DE2623377A1 - 2-imidazoline und ihre anwendung in pharmazeutischen zubereitungen sowie verfahren zu ihrer herstellung - Google Patents

2-imidazoline und ihre anwendung in pharmazeutischen zubereitungen sowie verfahren zu ihrer herstellung

Info

Publication number
DE2623377A1
DE2623377A1 DE19762623377 DE2623377A DE2623377A1 DE 2623377 A1 DE2623377 A1 DE 2623377A1 DE 19762623377 DE19762623377 DE 19762623377 DE 2623377 A DE2623377 A DE 2623377A DE 2623377 A1 DE2623377 A1 DE 2623377A1
Authority
DE
Germany
Prior art keywords
imidazoline
group
lower alkyl
methyl
hydrogen atom
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19762623377
Other languages
German (de)
English (en)
Inventor
Heide Roebke
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
MSD International Holdings GmbH
Original Assignee
Scherico Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/582,313 external-priority patent/US3992403A/en
Application filed by Scherico Ltd filed Critical Scherico Ltd
Publication of DE2623377A1 publication Critical patent/DE2623377A1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/02—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms with only carbon-to-carbon double bonds as unsaturation
    • C07C57/13—Dicarboxylic acids
    • C07C57/15—Fumaric acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/02—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms with only carbon-to-carbon double bonds as unsaturation
    • C07C57/13—Dicarboxylic acids
    • C07C57/145—Maleic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/06—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/20—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with substituted hydrocarbon radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DE19762623377 1975-05-30 1976-05-25 2-imidazoline und ihre anwendung in pharmazeutischen zubereitungen sowie verfahren zu ihrer herstellung Pending DE2623377A1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US58231275A 1975-05-30 1975-05-30
US05/582,313 US3992403A (en) 1975-05-30 1975-05-30 2-Imidazolines and their use as hypoglycemic agents

Publications (1)

Publication Number Publication Date
DE2623377A1 true DE2623377A1 (de) 1976-12-09

Family

ID=27078537

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19762623377 Pending DE2623377A1 (de) 1975-05-30 1976-05-25 2-imidazoline und ihre anwendung in pharmazeutischen zubereitungen sowie verfahren zu ihrer herstellung

Country Status (9)

Country Link
JP (1) JPS51143668A (enExample)
AU (1) AU1432676A (enExample)
DE (1) DE2623377A1 (enExample)
DK (1) DK229376A (enExample)
FR (1) FR2312244A1 (enExample)
IL (1) IL49664A0 (enExample)
LU (1) LU75035A1 (enExample)
NL (1) NL7605609A (enExample)
SE (1) SE7605958L (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0552631A1 (de) * 1992-01-23 1993-07-28 Bayer Ag Alpha-Aryl-alpha-hydroxy-beta-imidazolinylpropionsäureamide

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2096987B (en) * 1981-04-22 1984-04-04 Farmos Oy Substituted imidazole and imidazole derivatives and their preparation and use
US6410562B1 (en) 1998-12-18 2002-06-25 Eli Lilly And Company Hypoglycemic imidazoline compounds
EP1981499A1 (en) * 2006-01-27 2008-10-22 F.Hoffmann-La Roche Ag Use of 2-imidazoles for the treatment of cns disorders

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2919274A (en) * 1957-09-17 1959-12-29 Sahyun Melville Amidines
GB877306A (en) * 1958-04-21 1961-09-13 Pfizer & Co C Halogenated derivatives of tetrahydro-1-naphthyl cyclic amidines
GB1417174A (en) * 1972-11-30 1975-12-10 Hexachimie 1-2-delta2-imidazolinyl-2,2-diarylcoclopropanes

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0552631A1 (de) * 1992-01-23 1993-07-28 Bayer Ag Alpha-Aryl-alpha-hydroxy-beta-imidazolinylpropionsäureamide

Also Published As

Publication number Publication date
FR2312244A1 (fr) 1976-12-24
AU1432676A (en) 1977-12-01
IL49664A0 (en) 1976-07-30
LU75035A1 (enExample) 1977-02-15
DK229376A (da) 1976-12-01
FR2312244B1 (enExample) 1979-09-21
JPS51143668A (en) 1976-12-10
SE7605958L (sv) 1976-12-01
NL7605609A (nl) 1976-12-02

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