DE19542499A1 - Verfahren und Vorrichtung zur Herstellung einer parenteralen Arzneistoffzubereitung - Google Patents

Verfahren und Vorrichtung zur Herstellung einer parenteralen Arzneistoffzubereitung

Info

Publication number
DE19542499A1
DE19542499A1 DE19542499A DE19542499A DE19542499A1 DE 19542499 A1 DE19542499 A1 DE 19542499A1 DE 19542499 A DE19542499 A DE 19542499A DE 19542499 A DE19542499 A DE 19542499A DE 19542499 A1 DE19542499 A1 DE 19542499A1
Authority
DE
Germany
Prior art keywords
dispersion
nozzle
homogenizing
bar
homogenizing nozzle
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
DE19542499A
Other languages
German (de)
English (en)
Inventor
Bernd Dipl Ing Klinksiek
Said Dr Mahiout
Ricarda Dipl Ing Nothelle
Hans Juergen Dr Hamann
Juergen Dipl Ing Sdebik
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Priority to DE19542499A priority Critical patent/DE19542499A1/de
Priority to JP51854497A priority patent/JP4049391B2/ja
Priority to ES96938066T priority patent/ES2180807T3/es
Priority to CA002237554A priority patent/CA2237554C/en
Priority to PT96938066T priority patent/PT861068E/pt
Priority to DK96938066T priority patent/DK0861068T3/da
Priority to EP96938066A priority patent/EP0861068B1/de
Priority to US09/068,812 priority patent/US6331314B1/en
Priority to AT96938066T priority patent/ATE222097T1/de
Priority to DE59609564T priority patent/DE59609564D1/de
Priority to PCT/EP1996/004795 priority patent/WO1997017946A2/de
Publication of DE19542499A1 publication Critical patent/DE19542499A1/de
Priority to MX9803633A priority patent/MX9803633A/es
Withdrawn legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/44221,4-Dihydropyridines, e.g. nifedipine, nicardipine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
    • A61K9/1277Preparation processes; Proliposomes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B01PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01FMIXING, e.g. DISSOLVING, EMULSIFYING OR DISPERSING
    • B01F25/00Flow mixers; Mixers for falling materials, e.g. solid particles
    • B01F25/40Static mixers
    • B01F25/46Homogenising or emulsifying nozzles
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B01PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01FMIXING, e.g. DISSOLVING, EMULSIFYING OR DISPERSING
    • B01F33/00Other mixers; Mixing plants; Combinations of mixers
    • B01F33/70Mixers specially adapted for working at sub- or super-atmospheric pressure, e.g. combined with de-foaming
    • B01F33/71Mixers specially adapted for working at sub- or super-atmospheric pressure, e.g. combined with de-foaming working at super-atmospheric pressure, e.g. in pressurised vessels
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10TTECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T428/00Stock material or miscellaneous articles
    • Y10T428/29Coated or structually defined flake, particle, cell, strand, strand portion, rod, filament, macroscopic fiber or mass thereof
    • Y10T428/2982Particulate matter [e.g., sphere, flake, etc.]
    • Y10T428/2984Microcapsule with fluid core [includes liposome]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Dispersion Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Manufacturing Of Micro-Capsules (AREA)
  • Medical Preparation Storing Or Oral Administration Devices (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
DE19542499A 1995-11-15 1995-11-15 Verfahren und Vorrichtung zur Herstellung einer parenteralen Arzneistoffzubereitung Withdrawn DE19542499A1 (de)

Priority Applications (12)

