DE2901362A1 - Guanidinderivate, ihre herstellung und verwendung - Google Patents

Guanidinderivate, ihre herstellung und verwendung

Info

Publication number
DE2901362A1
DE2901362A1 DE19792901362 DE2901362A DE2901362A1 DE 2901362 A1 DE2901362 A1 DE 2901362A1 DE 19792901362 DE19792901362 DE 19792901362 DE 2901362 A DE2901362 A DE 2901362A DE 2901362 A1 DE2901362 A1 DE 2901362A1
Authority
DE
Germany
Prior art keywords
formula
carbon atoms
compounds
alkyl
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
DE19792901362
Other languages
German (de)
English (en)
Inventor
Peter Dr Neumann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sandoz AG
Original Assignee
Sandoz AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz AG filed Critical Sandoz AG
Publication of DE2901362A1 publication Critical patent/DE2901362A1/de
Withdrawn legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/42Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms with nitro or nitroso radicals directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/22Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/28Halogen atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Furan Compounds (AREA)
  • Pyrrole Compounds (AREA)
DE19792901362 1978-01-25 1979-01-15 Guanidinderivate, ihre herstellung und verwendung Withdrawn DE2901362A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH79978 1978-01-25

Publications (1)

Publication Number Publication Date
DE2901362A1 true DE2901362A1 (de) 1979-07-26

Family

ID=4195448

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19792901362 Withdrawn DE2901362A1 (de) 1978-01-25 1979-01-15 Guanidinderivate, ihre herstellung und verwendung

Country Status (12)

Country Link
JP (1) JPS54112859A (it)
AU (1) AU4359279A (it)
BE (1) BE873658A (it)
DE (1) DE2901362A1 (it)
FR (1) FR2415636A1 (it)
GB (1) GB2013192A (it)
IE (1) IE790126L (it)
IL (1) IL56486A0 (it)
IT (1) IT7947732A0 (it)
NL (1) NL7900444A (it)
SE (1) SE7900459L (it)
ZA (1) ZA79315B (it)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20060459A1 (es) 2004-06-16 2006-05-30 Wyeth Corp DERIVADOS DE AMINO-5,5-DIFENILIMIDAZOLONA COMO INHIBIDORES DE LA ß-SECRETASA
AU2005264917A1 (en) 2004-06-16 2006-01-26 Wyeth Diphenylimidazopyrimidine and -imidazole amines as inhibitors of B-secretase
CN101103034A (zh) 2005-01-14 2008-01-09 惠氏公司 抑制β-分泌酶的氨基-咪唑酮
WO2006083760A1 (en) 2005-02-01 2006-08-10 Wyeth AMINO-PYRIDINES AS INHIBITORS OF β-SECRETASE
WO2006088694A1 (en) 2005-02-14 2006-08-24 Wyeth SUBSTITUTED THIENYL AND FURYL ACYLGUANIDINES AS β-SECRETASE MODULATORS
CN101146769A (zh) 2005-02-14 2008-03-19 惠氏公司 作为β-分泌酶抑制剂的唑基酰基胍
WO2007005404A1 (en) 2005-06-30 2007-01-11 Wyeth AMINO-5-(6-MEMBERED)HETEROARYLIMIDAZOLONE COMPOUNDS AND THE USE THEREOF FOR ß-SECRETASE MODULATION
TW200738683A (en) 2005-06-30 2007-10-16 Wyeth Corp Amino-5-(5-membered)heteroarylimidazolone compounds and the use thereof for β-secretase modulation
EP2256107A1 (en) 2005-09-26 2010-12-01 Wyeth LLC Amino-5-[4-(difluoromethoxy)phenyl]-5-phenylimidazolone compounds as inhibitors of the beta-secretase (BACE)
WO2007100536A1 (en) 2006-02-24 2007-09-07 Wyeth DIHYDROSPIRO[DIBENZO[A,D][7]ANNULENE-5,4'-IMIDAZOL] COMPOUNDS FOR THE INHIBITION OF β-SECRETASE
US7700606B2 (en) 2006-08-17 2010-04-20 Wyeth Llc Imidazole amines as inhibitors of β-secretase
PE20090617A1 (es) 2007-03-23 2009-05-08 Wyeth Corp Compuestos amino-5-[-4-(difluorometoxi)fenil]-5-fenilimidazolona para la inhibicion de -secretasa

