DE3025579A1 - Aryl-1-arylsulfonyl-4 gamma -aminopropoxy-3-1h-pyrazole, verfahren zu ihrer herstellung und sie enthaltende mittel - Google Patents

Aryl-1-arylsulfonyl-4 gamma -aminopropoxy-3-1h-pyrazole, verfahren zu ihrer herstellung und sie enthaltende mittel

Info

Publication number
DE3025579A1
DE3025579A1 DE19803025579 DE3025579A DE3025579A1 DE 3025579 A1 DE3025579 A1 DE 3025579A1 DE 19803025579 DE19803025579 DE 19803025579 DE 3025579 A DE3025579 A DE 3025579A DE 3025579 A1 DE3025579 A1 DE 3025579A1
Authority
DE
Germany
Prior art keywords
formula
radical
aryl
arylsulfonyl
reaction
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
DE19803025579
Other languages
German (de)
English (en)
Inventor
Gilles Monnier
Marcel Pesson
Henri Techer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Laboratoire Roger Bellon SA
Original Assignee
Laboratoire Roger Bellon SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratoire Roger Bellon SA filed Critical Laboratoire Roger Bellon SA
Publication of DE3025579A1 publication Critical patent/DE3025579A1/de
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/28—Two oxygen or sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DE19803025579 1979-07-05 1980-07-05 Aryl-1-arylsulfonyl-4 gamma -aminopropoxy-3-1h-pyrazole, verfahren zu ihrer herstellung und sie enthaltende mittel Withdrawn DE3025579A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7917507A FR2460299A1 (fr) 1979-07-05 1979-07-05 Nouveaux derives du pyrazole et leur application therapeutique

Publications (1)

Publication Number Publication Date
DE3025579A1 true DE3025579A1 (de) 1981-01-15

Family

ID=9227565

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19803025579 Withdrawn DE3025579A1 (de) 1979-07-05 1980-07-05 Aryl-1-arylsulfonyl-4 gamma -aminopropoxy-3-1h-pyrazole, verfahren zu ihrer herstellung und sie enthaltende mittel

Country Status (10)

Country Link
US (1) US4337263A (enExample)
JP (1) JPS5615271A (enExample)
BE (1) BE884189A (enExample)
CA (1) CA1152507A (enExample)
DE (1) DE3025579A1 (enExample)
ES (1) ES8102561A1 (enExample)
FR (1) FR2460299A1 (enExample)
GB (2) GB2063870B (enExample)
IT (1) IT8068062A0 (enExample)
NL (1) NL8003888A (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1994013643A1 (en) * 1992-12-17 1994-06-23 Pfizer Inc. Pyrazoles and pyrazolopyrimidines having crf antagonist activity
EP0691128A1 (en) * 1994-06-15 1996-01-10 Pfizer Inc. Methods of administering CRF antagonists