Application Number Priority Date Filing Date Title
DE19542499A DE19542499A1 (de) 1995-11-15 1995-11-15 Verfahren und Vorrichtung zur Herstellung einer parenteralen Arzneistoffzubereitung
DK96938066T DK0861068T3 (da) 1995-11-15 1996-11-04 Fremgangsmåde og apparat til fremstilling af et lægemiddel til parenteral indgivelse
ES96938066T ES2180807T3 (es) 1995-11-15 1996-11-04 Procedimiento y dispositivo para la obtencion de una preparacion medicamentosa parenteral.
CA002237554A CA2237554C (en) 1995-11-15 1996-11-04 A method and apparatus for producing liposomal parenteral medicaments via high pressure homogenization
PT96938066T PT861068E (pt) 1995-11-15 1996-11-04 Processo e dispositivo para a producao de um preparado medicinal de administracao por via parenterica
JP51854497A JP4049391B2 (ja) 1995-11-15 1996-11-04 非経口的薬剤の製造のための方法及び装置
EP96938066A EP0861068B1 (de) 1995-11-15 1996-11-04 Verfahren und vorrichtung zur herstellung einer parenteralen arzneistoff-zubereitung
US09/068,812 US6331314B1 (en) 1995-11-15 1996-11-04 Method and device for producing a parenteral medicament
AT96938066T ATE222097T1 (de) 1995-11-15 1996-11-04 Verfahren und vorrichtung zur herstellung einer parenteralen arzneistoff-zubereitung
DE59609564T DE59609564D1 (de) 1995-11-15 1996-11-04 Verfahren und vorrichtung zur herstellung einer parenteralen arzneistoff-zubereitung
PCT/EP1996/004795 WO1997017946A2 (de) 1995-11-15 1996-11-04 Verfahren und vorrichtung zur herstellung einer parenteralen arzneistoff-zubereitung
MX9803633A MX9803633A (es) 1995-11-15 1998-05-07 Procedimiento y dispositivo para la produccion de un preparado farmaceutico parenteral.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19542499A DE19542499A1 (de) 1995-11-15 1995-11-15 Verfahren und Vorrichtung zur Herstellung einer parenteralen Arzneistoffzubereitung

Publications (1)

Publication Number Publication Date
DE19542499A1 true DE19542499A1 (de) 1997-05-22

Family

ID=7777475

Family Applications (2)

Application Number Title Priority Date Filing Date
DE19542499A Withdrawn DE19542499A1 (de) 1995-11-15 1995-11-15 Verfahren und Vorrichtung zur Herstellung einer parenteralen Arzneistoffzubereitung
DE59609564T Expired - Lifetime DE59609564D1 (de) 1995-11-15 1996-11-04 Verfahren und vorrichtung zur herstellung einer parenteralen arzneistoff-zubereitung

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE59609564T Expired - Lifetime DE59609564D1 (de) 1995-11-15 1996-11-04 Verfahren und vorrichtung zur herstellung einer parenteralen arzneistoff-zubereitung

Country Status (11)

Country Link
US (1) US6331314B1 (enExample)
EP (1) EP0861068B1 (enExample)
JP (1) JP4049391B2 (enExample)
AT (1) ATE222097T1 (enExample)
CA (1) CA2237554C (enExample)
DE (2) DE19542499A1 (enExample)
DK (1) DK0861068T3 (enExample)
ES (1) ES2180807T3 (enExample)
MX (1) MX9803633A (enExample)
PT (1) PT861068E (enExample)
WO (1) WO1997017946A2 (enExample)

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1008380A3 (en) * 1998-12-07 2000-12-13 F. Hoffmann-La Roche Ag Process and apparatus for mixing or dispersing liquids
EP1222957A1 (en) * 2000-12-22 2002-07-17 Société des Produits Nestlé S.A. Process and device for producing a food grade oil-in-water emulsion
US8678184B2 (en) 2009-12-03 2014-03-25 Novartis Ag Methods for producing vaccine adjuvants
US8778275B2 (en) 2009-12-03 2014-07-15 Novartis Ag Methods for producing vaccine adjuvants
US8871816B2 (en) 2009-12-03 2014-10-28 Novartis Ag Methods for producing vaccine adjuvants
US8895629B2 (en) 2009-12-03 2014-11-25 Novartis Ag Circulation of components during homogenization of emulsions
USRE46906E1 (en) 2009-12-03 2018-06-26 Novartis Ag Methods for producing vaccine adjuvants
US10213383B2 (en) 2009-12-03 2019-02-26 Novartis Ag Hydrophilic filtration during manufacture of vaccine adjuvants

