DE2454805A1 - Acylderivate - Google Patents

Acylderivate

Info

Publication number
DE2454805A1
DE2454805A1 DE19742454805 DE2454805A DE2454805A1 DE 2454805 A1 DE2454805 A1 DE 2454805A1 DE 19742454805 DE19742454805 DE 19742454805 DE 2454805 A DE2454805 A DE 2454805A DE 2454805 A1 DE2454805 A1 DE 2454805A1
Authority
DE
Germany
Prior art keywords
acid addition
glycyl
formula
ohh
hydrogen atom
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19742454805
Other languages
German (de)
English (en)
Inventor
Roland Dr Reiner
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of DE2454805A1 publication Critical patent/DE2454805A1/de
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/095—Sulfur, selenium, or tellurium compounds, e.g. thiols
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/095—Sulfur, selenium, or tellurium compounds, e.g. thiols
    • A61K31/10—Sulfides; Sulfoxides; Sulfones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/485—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C313/00—Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C315/00—Preparation of sulfones; Preparation of sulfoxides
    • C07C315/04—Preparation of sulfones; Preparation of sulfoxides by reactions not involving the formation of sulfone or sulfoxide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/26—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C317/32—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Emergency Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Inorganic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DE19742454805 1973-11-22 1974-11-19 Acylderivate Pending DE2454805A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH1646873A CH589617A5 (enExample) 1973-11-22 1973-11-22

Publications (1)

Publication Number Publication Date
DE2454805A1 true DE2454805A1 (de) 1975-05-28

Family

ID=4417636

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19742454805 Pending DE2454805A1 (de) 1973-11-22 1974-11-19 Acylderivate

Country Status (13)

Country Link
JP (1) JPS5083347A (enExample)
AT (1) AT338764B (enExample)
BE (1) BE822446A (enExample)
CH (1) CH589617A5 (enExample)
DE (1) DE2454805A1 (enExample)
DK (1) DK606074A (enExample)
FR (1) FR2252092B1 (enExample)
GB (1) GB1433977A (enExample)
HU (1) HU170835B (enExample)
IL (1) IL45776A (enExample)
NL (1) NL7413346A (enExample)
SE (1) SE7414606L (enExample)
ZA (1) ZA746222B (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0224902A1 (de) * 1985-12-05 1987-06-10 Roche Diagnostics GmbH Verbesserte Verfahren zur Herstellung von D-threo-1-(p-Methylsulfonylphenyl)-2-dichloracetamido-propandiol-1,3-(Thiamphenicol)sowie Verwendung geeigneter Zwischenprodukte
US5336664A (en) * 1990-04-24 1994-08-09 Zambon Group S.P.A. Compositions having herbicidal activity containing N-alkyl-amides as active ingredient

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0224902A1 (de) * 1985-12-05 1987-06-10 Roche Diagnostics GmbH Verbesserte Verfahren zur Herstellung von D-threo-1-(p-Methylsulfonylphenyl)-2-dichloracetamido-propandiol-1,3-(Thiamphenicol)sowie Verwendung geeigneter Zwischenprodukte
US4945181A (en) * 1985-12-05 1990-07-31 Boehringer Mannheim Gmbh Method for resolution of racemic thiamphenicol precursors and intermediates therefor
US5336664A (en) * 1990-04-24 1994-08-09 Zambon Group S.P.A. Compositions having herbicidal activity containing N-alkyl-amides as active ingredient
US5556829A (en) * 1990-04-24 1996-09-17 Zambon Group S.P.A. Compositions having herbicidal activity containing N-alkyl-amides as active ingredient

Also Published As

Publication number Publication date
AT338764B (de) 1977-09-12
HU170835B (hu) 1977-09-28
CH589617A5 (enExample) 1977-07-15
SE7414606L (enExample) 1975-05-23
JPS5083347A (enExample) 1975-07-05
IL45776A (en) 1977-12-30
ZA746222B (en) 1975-11-26
GB1433977A (en) 1976-04-28
FR2252092A1 (enExample) 1975-06-20
BE822446A (fr) 1975-05-21
ATA933274A (de) 1977-01-15
IL45776A0 (en) 1974-12-31
AU7408074A (en) 1976-04-15
FR2252092B1 (enExample) 1978-07-28
DK606074A (enExample) 1975-07-21
NL7413346A (nl) 1975-05-26

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Legal Events

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