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1298112A (en) * 1969-02-20 1972-11-29 Wander Ag Dr A Phenyl acetyl guanidine derivatives

Also Published As

Publication number Publication date
IT7947732A0 (it) 1979-01-23
BE873658A (fr) 1979-07-23
JPS54112859A (en) 1979-09-04
ZA79315B (en) 1980-09-24
AU4359279A (en) 1979-08-02
NL7900444A (nl) 1979-07-27
GB2013192A (en) 1979-08-08
SE7900459L (sv) 1979-07-26
FR2415636A1 (fr) 1979-08-24
IL56486A0 (en) 1979-03-12
IE790126L (en) 1979-07-25

Similar Documents

Publication Publication Date Title
DE2614406C2 (it)
CH649527A5 (de) 1,2-diaminocyclobuten-3,4-dione, verfahren zu deren herstellung und pharmazeutische mittel, die diese verbindungen enthalten.
DE2901362A1 (de) Guanidinderivate, ihre herstellung und verwendung
DE60304599T2 (de) Pyridopyrimidinon-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen
EP0496238A1 (de) Substituierte Benzoxazepine und Benzthiazepine, Verfahren zu ihrer Herstellung und ihre Verwendung in Arzneimitteln
DE1620329B2 (de) 8-halogen-10-piperazino-10,11-dihydrobenzo (b,f) thiepinderivate und verfahren zu deren herstellung
CH649553A5 (de) Azepinoindole und verfahren zu deren herstellung.
DE2006895A1 (de) Neue Phenacetylguanidine und Verfahren zu ihrer Herstellung
DE2748920A1 (de) 3-fluor-morphanthridine, ihre herstellung und verwendung
DE2845857C2 (de) Benzo [d] thiazolderivate, Verfahren zu ihrer Herstellung und sie enthaltende Arzneimittelzubereitungen
CH632268A5 (de) Verfahren zur herstellung von neuen heterocyclylaminoderivaten.
AT391316B (de) Neue thienyloxy-alkylamin-derivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE2557792A1 (de) Neue heterocyclische verbindungen, ihre herstellung und ihre verwendung
DE1468135A1 (de) Organische Amine und Verfahren zu deren Herstellung
DE2755045A1 (de) Dicarboximidamide und deren salze, verfahren zu ihrer herstellung und ihre verwendung bei der bekaempfung von entzuendungen
DE2633782A1 (de) Neue organische verbindungen, ihre herstellung und verwendung
EP0160173A1 (de) Benzothiazolderivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltendes Arzneimittel
DE2321786C2 (de) S↑IV↑ -Benzo-1,2,4-thiadiazine
AT317227B (de) Verfahren zur Herstellung von neuen 4-Amino-6,7,8-trialkoxy-chinazolinen und deren Salzen
DE2222931C3 (de) Piperidinoalkylphenthiazine, Verfahren zur Herstellung derselben sowie diese enthaltende pharmazeutische Mittel
AT321302B (de) Verfahren zur Herstellung von neuen Aminophenylketonderivaten und ihren Säureadditionssalzen
DE1937629B2 (de) Nitrofuryl-aminoalkoxy-pyrimidine
DE2445335A1 (de) Neue organische verbindungen und verfahren zu deren herstellung
AT359492B (de) Verfahren zur herstellung neuer indazolderivate und ihrer salze
AT337181B (de) Verfahren zur herstellung neuer 4-(4-piperidyliden)-4h-benzo(4,5)cyclohepta(1,2-b)thiophen-derivate und ihrer saureadditionssalze

Legal Events

Date Code Title Description
8139 Disposal/non-payment of the annual fee