JP2008520605A - 置換［（フェニルエタノイル）アミノ］ベンズアミドおよび炎症性および心臓血管疾患の処置におけるその使用 - Google Patents

置換［（フェニルエタノイル）アミノ］ベンズアミドおよび炎症性および心臓血管疾患の処置におけるその使用 Download PDF

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JP2008520605A
JP2008520605A JP2007541790A JP2007541790A JP2008520605A JP 2008520605 A JP2008520605 A JP 2008520605A JP 2007541790 A JP2007541790 A JP 2007541790A JP 2007541790 A JP2007541790 A JP 2007541790A JP 2008520605 A JP2008520605 A JP 2008520605A
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benzothien
alkyl
amino
naphth
substituents
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JP2008520605A5 (https=
Inventor
ウルフ・ブリュックマイヤー
ペトロス・ガツィオス
マルク・マイニングハウス
ライラ・テラン
エリーザベト・ヴォルテリング
マルティナ・ヴットケ
ハルトムート・ベック
ニールス・グリーベノウ
フランク・ジュースマイヤー
ニールス・スフェンストルップ
アクセル・クレッチュマー
マルクス・バウザー
ヨハネス・ケーベルリング
ヴァヘト・モラディ
ジークフリート・ツァイス
クラウディア・ヒルト−ディートリッヒ
バルバラ・アルブレヒト
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Bayer AG
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Bayer Healthcare AG
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    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/81—Radicals substituted by nitrogen atoms not forming part of a nitro radical
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    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
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    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
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  • Health & Medical Sciences (AREA)
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  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Communicable Diseases (AREA)
  • Diabetes (AREA)
  • Oncology (AREA)
  • Biomedical Technology (AREA)
  • Molecular Biology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Biotechnology (AREA)
  • Hematology (AREA)
  • Otolaryngology (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
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JP2007541790A 2004-11-20 2005-11-17 置換［（フェニルエタノイル）アミノ］ベンズアミドおよび炎症性および心臓血管疾患の処置におけるその使用 Withdrawn JP2008520605A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102004056078 2004-11-20
DE102005023834A DE102005023834A1 (de) 2004-11-20 2005-05-24 Substituierte[(Phenylethanoyl)amino]benzamide
PCT/EP2005/012322 WO2006053748A1 (de) 2004-11-20 2005-11-17 Substituierte [(phenylethanoyl)amino] benzamide und deren verwendung zur behandlung von inflammatorischen sowie herz-kreislauf-erkrankungen

Publications (2)

Publication Number Publication Date
JP2008520605A true JP2008520605A (ja) 2008-06-19
JP2008520605A5 JP2008520605A5 (https=) 2009-01-08

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JP2007541790A Withdrawn JP2008520605A (ja) 2004-11-20 2005-11-17 置換［（フェニルエタノイル）アミノ］ベンズアミドおよび炎症性および心臓血管疾患の処置におけるその使用

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US (1) US7776922B2 (https=)
EP (1) EP1814872A1 (https=)
JP (1) JP2008520605A (https=)
CA (1) CA2587511A1 (https=)
DE (1) DE102005023834A1 (https=)
WO (1) WO2006053748A1 (https=)

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AU2003284237A1 (en) * 2002-10-16 2004-05-04 Transport Systems, Inc. Monorail sortation system
US20100256157A1 (en) * 2002-10-29 2010-10-07 Jakob Busch-Petersen Method of treatment
CA2615374A1 (en) 2005-07-18 2007-01-25 Ernest Kun Kun Treatment of cancer
CA2662337A1 (en) * 2006-09-05 2008-03-13 Bipar Sciences, Inc. Inhibition of fatty acid synthesis by parp inhibitors and methods of treatment thereof
JP2010502730A (ja) 2006-09-05 2010-01-28 バイパー サイエンシズ，インコーポレイティド 癌の治療法
JO3598B1 (ar) 2006-10-10 2020-07-05 Infinity Discovery Inc الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني
EP2203432A4 (en) * 2007-09-21 2011-04-27 Glaxosmithkline Llc PROCESSING METHOD
CA2713156A1 (en) * 2008-02-04 2009-08-13 Bipar Sciences, Inc. Methods of diagnosing and treating parp-mediated diseases
TW201000107A (en) * 2008-04-09 2010-01-01 Infinity Pharmaceuticals Inc Inhibitors of fatty acid amide hydrolase
CA2757622A1 (en) 2009-04-07 2010-10-14 Infinity Pharmaceuticals, Inc. Inhibitors of fatty acid amide hydrolase
WO2010118155A1 (en) 2009-04-07 2010-10-14 Infinity Pharmaceuticals, Inc. Inhibitors of fatty acid amide hydrolase
MX361692B (es) 2010-02-03 2018-12-13 Infinity Pharmaceuticals Inc Inhibidores de amida hidrolasa de ácido graso.
DK3362462T3 (da) 2015-10-12 2021-10-11 Advanced Cell Diagnostics Inc In situ-detektion af nukleotidvarianter i prøver med højt støjniveau, og sammensætninger og fremgangsmåder relateret dertil
CN110776486B (zh) * 2019-10-23 2022-05-20 中国药科大学 一种苯并呋喃类小分子p2y14受体抑制剂，及其制备和应用

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GB9816837D0 (en) 1998-08-04 1998-09-30 Zeneca Ltd Amide derivatives
AU761291B2 (en) * 1999-03-17 2003-05-29 Astrazeneca Ab Amide derivatives

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DE102005023834A1 (de) 2006-05-24
WO2006053748A1 (de) 2006-05-26
EP1814872A1 (de) 2007-08-08
US7776922B2 (en) 2010-08-17
CA2587511A1 (en) 2006-05-26
US20080171786A1 (en) 2008-07-17

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