DE60225571D1 - Stabilisierung aktiver wirkstoffe durch formulierung als nanopartikuläre zusammensetzungen - Google Patents

Stabilisierung aktiver wirkstoffe durch formulierung als nanopartikuläre zusammensetzungen

Info

Publication number
DE60225571D1
DE60225571D1 DE60225571T DE60225571T DE60225571D1 DE 60225571 D1 DE60225571 D1 DE 60225571D1 DE 60225571 T DE60225571 T DE 60225571T DE 60225571 T DE60225571 T DE 60225571T DE 60225571 D1 DE60225571 D1 DE 60225571D1
Authority
DE
Germany
Prior art keywords
active agents
agents
nanoparticular
stabilization
formulation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60225571T
Other languages
English (en)
Other versions
DE60225571T2 (de
Inventor
Elaine Merisko-Liversidge
Linden Wei
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Elan Pharma International Ltd
Original Assignee
Elan Pharma International Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25492513&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE60225571(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Elan Pharma International Ltd filed Critical Elan Pharma International Ltd
Application granted granted Critical
Publication of DE60225571D1 publication Critical patent/DE60225571D1/de
Publication of DE60225571T2 publication Critical patent/DE60225571T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T428/00—Stock material or miscellaneous articles
    • Y10T428/29—Coated or structually defined flake, particle, cell, strand, strand portion, rod, filament, macroscopic fiber or mass thereof
    • Y10T428/2982—Particulate matter [e.g., sphere, flake, etc.]
    • Y10T428/2991—Coated

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Transplantation (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DE60225571T 2001-09-14 2002-09-13 Stabilisierung aktiver wirkstoffe durch formulierung als nanopartikuläre zusammensetzungen Expired - Lifetime DE60225571T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US09/952,032 US20030054042A1 (en) 2001-09-14 2001-09-14 Stabilization of chemical compounds using nanoparticulate formulations
US952032 2001-09-14
PCT/US2002/025979 WO2003024424A1 (en) 2001-09-14 2002-09-13 Stabilization of active agents by formulation into nanoparticulate form

Publications (2)

Publication Number Publication Date
DE60225571D1 true DE60225571D1 (de) 2008-04-24
DE60225571T2 DE60225571T2 (de) 2009-04-23

Family

ID=25492513

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60225571T Expired - Lifetime DE60225571T2 (de) 2001-09-14 2002-09-13 Stabilisierung aktiver wirkstoffe durch formulierung als nanopartikuläre zusammensetzungen

Country Status (11)

Country Link
US (4) US20030054042A1 (de)
EP (2) EP1427395B1 (de)
JP (2) JP2005505568A (de)
AT (1) ATE388690T1 (de)
CA (1) CA2460436C (de)
CY (1) CY1108130T1 (de)
DE (1) DE60225571T2 (de)
DK (1) DK1427395T3 (de)
ES (1) ES2303553T3 (de)
PT (1) PT1427395E (de)
WO (1) WO2003024424A1 (de)

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PT1427395E (pt) 2008-05-20
JP2010280687A (ja) 2010-12-16
EP1427395B1 (de) 2008-03-12
EP1427395A1 (de) 2004-06-16
WO2003024424A1 (en) 2003-03-27
EP1829530A3 (de) 2009-05-06
CY1108130T1 (el) 2014-02-12
EP1829530A2 (de) 2007-09-05
CA2460436C (en) 2011-05-10
DE60225571T2 (de) 2009-04-23
ES2303553T3 (es) 2008-08-16
ATE388690T1 (de) 2008-03-15
CA2460436A1 (en) 2003-03-27
DK1427395T3 (da) 2008-06-30
US20030054042A1 (en) 2003-03-20
US20120087984A1 (en) 2012-04-12
US20090175951A1 (en) 2009-07-09
US20070224279A1 (en) 2007-09-27

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