DK0390558T3 - Aromatasehæmmende 4(5)-imidazoler - Google Patents

Aromatasehæmmende 4(5)-imidazoler

Info

Publication number
DK0390558T3
DK0390558T3 DK90303362.9T DK90303362T DK0390558T3 DK 0390558 T3 DK0390558 T3 DK 0390558T3 DK 90303362 T DK90303362 T DK 90303362T DK 0390558 T3 DK0390558 T3 DK 0390558T3
Authority
DK
Denmark
Prior art keywords
bond
chem
together form
halogen
imidazoles
Prior art date
Application number
DK90303362.9T
Other languages
English (en)
Inventor
Arto Johannes Karjalainen
Arja Leena Karjalainen
Reino Olavi Pelkonen
Marja-Liisa Sodervall
Matti Antero Lahde
Risto Arvo Sakari Lammintausta
Arja Marketta Kalapudas
Original Assignee
Orion Yhtymae Oy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB8907218A external-priority patent/GB2229719B/en
Priority claimed from GB8907309A external-priority patent/GB2231568B/en
Application filed by Orion Yhtymae Oy filed Critical Orion Yhtymae Oy
Application granted granted Critical
Publication of DK0390558T3 publication Critical patent/DK0390558T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Epoxy Resins (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Ceramic Products (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK90303362.9T 1989-03-30 1990-03-29 Aromatasehæmmende 4(5)-imidazoler DK0390558T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8907218A GB2229719B (en) 1989-03-30 1989-03-30 Novel aromatase inhibiting 4(5)-imidazoles
GB8907309A GB2231568B (en) 1989-03-31 1989-03-31 New aromatase inhibiting 4(5)-imidazoles

Publications (1)

Publication Number Publication Date
DK0390558T3 true DK0390558T3 (da) 1994-10-10

Family

ID=26295152

Family Applications (1)

Application Number Title Priority Date Filing Date
DK90303362.9T DK0390558T3 (da) 1989-03-30 1990-03-29 Aromatasehæmmende 4(5)-imidazoler

Country Status (19)

Country Link
EP (1) EP0390558B1 (da)
JP (1) JPH032168A (da)
CN (2) CN1046527A (da)
AT (1) ATE111084T1 (da)
AU (1) AU627559B2 (da)
CZ (1) CZ281611B6 (da)
DE (1) DE69012184T2 (da)
DK (1) DK0390558T3 (da)
ES (1) ES2063260T3 (da)
HU (2) HU206685B (da)
IE (1) IE64655B1 (da)
IL (1) IL93940A (da)
LV (1) LV11027B (da)
NO (1) NO172797C (da)
NZ (1) NZ233127A (da)
PL (1) PL162513B1 (da)
PT (1) PT93606B (da)
RU (1) RU1836354C (da)
UA (1) UA13471A (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2210875B (en) 1987-10-09 1991-05-29 Farmos Oy Aromatase inhibiting 4(5)-imidazoles
GB2229719B (en) 1989-03-30 1992-04-29 Farmos Oy Novel aromatase inhibiting 4(5)-imidazoles
GB2248058B (en) * 1990-09-21 1994-09-14 Orion Yhtymae Oy Aromatase inhibiting 4(5)-imidazoles
GB9125924D0 (en) * 1991-06-18 1992-02-05 Orion Yhtymae Oy Stereoisomers of an imidazole derivative
GB2273704B (en) * 1992-12-16 1997-01-22 Orion Yhtymae Oy Triazolyl diaryl selective aromatase inhibiting compounds
US7902247B2 (en) * 2008-01-09 2011-03-08 Allergan, Inc. Substituted-aryl-2-phenylethyl-1H-imidazole compounds as subtype selective modulators of alpha 2B and/or alpha 2C adrenergic receptors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2092569B (en) * 1981-02-05 1984-09-19 Farmos Oy Substituted imidazole derivatives and their preparation and use
GB2110663B (en) * 1981-12-04 1985-08-07 Farmos Group Ltd Imidazole derivatives
LU85747A1 (fr) * 1985-01-28 1986-08-04 Continental Pharma Derives d'imidazole leur preparation et utilisation ainsi que les compositions pharmaceutiques contenant des derives
GB2210875B (en) * 1987-10-09 1991-05-29 Farmos Oy Aromatase inhibiting 4(5)-imidazoles

Also Published As

Publication number Publication date
PT93606A (pt) 1990-11-20
IL93940A0 (en) 1990-12-23
NO172797C (no) 1993-09-08
CZ281611B6 (cs) 1996-11-13
DE69012184T2 (de) 1995-01-05
EP0390558A1 (en) 1990-10-03
AU5232590A (en) 1990-10-04
DE69012184D1 (de) 1994-10-13
IL93940A (en) 1994-10-07
NO901451D0 (no) 1990-03-29
PL284552A1 (en) 1991-07-29
ATE111084T1 (de) 1994-09-15
PT93606B (pt) 1996-08-30
CZ155590A3 (en) 1996-08-14
JPH032168A (ja) 1991-01-08
PL162513B1 (pl) 1993-12-31
UA13471A (uk) 1997-02-28
HU914010D0 (en) 1992-03-30
EP0390558B1 (en) 1994-09-07
CN1046527A (zh) 1990-10-31
CN1086812A (zh) 1994-05-18
LV11027B (en) 1996-08-20
IE64655B1 (en) 1995-08-23
NZ233127A (en) 1991-03-26
HU206685B (en) 1992-12-28
RU1836354C (ru) 1993-08-23
NO901451L (no) 1990-10-01
HU205345B (en) 1992-04-28
AU627559B2 (en) 1992-08-27
LV11027A (lv) 1996-02-20
ES2063260T3 (es) 1995-01-01
HUT53357A (en) 1990-10-28
HU901894D0 (en) 1990-08-28
NO172797B (no) 1993-06-01
IE901152L (en) 1990-09-30

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