DE69600620T2 - Arzneimittel mit gesteuerter wirkstofffreisetzung für basische schwerlösliche wirkstoffe - Google Patents

Arzneimittel mit gesteuerter wirkstofffreisetzung für basische schwerlösliche wirkstoffe

Info

Publication number
DE69600620T2
DE69600620T2 DE69600620T DE69600620T DE69600620T2 DE 69600620 T2 DE69600620 T2 DE 69600620T2 DE 69600620 T DE69600620 T DE 69600620T DE 69600620 T DE69600620 T DE 69600620T DE 69600620 T2 DE69600620 T2 DE 69600620T2
Authority
DE
Germany
Prior art keywords
medicinal products
substance release
active substance
active substances
controlled
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Revoked
Application number
DE69600620T
Other languages
English (en)
Other versions
DE69600620D1 (de
Inventor
Neville W Board
Alan F Carmody
Liam C Feely
Brian C Withers
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Laboratories
Original Assignee
Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24298013&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE69600620(T2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Publication of DE69600620D1 publication Critical patent/DE69600620D1/de
Application granted granted Critical
Publication of DE69600620T2 publication Critical patent/DE69600620T2/de
Anticipated expiration legal-status Critical
Revoked legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/02—Local antiseptics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE69600620T 1995-12-19 1996-11-25 Arzneimittel mit gesteuerter wirkstofffreisetzung für basische schwerlösliche wirkstoffe Revoked DE69600620T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/574,877 US5705190A (en) 1995-12-19 1995-12-19 Controlled release formulation for poorly soluble basic drugs
PCT/US1996/018960 WO1997022335A1 (en) 1995-12-19 1996-11-25 A controlled release formulation for poorly soluble basic drugs

Publications (2)

Publication Number Publication Date
DE69600620D1 DE69600620D1 (de) 1998-10-15
DE69600620T2 true DE69600620T2 (de) 1999-05-06

Family

ID=24298013

Family Applications (2)

Application Number Title Priority Date Filing Date
DE29624506U Expired - Lifetime DE29624506U1 (de) 1995-12-19 1996-11-25 Formulierung mit gesteuerter Wirkstofffreisetzung für schwerlösliche basische Wirkstoffe
DE69600620T Revoked DE69600620T2 (de) 1995-12-19 1996-11-25 Arzneimittel mit gesteuerter wirkstofffreisetzung für basische schwerlösliche wirkstoffe

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DE29624506U Expired - Lifetime DE29624506U1 (de) 1995-12-19 1996-11-25 Formulierung mit gesteuerter Wirkstofffreisetzung für schwerlösliche basische Wirkstoffe

Country Status (27)

Country Link
US (1) US5705190A (de)
EP (1) EP0799028B1 (de)
JP (1) JP3292732B2 (de)
KR (1) KR100632187B1 (de)
CN (1) CN1131027C (de)
AR (1) AR004391A1 (de)
AT (2) ATE170744T1 (de)
AU (1) AU701268B2 (de)
CA (1) CA2209714C (de)
CZ (1) CZ289158B6 (de)
DE (2) DE29624506U1 (de)
DK (1) DK0799028T3 (de)
ES (1) ES2122810T3 (de)
HK (1) HK1016873A1 (de)
HU (1) HUP9800516A3 (de)
IL (1) IL121275A (de)
IT (1) ITMI20050383U1 (de)
NZ (1) NZ323332A (de)
PL (1) PL186696B1 (de)
PT (1) PT103379B (de)
RO (1) RO117501B1 (de)
RU (1) RU2142793C1 (de)
TR (1) TR199800777T2 (de)
TW (1) TW429154B (de)
UA (1) UA40663C2 (de)
WO (1) WO1997022335A1 (de)
ZA (1) ZA9610110B (de)

Families Citing this family (100)

* Cited by examiner, † Cited by third party
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DE69600620D1 (de) 1998-10-15
UA40663C2 (uk) 2001-08-15
NZ323332A (en) 1998-04-27
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HUP9800516A3 (en) 2000-07-28
CA2209714A1 (en) 1997-06-26
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ZA9610110B (en) 1997-06-18
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HUP9800516A2 (hu) 1998-08-28
CA2209714C (en) 2002-07-30
EP0799028B1 (de) 1998-09-09
AT7918U1 (de) 2005-11-15
PT103379B (pt) 2007-02-28
EP0799028A1 (de) 1997-10-08
ATE170744T1 (de) 1998-09-15
RU2142793C1 (ru) 1999-12-20
ITMI20050383U1 (it) 2006-06-20
JP3292732B2 (ja) 2002-06-17
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