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20020119188A1 (en) * 2000-02-08 2002-08-29 Susan Niemiec Method of manufacturing liposomes
DE102004055507A1 (de) * 2004-11-17 2006-05-18 Basf Ag Verfahren zur Herstellung feinteiliger flüssig-flüssig Formulierungen und Vorrichtung zur Herstellung feinteiliger flüssig-flüssig Formulierungen
WO2007111937A1 (en) * 2006-03-23 2007-10-04 Applera Corporation Directed enrichment of genomic dna for high-throughput sequencing
US7985058B2 (en) * 2007-01-12 2011-07-26 Mark Gray Method and apparatus for making uniformly sized particles
US7491856B2 (en) * 2007-06-27 2009-02-17 H R D Corporation Method of making alkylene glycols
US7479576B1 (en) * 2007-06-27 2009-01-20 H R D Corporation Method of hydrogenating aldehydes and ketones
US8304584B2 (en) * 2007-06-27 2012-11-06 H R D Corporation Method of making alkylene glycols
US7652175B2 (en) * 2007-06-27 2010-01-26 H R D Corporation High shear process for the production of acetaldehyde
PL2158028T3 (pl) * 2007-06-28 2013-04-30 Procter & Gamble Urządzenie i sposób mieszania poprzez wytworzenie ścinania i kawitacji w płynie
US8322910B2 (en) 2008-07-25 2012-12-04 The Procter & Gamble Company Apparatus and method for mixing by producing shear and/or cavitation, and components for apparatus
CN101617990B (zh) * 2009-07-31 2013-01-23 中国人民解放军第三军医大学 脂质体制备装置以及使用该装置制备脂质体的方法
JP5771366B2 (ja) * 2009-09-02 2015-08-26 株式会社バイオメッドコア リポソーム製造装置及び方法
EP4651984A1 (en) * 2023-01-17 2025-11-26 DSM IP Assets B.V. Liquid dispersion preparation processes

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4529561A (en) * 1978-03-24 1985-07-16 The Regents Of The University Of California Method for producing liposomes in selected size range
EP0185756B1 (en) * 1984-06-20 1990-08-29 The Liposome Company, Inc. Extrusion techniques for producing liposomes
DE4207481A1 (de) * 1992-03-10 1993-09-16 Bayer Ag Liposomale wirkstoff-formulierungen und verfahren zu ihrer herstellung
DE4328331A1 (de) * 1993-08-18 1995-02-23 Andreas Dr Sachse Kontinuierliches Hochdruckextrusionsverfahren zur Herstellung von Liposomen und Emulsionen

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0082877A1 (en) * 1981-07-06 1983-07-06 Rush-Presbyterian-St.Luke's Medical Center Preparation of synthetic erythrocytes
DE3515335C2 (de) 1985-04-27 1995-01-26 Bayer Ag Arzneizubereitung enthaltend Dihydropyridine und Verfahren zu ihrer Herstellung
CA2146963A1 (en) * 1992-10-16 1994-04-28 Andreas Sachse Process and device for producing liquid, dispersed systems

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4529561A (en) * 1978-03-24 1985-07-16 The Regents Of The University Of California Method for producing liposomes in selected size range
EP0185756B1 (en) * 1984-06-20 1990-08-29 The Liposome Company, Inc. Extrusion techniques for producing liposomes
DE4207481A1 (de) * 1992-03-10 1993-09-16 Bayer Ag Liposomale wirkstoff-formulierungen und verfahren zu ihrer herstellung
DE4328331A1 (de) * 1993-08-18 1995-02-23 Andreas Dr Sachse Kontinuierliches Hochdruckextrusionsverfahren zur Herstellung von Liposomen und Emulsionen

