN1189834A (zh) 1998-08-05
TW474939B (en) 2002-02-01
NZ312130A (en) 1999-08-30
BG63206B1 (bg) 2001-06-29
BG102084A (en) 1998-08-31
ZA965494B (en) 1997-12-29
WO1997002269A1 (en) 1997-01-23
CZ376297A3 (cs) 1998-06-17
GB9513467D0 (en) 1995-09-06
DK0836606T3 (da) 2000-11-20
US5869492A (en) 1999-02-09
HUP9901258A2 (hu) 1999-08-30
AU708789B2 (en) 1999-08-12
AU6358996A (en) 1997-02-05
ATE195942T1 (de) 2000-09-15
NO310660B1 (no) 2001-08-06
SK179297A3 (en) 1998-07-08
DE69610104T2 (de) 2001-01-18
PT836606E (pt) 2001-02-28
EP0836606A1 (en) 1998-04-22
HRP960306A2 (en) 1998-04-30
TR199701756T1 (xx) 1998-04-21
ES2151175T3 (es) 2000-12-16

Similar Documents

Publication Publication Date Title
GR3033626T3 (en) 3-pyrazolecarboxamide derivatives having cannabinoid receptor affinity
GR3035075T3 (en) Indole derivatives as 5-ht receptor antagonist
AU4616696A (en) Indole derivatives with affinity for the cannabinoid receptor
TW356142U (en) Suspension arm
PL329121A1 (en) Substituted derivatives of 1,2,3,4-tetrahydronaphtalene
AU3934695A (en) N-methyl piperazine compounds having dopamine receptor affinity
AU3934595A (en) Alkyl-substituted compounds having dopamine receptor affinity
EP0853629A4 (en) HEPATITIS DNA VIRUS RECEPTOR
DK0708105T3 (da) 5-HT4-receptoragonister
AU2314195A (en) Benzofuran derivatives as d4 receptor antagonists
TW310087U (en) Joint for extension rod
HU9601565D0 (en) N-acyl-(2-aryl-cyclopropyl-methyl)-amine derivatives
HRP960306B1 (en) Condensed thiazole derivatives having 5-ht receptor affinity
GB9517098D0 (en) Receptor
AU3934995A (en) Benzyl-substituted compounds having dopamine receptor affinity
PL330708A1 (en) Derivatives of indolydine useful as antagonists of 5-ht-2c receptor
FI971854A (fi) Substituoituja tetrasyklisiä atsepiinijohdannaisia, joilla on 5-HT2-reseptoriaffiniteetti
GB2313403B (en) Adjustable fixing arm for friction stays
SI0836606T1 (en) Condensed thiazole derivatives, having 5-ht receptor affinity
IL139552A0 (en) N-benzodioxanylmethyl-1-piperidylmethylamine compounds having affinity for 5-ht receptors
AU7578396A (en) Substituted tetrahydropyridine derivatives acting on 5-ht receptors
GB9715018D0 (en) 3-Fluoro-4-aminopiperidine derivatives as 5-HT receptor agonists
AU1449997A (en) Diazabicyclo-octane derivatives as 5-ht receptor ligands
ZA9600758D (en) Idole derivatives as 5-ht receptor antagonist.
SI0712406T1 (en) Condensed indole derivatives as 5-ht 4-receptor antagonists

Legal Events

Date Code Title Description
A1OB Publication of a patent application
AIPI Request for the grant of a patent on the basis of a substantive examination of a patent application
ODRP Renewal fee for the maintenance of a patent

Payment date: 20010701

Year of fee payment: 6

B1PR Patent granted
PBON Lapse due to non-payment of renewal fee

Effective date: 20020702