DE2540134C3 - L-Phenylalaninderivate, Verfahren zu ihrer Herstellung und ihre Verwendung - Google Patents

L-Phenylalaninderivate, Verfahren zu ihrer Herstellung und ihre Verwendung

Info

Publication number
DE2540134C3
DE2540134C3 DE2540134A DE2540134A DE2540134C3 DE 2540134 C3 DE2540134 C3 DE 2540134C3 DE 2540134 A DE2540134 A DE 2540134A DE 2540134 A DE2540134 A DE 2540134A DE 2540134 C3 DE2540134 C3 DE 2540134C3
Authority
DE
Germany
Prior art keywords
product
phenylalanine
guanidino
methanol
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE2540134A
Other languages
German (de)
English (en)
Other versions
DE2540134A1 (de
DE2540134B2 (de
Inventor
Yakir Klausner
Pierre Lefrancier
Meir Rigbi
Edgar Sache
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Choay SA
Yissum Research Development Co of Hebrew University of Jerusalem
Original Assignee
Choay SA
Yissum Research Development Co of Hebrew University of Jerusalem
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Choay SA, Yissum Research Development Co of Hebrew University of Jerusalem filed Critical Choay SA
Publication of DE2540134A1 publication Critical patent/DE2540134A1/de
Publication of DE2540134B2 publication Critical patent/DE2540134B2/de
Application granted granted Critical
Publication of DE2540134C3 publication Critical patent/DE2540134C3/de
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/45—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups at least one of the singly-bound nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfonamides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Investigating Or Analyzing Non-Biological Materials By The Use Of Chemical Means (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
DE2540134A 1974-09-09 1975-09-09 L-Phenylalaninderivate, Verfahren zu ihrer Herstellung und ihre Verwendung Expired DE2540134C3 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7430509A FR2283888A1 (fr) 1974-09-09 1974-09-09 Nouveaux derives de la phenylalanine

Publications (3)

Publication Number Publication Date
DE2540134A1 DE2540134A1 (de) 1976-03-25
DE2540134B2 DE2540134B2 (de) 1978-03-30
DE2540134C3 true DE2540134C3 (de) 1978-11-23

Family

ID=9142895

Family Applications (1)

Application Number Title Priority Date Filing Date
DE2540134A Expired DE2540134C3 (de) 1974-09-09 1975-09-09 L-Phenylalaninderivate, Verfahren zu ihrer Herstellung und ihre Verwendung

Country Status (6)

Country Link
US (1) US4118575A (Direct)
JP (1) JPS5152152A (Direct)
CH (2) CH612930A5 (Direct)
DE (1) DE2540134C3 (Direct)
FR (1) FR2283888A1 (Direct)
GB (2) GB1526557A (Direct)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10005631A1 (de) 2000-02-09 2001-08-23 Max Planck Gesellschaft Arginin-Mimetika als Faktor X¶a¶-Inhibitoren

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3622615A (en) * 1968-11-06 1971-11-23 Parke Davis & Co N{11 -(p-tolylsulfonyl)-L-arginine esters
GB1268867A (en) * 1969-07-24 1972-03-29 Sumitomo Chemical Co THE PREPARATION OF D-THREO-beta-p-METHYLSULPHONYLPHENYLSERINE ESTER
CH553161A (de) * 1970-10-30 1974-08-30 Hoffmann La Roche Verfahren zur herstellung von phenylalaninderivaten.

Also Published As

Publication number Publication date
JPS5152152A (en) 1976-05-08
CH615903A5 (Direct) 1980-02-29
FR2283888B1 (Direct) 1979-03-09
FR2283888A1 (fr) 1976-04-02
GB1526557A (en) 1978-09-27
CH612930A5 (Direct) 1979-08-31
DE2540134A1 (de) 1976-03-25
GB1526558A (en) 1978-09-27
DE2540134B2 (de) 1978-03-30
US4118575A (en) 1978-10-03

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Legal Events

Date Code Title Description
C3 Grant after two publication steps (3rd publication)
8339 Ceased/non-payment of the annual fee