DD146953A5 - Verfahren zur herstellung von pyrimidonderivaten - Google Patents

Verfahren zur herstellung von pyrimidonderivaten Download PDF

Info

Publication number
DD146953A5
DD146953A5 DD79216837A DD21683779A DD146953A5 DD 146953 A5 DD146953 A5 DD 146953A5 DD 79216837 A DD79216837 A DD 79216837A DD 21683779 A DD21683779 A DD 21683779A DD 146953 A5 DD146953 A5 DD 146953A5
Authority
DD
German Democratic Republic
Prior art keywords
group
radical
general formula
pyridyl
substituted
Prior art date
Application number
DD79216837A
Other languages
German (de)
English (en)
Inventor
Thomas H Brown
Robert J Ife
Original Assignee
Smith Kline French Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smith Kline French Lab filed Critical Smith Kline French Lab
Publication of DD146953A5 publication Critical patent/DD146953A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
DD79216837A 1978-11-13 1979-11-12 Verfahren zur herstellung von pyrimidonderivaten DD146953A5 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7844260 1978-11-13
GB7929013 1979-08-21

Publications (1)

Publication Number Publication Date
DD146953A5 true DD146953A5 (de) 1981-03-11

Family

ID=26269556

Family Applications (1)

Application Number Title Priority Date Filing Date
DD79216837A DD146953A5 (de) 1978-11-13 1979-11-12 Verfahren zur herstellung von pyrimidonderivaten

Country Status (22)

Country Link
US (1) US4496567A (cs)
EP (1) EP0013071B1 (cs)
JP (1) JPS55500898A (cs)
AU (1) AU534802B2 (cs)
CA (1) CA1137984A (cs)
CS (1) CS214813B2 (cs)
DD (1) DD146953A5 (cs)
DE (1) DE2966413D1 (cs)
DK (1) DK298180A (cs)
ES (1) ES485912A1 (cs)
FI (1) FI793533A7 (cs)
GR (1) GR78338B (cs)
HU (1) HU182740B (cs)
IE (1) IE49205B1 (cs)
IL (1) IL58676A (cs)
NO (1) NO793642L (cs)
NZ (1) NZ192096A (cs)
PH (1) PH15579A (cs)
PL (1) PL126169B1 (cs)
PT (1) PT70441A (cs)
RO (1) RO78491A (cs)
WO (1) WO1980000966A1 (cs)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1140129A (en) * 1979-08-21 1983-01-25 Ronald J. King 4-pyrimidone derivatives
DE3275291D1 (en) * 1981-07-24 1987-03-05 Glaxo Group Ltd Heterocyclic derivatives
US4745110A (en) * 1983-04-29 1988-05-17 Rorer Pharmaceutical Corporation Bicyclic benzenoid aminoalkylene ethers and thioethers, pharmaceutical compositions and use
GB8318638D0 (en) * 1983-07-09 1983-08-10 Smith Kline French Lab Chemical compounds
GB8320505D0 (en) * 1983-07-29 1983-09-01 Smith Kline French Lab Chemical compounds
US4772704A (en) * 1983-09-21 1988-09-20 Bristol-Myers Company 2,5-disubstituted-4(3H)-pyrimidones having histamine H2 -receptor antagonist activity
GB8332091D0 (en) * 1983-12-01 1984-01-11 Smith Kline French Lab Chemical compounds
GB8421427D0 (en) * 1984-08-23 1984-09-26 Smith Kline French Lab Chemical compounds
JO1410B1 (en) * 1984-11-03 1986-11-30 سميث كلاين اند فرينش لابوراتوريز ليمتد Compounds
JPS61155373A (ja) * 1984-12-28 1986-07-15 Yamanouchi Pharmaceut Co Ltd 新規な２−置換アミノ−４（１ｈ）−ピリミドン誘導体及びその製造法
JP2807577B2 (ja) * 1990-06-15 1998-10-08 エーザイ株式会社 環状アミド誘導体
EP3909449A1 (en) 2020-05-11 2021-11-17 Bisaf Spolka Z Ograniczona Odpowiedzialnoscia Protective filtering half mask

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1223686A (en) * 1967-02-24 1971-03-03 Ici Ltd Salts of pyrimidine derivatives and the use thereof as fungicides
US3980781A (en) * 1966-03-31 1976-09-14 Imperial Chemical Industries Limited Fungicidal composition and method containing 2-amino-pyrimidines
GB1419994A (en) * 1973-05-03 1976-01-07 Smith Kline French Lab Heterocyclicalkylaminotheterocyclic compounds methods for their preparation and compositions comprising them
IN146736B (cs) * 1975-10-02 1979-08-25 Smith Kline French Lab
US4145546A (en) * 1975-10-02 1979-03-20 Smith Kline & French Laboratories Limited 4-Pyrimidone compounds
US4154834A (en) * 1975-12-29 1979-05-15 Smith Kline & French Laboratories Limited Substituted isocytosines having histamine H2 -antagonist activity
MW5076A1 (en) * 1975-12-29 1978-02-08 Smith Kline French Lab Pharmacologicalle active compounds
US4117131A (en) * 1976-12-07 1978-09-26 Warner-Lambert Company Method of inhibiting gastric acid secretions with 2-(4-pyrimidinyl)thioacetamides
GB1604674A (en) * 1977-05-17 1981-12-16 Allen & Hanburys Ltd Aminoalkyl-benzene derivatives
ZA793443B (en) * 1978-07-26 1980-12-31 Glaxo Group Ltd Heterocyclic derivatives

Also Published As

Publication number Publication date
EP0013071A1 (en) 1980-07-09
PH15579A (en) 1983-02-17
PL126169B1 (en) 1983-07-30
IL58676A0 (en) 1980-02-29
US4496567A (en) 1985-01-29
PL219563A1 (cs) 1980-12-01
GR78338B (cs) 1984-09-26
HU182740B (en) 1984-03-28
WO1980000966A1 (en) 1980-05-15
PT70441A (en) 1979-12-01
EP0013071B1 (en) 1983-11-16
JPS55500898A (cs) 1980-11-06
CS214813B2 (en) 1982-06-25
AU534802B2 (en) 1984-02-16
DK298180A (da) 1980-07-10
IL58676A (en) 1983-07-31
IE49205B1 (en) 1985-08-21
RO78491A (ro) 1982-02-26
AU5272279A (en) 1980-05-22
FI793533A7 (fi) 1981-01-01
IE792169L (en) 1980-05-13
NO793642L (no) 1980-05-14
DE2966413D1 (en) 1983-12-22
CA1137984A (en) 1982-12-21
ES485912A1 (es) 1980-07-01
NZ192096A (en) 1981-11-19

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