DE60221569T2 - Acrylsulfonamidderivate zur verwendung als ccr3-antagonisten bei der behandlung von inflammatorischen und immunologischen erkrankungen - Google Patents

Acrylsulfonamidderivate zur verwendung als ccr3-antagonisten bei der behandlung von inflammatorischen und immunologischen erkrankungen Download PDF

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DE60221569T2
DE60221569T2 DE60221569T DE60221569T DE60221569T2 DE 60221569 T2 DE60221569 T2 DE 60221569T2 DE 60221569 T DE60221569 T DE 60221569T DE 60221569 T DE60221569 T DE 60221569T DE 60221569 T2 DE60221569 T2 DE 60221569T2
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straight
hydrogen
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alkyl
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DE60221569D1 (de
Inventor
Yingfu Nara-shi LI
Akihiko Watanabe
Timothy B. Lowinger
Kevin Bacon
Norihiro Nara-shi KAWAMURA
Takuya Soraku-gun SHINTANI
Tetsuo Nara-shi KIKUCHI
Toshiya Ikoma-shi MORIWAKI
Klaus Kobe-shi URBAHNS
Keiko Saitama-ken FUKUSHIMA
Noriko Nara-shi NUNAMI
Takashi Shiga-ken YOSHINO
Toshiki Ikoma-shi MURATA
Megumi Shiga-ken YAMAUCHI
Hiroko Shiga-ken YOSHINO
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Axikin Pharmaceuticals Inc
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Actimis Pharmaceuticals Inc
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    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
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    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
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DE60221569T 2001-09-07 2002-09-04 Acrylsulfonamidderivate zur verwendung als ccr3-antagonisten bei der behandlung von inflammatorischen und immunologischen erkrankungen Expired - Lifetime DE60221569T2 (de)

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