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
GREGORIADIS,Gregory: Liposome Technology 2nd Edition, Vol.I, Liposome Preparation and Related Techniques, CRC Press, Boca Raton, Ann Arbor, London, Tokyo, 1993, S.49-63 *

Cited By (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1008380A3 (en) * 1998-12-07 2000-12-13 F. Hoffmann-La Roche Ag Process and apparatus for mixing or dispersing liquids
US6530684B1 (en) 1998-12-07 2003-03-11 Roche Vitamins Inc. Preparation of liquid dispersions
US6536940B1 (en) 1998-12-07 2003-03-25 Roche Vitamins Inc. Preparation of liquid dispersions
US6722780B2 (en) 1998-12-07 2004-04-20 Roche Vitamins Inc. Preparation of liquid dispersions
EP1222957A1 (en) * 2000-12-22 2002-07-17 Société des Produits Nestlé S.A. Process and device for producing a food grade oil-in-water emulsion
US8895629B2 (en) 2009-12-03 2014-11-25 Novartis Ag Circulation of components during homogenization of emulsions
US9750690B2 (en) 2009-12-03 2017-09-05 Novartis Ag Circulation of components during microfluidization and/or homogenization of emulsions
US8871816B2 (en) 2009-12-03 2014-10-28 Novartis Ag Methods for producing vaccine adjuvants
US8678184B2 (en) 2009-12-03 2014-03-25 Novartis Ag Methods for producing vaccine adjuvants
US9463240B2 (en) 2009-12-03 2016-10-11 Novartis Ag Arranging interaction and back pressure chambers for microfluidization
USRE46441E1 (en) 2009-12-03 2017-06-20 Novartis Ag Circulation of components during homogenization of emulsions
US9700616B2 (en) 2009-12-03 2017-07-11 Novartis Ag Arranging interaction and back pressure chambers for microfluidization
US8778275B2 (en) 2009-12-03 2014-07-15 Novartis Ag Methods for producing vaccine adjuvants
USRE46906E1 (en) 2009-12-03 2018-06-26 Novartis Ag Methods for producing vaccine adjuvants
US10213383B2 (en) 2009-12-03 2019-02-26 Novartis Ag Hydrophilic filtration during manufacture of vaccine adjuvants
US10463615B2 (en) 2009-12-03 2019-11-05 Novartis Ag Circulation of components during microfluidization and/or homogenization of emulsions
US10799454B2 (en) 2009-12-03 2020-10-13 Novartis Ag Hydrophilic filtration during manufacture of vaccine adjuvants
DE102009056884B4 (de) * 2009-12-03 2021-03-18 Novartis Ag Impfstoff-Adjuvantien und verbesserte Verfahren zur Herstellung derselben
US11141376B2 (en) 2009-12-03 2021-10-12 Novartis Ag Circulation of components during microfluidization and/or homogenization of emulsions

Also Published As

Publication number Publication date
DK0861068T3 (da) 2002-12-02
EP0861068B1 (de) 2002-08-14
CA2237554C (en) 2007-01-09
PT861068E (pt) 2002-12-31
CA2237554A1 (en) 1997-05-22
MX9803633A (es) 1998-09-30
WO1997017946A3 (de) 1997-09-12
DE59609564D1 (de) 2002-09-19
JP2000500146A (ja) 2000-01-11
ATE222097T1 (de) 2002-08-15
WO1997017946A2 (de) 1997-05-22
US6331314B1 (en) 2001-12-18
ES2180807T3 (es) 2003-02-16
EP0861068A2 (de) 1998-09-02
JP4049391B2 (ja) 2008-02-20

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OM8 Search report available as to paragraph 43 lit. 1 sentence 1 patent law
OP8 Request for examination as to paragraph 44 patent law
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