DE69230225D1 - Triazolylierte tertiäre aminverbindungen oder ihre salze - Google Patents

Triazolylierte tertiäre aminverbindungen oder ihre salze

Info

Publication number
DE69230225D1
DE69230225D1 DE69230225T DE69230225T DE69230225D1 DE 69230225 D1 DE69230225 D1 DE 69230225D1 DE 69230225 T DE69230225 T DE 69230225T DE 69230225 T DE69230225 T DE 69230225T DE 69230225 D1 DE69230225 D1 DE 69230225D1
Authority
DE
Germany
Prior art keywords
heterocyclic group
triazolylated
triazolyl
tertical
salts
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69230225T
Other languages
English (en)
Other versions
DE69230225T2 (de
Inventor
Minoru Okada
Eiji Kawaminami
Toru Yoden
Masafumi Kudou
Yasuo Isomura
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Astellas Pharma Inc
Original Assignee
Yamanouchi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yamanouchi Pharmaceutical Co Ltd filed Critical Yamanouchi Pharmaceutical Co Ltd
Application granted granted Critical
Publication of DE69230225D1 publication Critical patent/DE69230225D1/de
Publication of DE69230225T2 publication Critical patent/DE69230225T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Medicinal Preparation (AREA)
  • Treatments Of Macromolecular Shaped Articles (AREA)
  • Processes Of Treating Macromolecular Substances (AREA)
  • Cosmetics (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DE69230225T 1991-09-02 1992-08-27 Triazolylierte tertiäre aminverbindungen oder ihre salze Expired - Fee Related DE69230225T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP24826891 1991-09-02
JP34401191 1991-12-02
PCT/JP1992/001089 WO1993005027A1 (en) 1991-09-02 1992-08-27 Triazolylated tertiary amine compound or salt thereof

Publications (2)

Publication Number Publication Date
DE69230225D1 true DE69230225D1 (de) 1999-12-02
DE69230225T2 DE69230225T2 (de) 2000-05-31

Family

ID=26538684

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69230225T Expired - Fee Related DE69230225T2 (de) 1991-09-02 1992-08-27 Triazolylierte tertiäre aminverbindungen oder ihre salze

Country Status (20)

Country Link
US (1) US5674886A (de)
EP (1) EP0641785B1 (de)
KR (1) KR100204697B1 (de)
CN (1) CN1035817C (de)
AT (1) ATE186052T1 (de)
AU (1) AU665569B2 (de)
BG (1) BG61688B1 (de)
CA (1) CA2116773C (de)
DE (1) DE69230225T2 (de)
ES (1) ES2139605T3 (de)
FI (1) FI940988A (de)
HU (1) HU220863B1 (de)
MX (1) MX9204996A (de)
NO (1) NO305284B1 (de)
PT (1) PT100821B (de)
RO (1) RO114129B1 (de)
RU (1) RU2124010C1 (de)
TW (1) TW225526B (de)
UA (1) UA41295C2 (de)
WO (1) WO1993005027A1 (de)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5770616A (en) 1995-06-07 1998-06-23 The Procter & Gamble Company Pharmaceutical composition for inhibiting the growth of cancers
US7022702B2 (en) * 2000-04-07 2006-04-04 Qlt Inc. Antiproliferative 1,2,3-thiadiazole compounds
US6420400B1 (en) 2000-04-07 2002-07-16 Kinetek Pharmaceuticals, Inc. Antiproliferative 1,2,3-thiadiazole compounds
PT1355889E (pt) * 2000-12-22 2006-09-29 Ortho Mcneil Pharm Inc Derivados diamina triazole substituidos como inibidores de cinase
GB0120147D0 (en) * 2001-08-17 2001-10-10 Metris Therapeutics Ltd Treatment method
GB0127923D0 (en) * 2001-11-21 2002-01-16 Sterix Ltd Compound
MXPA04004802A (es) * 2001-11-21 2004-08-11 Sterix Ltd Derivados del 1,2,4-triazol que contienen un grupo sulfamato como inhibidores de aromatasa.
JP2004196795A (ja) * 2002-12-16 2004-07-15 Wyeth 外部寄生虫駆除剤としてのｎ−フェニル−３−シクロプロピルピラゾール−４−カルボニトリル
EP1431292A1 (de) * 2002-12-16 2004-06-23 Laboratoire Theramex 1-N-Phenylamino-1H-imidazolderivate und deren Verwendung als aromatase Inhibitoren
EP1544195A1 (de) * 2003-12-15 2005-06-22 Laboratoire Theramex 1-N-phenylamino-1H-imidazolderivate und sie enthaltende pharmazeutische Zusammensetzungen
CA2549603A1 (en) * 2003-12-15 2005-06-30 Laboratoire Theramex 1-n-phenyl-amino-1h-imidazole derivatives and pharmaceutical compositions containing them
AU2011226950B9 (en) * 2003-12-15 2013-04-11 Laboratoire Theramex 1-N-phenyl-amino-1H-imidazole derivatives and pharmaceutical compositions containing them
GB0411562D0 (en) * 2004-05-24 2004-06-23 Sterix Ltd Compound
WO2011002096A1 (ja) * 2009-07-03 2011-01-06 独立行政法人理化学研究所 Ｐｅｔ用標識化合物
GB0914767D0 (en) * 2009-08-24 2009-09-30 Sterix Ltd Compound
CN113387894B (zh) * 2021-06-22 2023-02-24 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 1-n-苯乙腈基氨基-三氮唑和嘧啶衍生物及其制备方法和应用

