DK0686641T3 - 2'-Deoxy-5-fluoruridinderivat, farmaceutisk acceptabelt salt deraf, fremgangsmåde til fremstilling deraf, og antitumorlægem - Google Patents

2'-Deoxy-5-fluoruridinderivat, farmaceutisk acceptabelt salt deraf, fremgangsmåde til fremstilling deraf, og antitumorlægem

Info

Publication number
DK0686641T3
DK0686641T3 DK95903918T DK95903918T DK0686641T3 DK 0686641 T3 DK0686641 T3 DK 0686641T3 DK 95903918 T DK95903918 T DK 95903918T DK 95903918 T DK95903918 T DK 95903918T DK 0686641 T3 DK0686641 T3 DK 0686641T3
Authority
DK
Denmark
Prior art keywords
deoxy
pharmaceutically acceptable
acceptable salt
preparation
tumor drug
Prior art date
Application number
DK95903918T
Other languages
English (en)
Inventor
Makoto Nomura
Makoto Kajitani
Junichi Yamashita
Masakazu Fukushima
Yuji Shimamoto
Original Assignee
Taiho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taiho Pharmaceutical Co Ltd filed Critical Taiho Pharmaceutical Co Ltd
Application granted granted Critical
Publication of DK0686641T3 publication Critical patent/DK0686641T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK95903918T 1993-12-24 1994-12-21 2'-Deoxy-5-fluoruridinderivat, farmaceutisk acceptabelt salt deraf, fremgangsmåde til fremstilling deraf, og antitumorlægem DK0686641T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP05327338A JP3074341B2 (ja) 1993-12-24 1993-12-24 2’−デオキシ−5−フルオロウリジン誘導体
PCT/JP1994/002167 WO1995018138A1 (fr) 1993-12-24 1994-12-21 Derive de 2'-desoxy-5-fluorouridine, sel pharmaceutiquement acceptable de ce dernier, son procede de production et medicament anti-tumoral

Publications (1)

Publication Number Publication Date
DK0686641T3 true DK0686641T3 (da) 1998-11-23

Family

ID=18198026

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95903918T DK0686641T3 (da) 1993-12-24 1994-12-21 2'-Deoxy-5-fluoruridinderivat, farmaceutisk acceptabelt salt deraf, fremgangsmåde til fremstilling deraf, og antitumorlægem

Country Status (9)

Country Link
US (1) US5869464A (da)
EP (1) EP0686641B1 (da)
JP (1) JP3074341B2 (da)
AT (1) ATE170188T1 (da)
AU (1) AU1370895A (da)
DE (1) DE69412794T2 (da)
DK (1) DK0686641T3 (da)
ES (1) ES2122521T3 (da)
WO (1) WO1995018138A1 (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107936154B (zh) 2017-12-01 2020-11-06 中国石油天然气股份有限公司 一种烷氧基镁催化剂载体及其制备方法和应用
JP2021161216A (ja) 2020-03-31 2021-10-11 住友化学株式会社 オレフィン重合用固体触媒成分

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS56113797A (en) * 1980-02-14 1981-09-07 Funai Corp 3-benzoyl-5-fluorouridine derivative, its preparation and antitumor agent containing the same
JPS5728083A (en) * 1980-07-25 1982-02-15 Funai Corp 4-position ether derivative of deoxydiacetyl-fluorouridine
JPS5750999A (en) * 1980-09-11 1982-03-25 Funai Corp Benzyloxy derivative at 4-position of deoxyfluorouridine
JPS57109722A (en) * 1980-12-26 1982-07-08 Funai Corp Antitumor agent containing deoxyfluorouridine benzyloxylated at 4-position
EP0081386B1 (en) * 1981-12-09 1985-05-29 Teijin Limited 5-fluoro-2'-deoxyuridine derivatives and a process for the preparation thereof
US4864021A (en) * 1984-10-30 1989-09-05 Otsuka Pharmaceutical Co., Ltd. 5-fluorouracil derivatives
JPH0696590B2 (ja) * 1985-04-16 1994-11-30 富山化学工業株式会社 新規な5−フルオロ−2′−デオキシウリジン−3′−ホスフエ−ト誘導体およびその塩
AU610913B2 (en) * 1987-07-31 1991-05-30 Taiho Pharmaceutical Co., Ltd. 2'-deoxy-5-fluorouridine derivatives
US4992534A (en) * 1987-08-12 1991-02-12 Otsuka Pharmaceutical Co., Ltd. 3'-O-,5'-O-derivatives of 2'-deoxy-5-fluorouridine

Also Published As

Publication number Publication date
EP0686641A1 (en) 1995-12-13
JP3074341B2 (ja) 2000-08-07
DE69412794T2 (de) 1999-04-29
DE69412794D1 (de) 1998-10-01
EP0686641B1 (en) 1998-08-26
JPH07188277A (ja) 1995-07-25
WO1995018138A1 (fr) 1995-07-06
ES2122521T3 (es) 1998-12-16
ATE170188T1 (de) 1998-09-15
AU1370895A (en) 1995-07-17
EP0686641A4 (en) 1996-07-10
US5869464A (en) 1999-02-09

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