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA857592B (en) * 1984-10-17 1986-05-28 Heumann Ludwig & Co Gmbh Pyrazole derivatives,processes for their preparation and pharmaceutical preparations containing these compounds
US4964895A (en) * 1987-06-08 1990-10-23 Monsanto Company Substituted 4-(4-nitrophenoxy) pyrazoles and their use as herbicides
US6005109A (en) * 1997-10-30 1999-12-21 Pflizer Inc. Pyrazoles and pyrazolopyrimidines having CRF antagonistic activity
US6103900A (en) * 1992-12-17 2000-08-15 Pfizer Inc Pyrazoles and pyrazolopyrimidines having CRF antagonistic activity
EP1634872A1 (en) * 2004-08-27 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Pyrazole derivatives as sigma receptor inhibitors
US7696199B2 (en) * 2004-08-27 2010-04-13 Laboratorios Del Dr. Esteve, S.A. Sigma receptor inhibitors
MX2007002341A (es) * 2004-08-27 2007-09-25 Esteve Labor Dr Inhibidores del receptor sigma.
WO2007098953A1 (en) * 2006-03-01 2007-09-07 Laboratorios Del Dr. Esteve, S.A. Pyrazole derivatives as sigma receptor inhibitors
EP1829875A1 (en) 2006-03-01 2007-09-05 Laboratorios Del Dr. Esteve, S.A. Pyrazole derivatives as sigma receptor inhibitors
EP1829866A1 (en) * 2006-03-02 2007-09-05 Laboratorios Del Dr. Esteve, S.A. Sigma receptor inhibitors
EP1829867A1 (en) 2006-03-03 2007-09-05 Laboratorios Del Dr. Esteve, S.A. Imidazole compounds having pharmaceutical activity towards the sigma receptor
EP2529793B1 (en) * 2007-06-08 2016-08-10 Georgia State University Research Foundation, Inc. Compositions for regulating or modulating quorum sensing in bacteria, methods of using the compounds, and methods of regulating or modulating quorum sensing in bacteria
EP2116539A1 (en) 2008-04-25 2009-11-11 Laboratorios Del. Dr. Esteve, S.A. 1-aryl-3-aminoalkoxy-pyrazoles as sigma ligands enhancing analgesic effects of opioids and attenuating the dependency thereof
EP2353591A1 (en) 2010-02-04 2011-08-10 Laboratorios Del. Dr. Esteve, S.A. Sigma ligands for potentiating the analgesic effect of opioids and opiates in post-operative pain and attenuating the dependency thereof
EP2388005A1 (en) 2010-05-21 2011-11-23 Laboratorios Del. Dr. Esteve, S.A. Sigma ligands for the prevention and/or treatment of emesis induced by chemotherapy or radiotherapy
EP2395003A1 (en) 2010-05-27 2011-12-14 Laboratorios Del. Dr. Esteve, S.A. Pyrazole compounds as sigma receptor inhibitors
EP2415471A1 (en) 2010-08-03 2012-02-08 Laboratorios Del. Dr. Esteve, S.A. Use of sigma ligands in opioid-induced hyperalgesia
EP2524694A1 (en) 2011-05-19 2012-11-21 Laboratorios Del. Dr. Esteve, S.A. Use of sigma ligands in diabetes type-2 associated pain
TW201607538A (zh) 2013-12-17 2016-03-01 以斯提夫博士實驗室股份有限公司 血清素－去甲腎上腺素再攝取抑制劑（ＳＮＲＩＳ）和σ受體配體組合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI34517A (fi) 1962-12-08 1964-10-10 Laeaeketehdas Orion Oy 5-pyratsolyylialkamiinieetterien valmistusmenetelmä
JPS4832112B1 (enExample) * 1969-10-03 1973-10-04
DE2409753A1 (de) * 1974-03-01 1975-09-11 Basf Ag Substituierte pyrazole
FR2301250A1 (fr) 1975-02-21 1976-09-17 Bellon Labor Sa Roger Nouveaux diaryl-1, 4o-aminoalcoxy-3 pyrazoles et leurs sels

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1994013643A1 (en) * 1992-12-17 1994-06-23 Pfizer Inc. Pyrazoles and pyrazolopyrimidines having crf antagonist activity
EP0691128A1 (en) * 1994-06-15 1996-01-10 Pfizer Inc. Methods of administering CRF antagonists

Also Published As

Publication number Publication date
JPS5615271A (en) 1981-02-14
IT8068062A0 (it) 1980-07-04
NL8003888A (nl) 1981-01-07
GB2063870B (en) 1983-06-22
US4337263A (en) 1982-06-29
GB2054566A (en) 1981-02-18
GB2054566B (en) 1983-05-18
CA1152507A (fr) 1983-08-23
GB2063870A (en) 1981-06-10
ES492986A0 (es) 1981-02-16
BE884189A (fr) 1981-01-05
ES8102561A1 (es) 1981-02-16
FR2460299B1 (enExample) 1983-01-14
FR2460299A1 (fr) 1981-01-23

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Legal Events

Date Code Title Description
8139 Disposal/non-payment of the annual fee