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4609666A (en) * 1984-06-18 1986-09-02 Eli Lilly And Company Aromatase inhibiting derivatives of α,α-bis(4-halophenyl)methyltetrazoles and triazoles
US4602025A (en) * 1984-06-18 1986-07-22 Eli Lilly And Company Aromatase inhibitors
US4749713A (en) 1986-03-07 1988-06-07 Ciba-Geigy Corporation Alpha-heterocycle substituted tolunitriles
CH677925A5 (de) * 1986-12-03 1991-07-15 Sandoz Ag
US5041458A (en) * 1987-03-20 1991-08-20 E. I. Du Pont De Nemours And Company Fungicidal aminotriazoles and aminoimidazoles
KR890700582A (ko) * 1987-03-20 1989-04-25 사무엘 에스. 블라이트 살진균성 아미노트리아졸 및 아미노이미다졸
NZ224714A (en) 1987-06-01 1990-03-27 Janssen Pharmaceutica Nv Substituted benzotriazole derivatives and pharmaceutical compositions
US4806554A (en) * 1988-01-11 1989-02-21 Hoechst-Roussel Pharmaceuticals, Inc. Pyrazol and indazolpyridinamines
GR900100380A (el) * 1989-05-20 1991-10-10 Fisons Plc Μέ?οδος παρασκευής αντι-φλεγμονωδών παραγώγων αμινοφενόλης.

Also Published As

Publication number Publication date
US5674886A (en) 1997-10-07
NO940686D0 (no) 1994-02-28
CN1035817C (zh) 1997-09-10
RO114129B1 (ro) 1999-01-29
AU2487492A (en) 1993-04-05
HUT67249A (en) 1995-03-28
HU220863B1 (en) 2002-06-29
BG98618A (bg) 1995-03-31
FI940988A0 (fi) 1994-03-02
NO305284B1 (no) 1999-05-03
EP0641785A4 (de) 1994-06-16
CN1069974A (zh) 1993-03-17
MX9204996A (es) 1993-08-01
FI940988A (fi) 1994-04-05
DE69230225T2 (de) 2000-05-31
CA2116773C (en) 2002-12-10
WO1993005027A1 (en) 1993-03-18
CA2116773A1 (en) 1993-03-18
UA41295C2 (uk) 2001-09-17
ES2139605T3 (es) 2000-02-16
RU2124010C1 (ru) 1998-12-27
PT100821B (pt) 1999-07-30
HU9400611D0 (en) 1994-09-28
NO940686L (de) 1994-04-29
TW225526B (de) 1994-06-21
PT100821A (pt) 1993-11-30
ATE186052T1 (de) 1999-11-15
KR100204697B1 (ko) 1999-06-15
AU665569B2 (en) 1996-01-11
BG61688B1 (bg) 1998-03-31
EP0641785B1 (de) 1999-10-27
EP0641785A1 (de) 1995-03-08

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8327 Change in the person/name/address of the patent owner

Owner name: ASTELLAS PHARMA INC., TOKIO/TOKYO, JP

8339 Ceased/non-payment of the annual fee