DE1695226A1 - Verfahren zur Herstellung von Benzodiazepin-Derivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepin-Derivaten

Info

Publication number
DE1695226A1
DE1695226A1 DE19681695226 DE1695226A DE1695226A1 DE 1695226 A1 DE1695226 A1 DE 1695226A1 DE 19681695226 DE19681695226 DE 19681695226 DE 1695226 A DE1695226 A DE 1695226A DE 1695226 A1 DE1695226 A1 DE 1695226A1
Authority
DE
Germany
Prior art keywords
compound
formula
halogen
general formula
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19681695226
Other languages
German (de)
English (en)
Inventor
Archer Giles Allan
Sternbach Leo Henryk
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of DE1695226A1 publication Critical patent/DE1695226A1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DE19681695226 1967-03-17 1968-03-02 Verfahren zur Herstellung von Benzodiazepin-Derivaten Pending DE1695226A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US62383467A 1967-03-17 1967-03-17

Publications (1)

Publication Number Publication Date
DE1695226A1 true DE1695226A1 (de) 1971-03-18

Family

ID=24499574

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19681695226 Pending DE1695226A1 (de) 1967-03-17 1968-03-02 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Country Status (16)

Country Link
US (1) US3553199A (enExample)
AT (1) AT278820B (enExample)
BE (1) BE712207A (enExample)
CH (1) CH493539A (enExample)
DE (1) DE1695226A1 (enExample)
DK (1) DK121125B (enExample)
ES (1) ES351720A1 (enExample)
FI (1) FI48088C (enExample)
FR (1) FR1556196A (enExample)
GB (1) GB1148288A (enExample)
IL (1) IL29640A (enExample)
MY (1) MY6900399A (enExample)
NL (1) NL6803724A (enExample)
NO (1) NO123037B (enExample)
SE (1) SE335736B (enExample)
YU (1) YU34201B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3817984A (en) * 1969-07-08 1974-06-18 Sumitomo Chemical Co Process for producing benzodiazepine derivatives
FR2054476A1 (en) * 1969-07-09 1971-04-23 Sumitomo Chemical Co Dihydro benzodiazpine derivs with tranqui- - lising, muscle-relaxant, antispasmodic and
BE785937A (fr) * 1971-07-08 1973-01-08 Sandoz Sa Nouveaux derives de la quinazoline, leur preparation et leur application comme medicaments
JPS6019753A (ja) * 1983-07-13 1985-01-31 Shionogi & Co Ltd オルト−（モノ置換アミノ）フエニルイミン類およびその製造法

Also Published As

Publication number Publication date
US3553199A (en) 1971-01-05
GB1148288A (en) 1969-04-10
CH493539A (de) 1970-07-15
DK121125B (da) 1971-09-13
SE335736B (enExample) 1971-06-07
AT278820B (de) 1970-02-10
IL29640A (en) 1972-06-28
NO123037B (enExample) 1971-09-20
FI48088B (enExample) 1974-02-28
BE712207A (enExample) 1968-09-16
ES351720A1 (es) 1969-06-16
YU58368A (en) 1978-06-30
MY6900399A (en) 1969-12-31
YU34201B (en) 1979-02-28
FI48088C (fi) 1974-06-10
FR1556196A (enExample) 1969-01-31
NL6803724A (enExample) 1968-09-18

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