DD157614A5 - Verfahren zur herstellung von pyrimidyl-chinazolinen - Google Patents

Verfahren zur herstellung von pyrimidyl-chinazolinen Download PDF

Info

Publication number
DD157614A5
DD157614A5 DD81228589A DD22858981A DD157614A5 DD 157614 A5 DD157614 A5 DD 157614A5 DD 81228589 A DD81228589 A DD 81228589A DD 22858981 A DD22858981 A DD 22858981A DD 157614 A5 DD157614 A5 DD 157614A5
Authority
DD
German Democratic Republic
Prior art keywords
formula
compound
atoms
amino
alkyl
Prior art date
Application number
DD81228589A
Other languages
German (de)
English (en)
Inventor
Heinz Bender
Thomas Raabe
Helmut Bohn
Piero Martorana
Original Assignee
Cassella Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cassella Ag filed Critical Cassella Ag
Publication of DD157614A5 publication Critical patent/DD157614A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Hospice & Palliative Care (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
  • Catching Or Destruction (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
DD81228589A 1980-03-27 1981-03-25 Verfahren zur herstellung von pyrimidyl-chinazolinen DD157614A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19803011809 DE3011809A1 (de) 1980-03-27 1980-03-27 Pyrimidyl-chinazoline, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische praeparate und ihre verwendung

Publications (1)

Publication Number Publication Date
DD157614A5 true DD157614A5 (de) 1982-11-24

Family

ID=6098481

Family Applications (1)

Application Number Title Priority Date Filing Date
DD81228589A DD157614A5 (de) 1980-03-27 1981-03-25 Verfahren zur herstellung von pyrimidyl-chinazolinen

Country Status (18)

Country Link
EP (1) EP0037495A1 (enrdf_load_stackoverflow)
JP (1) JPS56150088A (enrdf_load_stackoverflow)
AR (1) AR227542A1 (enrdf_load_stackoverflow)
AU (1) AU6877481A (enrdf_load_stackoverflow)
CA (1) CA1156656A (enrdf_load_stackoverflow)
CS (1) CS219898B2 (enrdf_load_stackoverflow)
DD (1) DD157614A5 (enrdf_load_stackoverflow)
DE (1) DE3011809A1 (enrdf_load_stackoverflow)
DK (1) DK115581A (enrdf_load_stackoverflow)
ES (1) ES500738A0 (enrdf_load_stackoverflow)
FI (1) FI810778L (enrdf_load_stackoverflow)
GR (1) GR71870B (enrdf_load_stackoverflow)
IL (1) IL62495A0 (enrdf_load_stackoverflow)
NO (1) NO810870L (enrdf_load_stackoverflow)
PL (2) PL230320A1 (enrdf_load_stackoverflow)
PT (1) PT72724B (enrdf_load_stackoverflow)
SU (1) SU1052158A3 (enrdf_load_stackoverflow)
ZA (1) ZA812034B (enrdf_load_stackoverflow)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61140568A (ja) * 1984-12-14 1986-06-27 Mitsui Petrochem Ind Ltd キナゾリン誘導体及びそれを有効成分とする血圧降下剤
JPS6267077A (ja) * 1985-09-18 1987-03-26 Mitsui Petrochem Ind Ltd キナゾリン誘導体及び医薬
CA2559302C (en) * 2004-03-15 2012-06-19 Takeda Pharmaceutical Company Limited 6-amino-1h-pyrimidine-2,4-dione derivatives as dipeptidyl peptidase inhibitors
WO2006014394A1 (en) 2004-07-02 2006-02-09 Corcept Therapeutics, Inc. Modified pyrimidine glucocorticoid receptor modulators
PE20141378A1 (es) 2011-03-18 2014-10-12 Corcept Therapeutics Inc Moduladores de receptores de glucocorticoides de pirimidina ciclohexilo
JP7196201B2 (ja) 2018-06-04 2022-12-26 コーセプト セラピューティクス， インコーポレイテッド ピリミジンシクロヘキセニル糖質コルチコイドレセプター調節因子
CA3158745A1 (en) 2019-12-11 2021-06-17 Corcept Therapeutics Incorporated Methods of treating antipsychotic-induced weight gain with miricorilant
CN115551836A (zh) 2020-05-06 2022-12-30 科赛普特治疗公司 嘧啶环己基糖皮质激素受体调节剂的多晶型物
IL297840A (en) 2020-05-06 2023-01-01 Corcept Therapeutics Inc Formulations of pyrimidine cyclohexyl glucocorticoid receptor modulators
CA3202353A1 (en) 2020-12-21 2022-06-30 Jeffrey Mark Dener Method of preparing pyrimidine cyclohexyl glucocorticoid receptor modulators

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2007656B (en) * 1977-11-05 1982-05-19 Pfizer Ltd Therapeutic agents

Also Published As

Publication number Publication date
FI810778A7 (fi) 1981-09-28
SU1052158A3 (ru) 1983-10-30
ZA812034B (en) 1982-05-26
ES8202000A1 (es) 1982-01-16
PL230320A1 (enrdf_load_stackoverflow) 1982-03-29
PT72724A (de) 1981-04-01
DE3011809A1 (de) 1981-10-01
NO810870L (no) 1981-09-28
GR71870B (enrdf_load_stackoverflow) 1983-07-08
PT72724B (de) 1982-03-24
PL233882A1 (enrdf_load_stackoverflow) 1982-05-10
JPS56150088A (en) 1981-11-20
AU6877481A (en) 1981-10-01
CS219898B2 (en) 1983-03-25
AR227542A1 (es) 1982-11-15
ES500738A0 (es) 1982-01-16
CA1156656A (en) 1983-11-08
EP0037495A1 (de) 1981-10-14
DK115581A (da) 1981-09-28
IL62495A0 (en) 1981-05-20
FI810778L (fi) 1981-09-28

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