DK0490689T3 - 3-(2-(Dimethylamino)ethyl)-N-methyl-1H-indol-5-methansulfonamid sulfatsalt (2:1) - Google Patents

3-(2-(Dimethylamino)ethyl)-N-methyl-1H-indol-5-methansulfonamid sulfatsalt (2:1)

Info

Publication number
DK0490689T3
DK0490689T3 DK91311583.8T DK91311583T DK0490689T3 DK 0490689 T3 DK0490689 T3 DK 0490689T3 DK 91311583 T DK91311583 T DK 91311583T DK 0490689 T3 DK0490689 T3 DK 0490689T3
Authority
DK
Denmark
Prior art keywords
indole
dimethylamino
ethyl
methyl
sulfate salt
Prior art date
Application number
DK91311583.8T
Other languages
Danish (da)
English (en)
Inventor
Joanne Craig
Derek Leslie Crookes
Stephen John Skittrall
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of DK0490689T3 publication Critical patent/DK0490689T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16—Tryptamines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Indole Compounds (AREA)
DK91311583.8T 1990-12-12 1991-12-12 3-(2-(Dimethylamino)ethyl)-N-methyl-1H-indol-5-methansulfonamid sulfatsalt (2:1) DK0490689T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB909026998A GB9026998D0 (en) 1990-12-12 1990-12-12 Medicaments

Publications (1)

Publication Number Publication Date
DK0490689T3 true DK0490689T3 (da) 1995-05-22

Family

ID=10686904

Family Applications (1)

Application Number Title Priority Date Filing Date
DK91311583.8T DK0490689T3 (da) 1990-12-12 1991-12-12 3-(2-(Dimethylamino)ethyl)-N-methyl-1H-indol-5-methansulfonamid sulfatsalt (2:1)

Country Status (36)

Country Link
US (2) US5554639A (cs)
EP (1) EP0490689B1 (cs)
JP (1) JP2994037B2 (cs)
KR (1) KR100211479B1 (cs)
CN (2) CN1030890C (cs)
AP (1) AP230A (cs)
AT (1) ATE119881T1 (cs)
AU (1) AU650706B2 (cs)
BE (1) BE1005085A3 (cs)
CA (1) CA2098302C (cs)
CH (1) CH684192A5 (cs)
CY (1) CY2005A (cs)
CZ (1) CZ281931B6 (cs)
DE (1) DE69108200T2 (cs)
DK (1) DK0490689T3 (cs)
EG (1) EG20219A (cs)
ES (1) ES2069836T3 (cs)
FR (1) FR2670487B1 (cs)
GB (2) GB9026998D0 (cs)
GR (1) GR3015430T3 (cs)
HK (1) HK82697A (cs)
HU (1) HU211937A9 (cs)
IE (1) IE62894B1 (cs)
IL (1) IL100330A (cs)
IS (1) IS1706B (cs)
IT (1) IT1252868B (cs)
MX (1) MX9102501A (cs)
MY (1) MY109265A (cs)
NL (1) NL9102071A (cs)
NZ (1) NZ240942A (cs)
PT (1) PT99757B (cs)
RU (1) RU2108328C1 (cs)
TW (2) TW300886B (cs)
WO (1) WO1992010477A1 (cs)
YU (1) YU48926B (cs)
ZA (1) ZA919750B (cs)

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US7074893B2 (en) * 2002-06-03 2006-07-11 Regents Of The University Of Michigan Methods and compositions for the treatment of diseases associated with signal transduction aberrations
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MX2007014613A (es) 2005-05-20 2008-04-02 Johnson & Johnson Procedimiento para la preparacion de derivados de sulfamida.
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AR058389A1 (es) 2005-12-19 2008-01-30 Janssen Pharmaceutica Nv Uso de derivados heterociclicos benzo-fusionados de sulfamida para el tratamiento de la obesidad
US8716231B2 (en) 2005-12-19 2014-05-06 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain
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KR20250036962A (ko) 2017-11-07 2025-03-14 더 리젠츠 오브 더 유니버시티 오브 미시건 공유 에피토프-칼레티쿨린 상호 작용의 소분자 억제제 및 사용 방법
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GB8928208D0 (en) * 1989-12-13 1990-02-14 Glaxo Group Ltd Medicaments

Also Published As

Publication number Publication date
ITRM910922A1 (it) 1993-06-11
TW205035B (cs) 1993-05-01
CZ281931B6 (cs) 1997-04-16
MX9102501A (es) 1992-09-01
EG20219A (en) 1997-11-30
PT99757A (pt) 1992-12-31
ATE119881T1 (de) 1995-04-15
CY2005A (en) 1997-12-05
IE914317A1 (en) 1992-06-17
AU650706B2 (en) 1994-06-30
JP2994037B2 (ja) 1999-12-27
US5554639A (en) 1996-09-10
NL9102071A (nl) 1992-07-01
DE69108200D1 (de) 1995-04-20
TW300886B (cs) 1997-03-21
CN1050831C (zh) 2000-03-29
HU211937A9 (en) 1996-01-29
CN1030890C (zh) 1996-02-07
AU9072091A (en) 1992-07-08
RU2108328C1 (ru) 1998-04-10
BE1005085A3 (fr) 1993-04-13
HK82697A (en) 1997-06-27
AP9100339A0 (en) 1992-01-31
CA2098302A1 (en) 1992-06-13
FR2670487B1 (fr) 1993-08-20
CN1063099A (zh) 1992-07-29
DE69108200T2 (de) 1995-07-20
ITRM910922A0 (it) 1991-12-11
ZA919750B (en) 1992-10-28
GR3015430T3 (en) 1995-06-30
EP0490689B1 (en) 1995-03-15
GB2251614B (en) 1994-12-14
YU191491A (sh) 1994-04-05
CN1128259A (zh) 1996-08-07
MY109265A (en) 1996-12-31
AP230A (en) 1993-01-27
GB9026998D0 (en) 1991-01-30
JPH06503560A (ja) 1994-04-21
US5705520A (en) 1998-01-06
WO1992010477A1 (en) 1992-06-25
IE62894B1 (en) 1995-03-08
IS3790A7 (is) 1992-06-13
NZ240942A (en) 1994-03-25
CH684192A5 (fr) 1994-07-29
GB9126297D0 (en) 1992-02-12
PT99757B (pt) 1999-05-31
ES2069836T3 (es) 1995-05-16
EP0490689A1 (en) 1992-06-17
KR100211479B1 (ko) 1999-08-02
IS1706B (is) 1998-12-10
CZ114093A3 (en) 1994-02-16
YU48926B (sh) 2002-12-10
IL100330A (en) 1996-06-18
IL100330A0 (en) 1992-09-06
IT1252868B (it) 1995-06-28
FR2670487A1 (fr) 1992-06-19
GB2251614A (en) 1992-07-15
CA2098302C (en) 2001-10-16

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