DD242407A5 - Verfahren zur herstellung von imidazoderivaten - Google Patents

Verfahren zur herstellung von imidazoderivaten Download PDF

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Publication number
DD242407A5
DD242407A5 DD85284542A DD28454285A DD242407A5 DD 242407 A5 DD242407 A5 DD 242407A5 DD 85284542 A DD85284542 A DD 85284542A DD 28454285 A DD28454285 A DD 28454285A DD 242407 A5 DD242407 A5 DD 242407A5
Authority
DD
German Democratic Republic
Prior art keywords
radicals
group
imidazo
general formula
methoxy
Prior art date
Application number
DD85284542A
Other languages
German (de)
English (en)
Inventor
Joachim Heider
Norbert Hauel
Volkhard Austel
Klaus Noll
Andreas Bomhard
Jacques Van Meel
Willi Diederen
Original Assignee
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Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ���@����������@��k�� filed Critical ���@����������@��k��
Publication of DD242407A5 publication Critical patent/DD242407A5/de

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DD85284542A 1984-12-21 1985-12-17 Verfahren zur herstellung von imidazoderivaten DD242407A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19843446778 DE3446778A1 (de) 1984-12-21 1984-12-21 Neue imidazoderivate, ihre herstellung und diese verbindungen enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
DD242407A5 true DD242407A5 (de) 1987-01-28

Family

ID=6253488

Family Applications (1)

Application Number Title Priority Date Filing Date
DD85284542A DD242407A5 (de) 1984-12-21 1985-12-17 Verfahren zur herstellung von imidazoderivaten

Country Status (14)

Country Link
US (1) US4716169A (el)
EP (1) EP0185345A1 (el)
JP (1) JPS61152681A (el)
AU (1) AU5154585A (el)
DD (1) DD242407A5 (el)
DE (1) DE3446778A1 (el)
DK (1) DK590185A (el)
ES (2) ES8703472A1 (el)
FI (1) FI855080A (el)
GR (1) GR853124B (el)
HU (1) HU194562B (el)
NO (1) NO855196L (el)
PT (1) PT81716B (el)
ZA (1) ZA859729B (el)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4833149A (en) * 1986-09-22 1989-05-23 Ortho Pharmaceutical Corporation 2- or 3-aryl substituted imidazo[1,2-a]pyridines
GB8719368D0 (en) * 1987-08-15 1987-09-23 Wellcome Found Heterocyclic compounds
SE8704248D0 (sv) * 1987-10-30 1987-10-30 Haessle Ab Medical use
CA2048110C (en) * 1990-07-30 2002-06-25 Muneo Takatani Imidazopyridine derivatives and their use
US6127576A (en) * 1996-12-20 2000-10-03 American Cyanamid Company Aminophenyl ketone derivatives and a method for the preparation thereof
JP4327915B2 (ja) * 1998-03-30 2009-09-09 株式会社デ・ウエスタン・セラピテクス研究所 スルフォンアミド誘導体
US6596731B2 (en) 2001-03-27 2003-07-22 Hoffmann-La Roche Inc. Substituted imidazo[1,2-A] pyridine derivatives
US20080219922A1 (en) * 2005-09-12 2008-09-11 Goodman Mark M Alzheimer's Disease Imaging Agents
US7723336B2 (en) * 2005-09-22 2010-05-25 Bristol-Myers Squibb Company Fused heterocyclic compounds useful as kinase modulators
US8703096B2 (en) * 2006-04-21 2014-04-22 The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services Beta-amyloid PET imaging agents
EP1964841A1 (en) * 2007-02-28 2008-09-03 sanofi-aventis Imidazo[1,2-a]azine and their use as pharmaceuticals
EP1964840A1 (en) * 2007-02-28 2008-09-03 sanofi-aventis Imidazo[1,2-a]pyridines and their use as pharmaceuticals
US7868001B2 (en) 2007-11-02 2011-01-11 Hutchison Medipharma Enterprises Limited Cytokine inhibitors
JP5394404B2 (ja) * 2008-02-06 2014-01-22 ブリストル−マイヤーズ スクイブ カンパニー キナーゼ阻害剤として有用な置換イミダゾピリダジン類
PT2280706E (pt) * 2008-05-14 2013-02-19 Otsuka Pharma Co Ltd Composições compreendendo derivados de benzeno que activam lipase de lipoproteína
AU2013251680A1 (en) 2012-04-26 2014-11-13 Bristol-Myers Squibb Company Imidazothiadiazole and imidazopyridazine derivatives as protease activated receptor 4 (par4) inhibitors for treating platelet aggregation
ES2625029T3 (es) 2012-04-26 2017-07-18 Bristol-Myers Squibb Company Derivados del imidazotiadiazol como inhibidores del receptor 4 activado por proteasa (Par4) para el tratamiento de la agregación de plaquetas
RS59882B1 (sr) * 2012-04-26 2020-03-31 Bristol Myers Squibb Co Derivati imidazotiadiazola i imidazopirazina kao inhibitori proteazom aktiviranog receptora 4 (par4) za lečenje agregacije trombocita
US9617279B1 (en) 2014-06-24 2017-04-11 Bristol-Myers Squibb Company Imidazooxadiazole compounds
US9598419B1 (en) 2014-06-24 2017-03-21 Universite De Montreal Imidazotriazine and imidazodiazine compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS523957B2 (el) * 1974-03-14 1977-01-31
US4166851A (en) * 1977-05-16 1979-09-04 Merck & Co., Inc. Certain imidazo(1,2a)pyridine derivatives
ZA839398B (en) * 1982-12-27 1985-08-28 Lilly Co Eli Substituted imidazopyrimidines-pyrazines,and-triazines

Also Published As

Publication number Publication date
DK590185D0 (da) 1985-12-18
US4716169A (en) 1987-12-29
ES8801276A1 (es) 1988-01-01
DK590185A (da) 1986-06-22
HUT40434A (en) 1986-12-28
ES556974A0 (es) 1988-01-01
ZA859729B (en) 1987-08-26
ES550241A0 (es) 1987-02-16
PT81716B (de) 1987-10-15
ES8703472A1 (es) 1987-02-16
JPS61152681A (ja) 1986-07-11
FI855080A (fi) 1986-06-22
EP0185345A1 (de) 1986-06-25
GR853124B (el) 1986-04-22
NO855196L (no) 1986-06-23
AU5154585A (en) 1986-06-26
PT81716A (de) 1986-01-01
HU194562B (en) 1988-02-29
DE3446778A1 (de) 1986-07-03
FI855080A0 (fi) 1985-12-19

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