DE102005023834A1 - Substituierte[(Phenylethanoyl)amino]benzamide - Google Patents

Substituierte[(Phenylethanoyl)amino]benzamide Download PDF

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Publication number
DE102005023834A1
DE102005023834A1 DE102005023834A DE102005023834A DE102005023834A1 DE 102005023834 A1 DE102005023834 A1 DE 102005023834A1 DE 102005023834 A DE102005023834 A DE 102005023834A DE 102005023834 A DE102005023834 A DE 102005023834A DE 102005023834 A1 DE102005023834 A1 DE 102005023834A1
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Germany
Prior art keywords
benzothien
alkyl
substituents
naphth
amino
Prior art date
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DE102005023834A
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German (de)
English (en)
Inventor
Ulf Dr. Brüggemeier
Petros Dr. Gatsios
Mark Dr. Meininghaus
Leila Dr. Telan
Elisabeth Dr. Woltering
Martina Dr. Wuttke
Hartmut Dr. Beck
Nils Dr. Griebenow
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Bayer AG
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Bayer Healthcare AG
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Publication date
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Priority to DE102005023834A priority Critical patent/DE102005023834A1/de
Priority to EP05813330A priority patent/EP1814872A1/de
Priority to CA002587511A priority patent/CA2587511A1/en
Priority to JP2007541790A priority patent/JP2008520605A/ja
Priority to PCT/EP2005/012322 priority patent/WO2006053748A1/de
Priority to US11/791,144 priority patent/US7776922B2/en
Publication of DE102005023834A1 publication Critical patent/DE102005023834A1/de
Withdrawn legal-status Critical Current

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/81—Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
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    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
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  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Virology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Communicable Diseases (AREA)
  • Diabetes (AREA)
  • Oncology (AREA)
  • Biomedical Technology (AREA)
  • Molecular Biology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Biotechnology (AREA)
  • Hematology (AREA)
  • Otolaryngology (AREA)
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  • Obesity (AREA)
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  • Vascular Medicine (AREA)
DE102005023834A 2004-11-20 2005-05-24 Substituierte[(Phenylethanoyl)amino]benzamide Withdrawn DE102005023834A1 (de)

Priority Applications (6)

Application Number Priority Date Filing Date Title
DE102005023834A DE102005023834A1 (de) 2004-11-20 2005-05-24 Substituierte[(Phenylethanoyl)amino]benzamide
EP05813330A EP1814872A1 (de) 2004-11-20 2005-11-17 Substituierte [(phenylethanoyl)amino] benzamide und deren verwendung zur behandlung von inflammatorischen sowie herz-kreislauf-erkrankungen
CA002587511A CA2587511A1 (en) 2004-11-20 2005-11-17 Substituted [(phenylethanoyl)amino] benzamides and the use thereof in the treatment of inflammatory and cardio-vascular diseases
JP2007541790A JP2008520605A (ja) 2004-11-20 2005-11-17 置換［（フェニルエタノイル）アミノ］ベンズアミドおよび炎症性および心臓血管疾患の処置におけるその使用
PCT/EP2005/012322 WO2006053748A1 (de) 2004-11-20 2005-11-17 Substituierte [(phenylethanoyl)amino] benzamide und deren verwendung zur behandlung von inflammatorischen sowie herz-kreislauf-erkrankungen
US11/791,144 US7776922B2 (en) 2004-11-20 2005-11-17 Substituted [(phenylethanoyl)amino]benzamides

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102004056078 2004-11-20
DE102004056078.1 2004-11-20
DE102005023834A DE102005023834A1 (de) 2004-11-20 2005-05-24 Substituierte[(Phenylethanoyl)amino]benzamide

Publications (1)

Publication Number Publication Date
DE102005023834A1 true DE102005023834A1 (de) 2006-05-24

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DE102005023834A Withdrawn DE102005023834A1 (de) 2004-11-20 2005-05-24 Substituierte[(Phenylethanoyl)amino]benzamide

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US (1) US7776922B2 (https=)
EP (1) EP1814872A1 (https=)
JP (1) JP2008520605A (https=)
CA (1) CA2587511A1 (https=)
DE (1) DE102005023834A1 (https=)
WO (1) WO2006053748A1 (https=)

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EP2061479A4 (en) * 2006-09-05 2010-08-04 Bipar Sciences Inc FETTIC ACID SYNTHESIS INHIBITED BY PARP HEMMER AND TREATMENT PROCEDURES THEREWITH
EP2203432A4 (en) * 2007-09-21 2011-04-27 Glaxosmithkline Llc PROCESSING METHOD
US8143447B2 (en) 2006-09-05 2012-03-27 Bipar Sciences, Inc. Treatment of cancer
US8377985B2 (en) 2005-07-18 2013-02-19 Bipar Sciences, Inc. Treatment of cancer

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AU2003284237A1 (en) * 2002-10-16 2004-05-04 Transport Systems, Inc. Monorail sortation system
US20100256157A1 (en) * 2002-10-29 2010-10-07 Jakob Busch-Petersen Method of treatment
JO3598B1 (ar) 2006-10-10 2020-07-05 Infinity Discovery Inc الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني
CA2713156A1 (en) * 2008-02-04 2009-08-13 Bipar Sciences, Inc. Methods of diagnosing and treating parp-mediated diseases
TW201000107A (en) * 2008-04-09 2010-01-01 Infinity Pharmaceuticals Inc Inhibitors of fatty acid amide hydrolase
CA2757622A1 (en) 2009-04-07 2010-10-14 Infinity Pharmaceuticals, Inc. Inhibitors of fatty acid amide hydrolase
WO2010118155A1 (en) 2009-04-07 2010-10-14 Infinity Pharmaceuticals, Inc. Inhibitors of fatty acid amide hydrolase
MX361692B (es) 2010-02-03 2018-12-13 Infinity Pharmaceuticals Inc Inhibidores de amida hidrolasa de ácido graso.
DK3362462T3 (da) 2015-10-12 2021-10-11 Advanced Cell Diagnostics Inc In situ-detektion af nukleotidvarianter i prøver med højt støjniveau, og sammensætninger og fremgangsmåder relateret dertil
CN110776486B (zh) * 2019-10-23 2022-05-20 中国药科大学 一种苯并呋喃类小分子p2y14受体抑制剂，及其制备和应用

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GB9816837D0 (en) 1998-08-04 1998-09-30 Zeneca Ltd Amide derivatives
AU761291B2 (en) * 1999-03-17 2003-05-29 Astrazeneca Ab Amide derivatives

Cited By (7)

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