GB1223686A - Salts of pyrimidine derivatives and the use thereof as fungicides - Google Patents

Salts of pyrimidine derivatives and the use thereof as fungicides

Info

Publication number
GB1223686A
GB1223686A GB3034867A GB3034867A GB1223686A GB 1223686 A GB1223686 A GB 1223686A GB 3034867 A GB3034867 A GB 3034867A GB 3034867 A GB3034867 A GB 3034867A GB 1223686 A GB1223686 A GB 1223686A
Authority
GB
United Kingdom
Prior art keywords
optionally substituted
sulphur
feb
hydrogen
substituted hydrocarbon
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB3034867A
Inventor
Brian Kenneth Snell
Richard Stewart Elias
Peter Frank Hilary Freeman
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Imperial Chemical Industries Ltd
Original Assignee
Imperial Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Imperial Chemical Industries Ltd filed Critical Imperial Chemical Industries Ltd
Priority to GB3034867A priority Critical patent/GB1223686A/en
Priority to IE19468A priority patent/IE31957B1/en
Priority to IL2949668A priority patent/IL29496A/en
Publication of GB1223686A publication Critical patent/GB1223686A/en
Priority to US05/207,530 priority patent/US3980781A/en
Priority to CY68273A priority patent/CY682A/en
Priority to MY7300294A priority patent/MY7300294A/en
Priority to US05/650,864 priority patent/US4000138A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/56—One oxygen atom and one sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/69—Benzenesulfonamido-pyrimidines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Abstract

1,223,686. Fungicidal seed dressings. IMPERIAL CHEMICAL INDUSTRIES Ltd. 12 Feb., 1968 [24 Feb., 1967; 30 June, 1967], Nos. 30348/67 and 30354/67. Heading A2Q. [Also in Divisions A5 and C2] A seed dressing having fungicidal properties comprises as active ingredient an acid addition salt or metal salt of a pyrimidine of the formula or an acid addition salt of an ether thereof, where X is oxygen or sulphur, R 1 and R 2 are hydrogen, optionally substituted hydrocarbon, heterocystic, benzylidine-imino, amino or sulphur-free substituted amino, cyano, optionally substituted carbamoyl or R.CO- or R.CO 2 groups (where R is optionally substituted hydrocarbon), or R 1 and R 2 together with the N atom complete an optionally substituted helerocyclic ring which may contain further hetero atoms, and R 3 and R 4 are hydrogen, halogen, an optionally substituted hydrocarbon group bound to the pyrimidine ring through -O- or -S-, heterocyclic-substituted alkyl, nitro, ajophenyl or alkylsulphonyl groups or R 3 and R 4 together form an optionally substituted alkylene or alkenylene bridging group, together with a solid diluent or liquid diluent containing a surface active agent. The dressing may be applied to.e.g., wheat barley or rice. Evample 42 describes a composition based on china clay containing the potassium salt of 2-dimethylamino- 4-methyl-5-n-butyl-6-hydroxypyrimidine.
GB3034867A 1966-03-31 1967-02-24 Salts of pyrimidine derivatives and the use thereof as fungicides Expired GB1223686A (en)

Priority Applications (7)

Application Number Priority Date Filing Date Title
GB3034867A GB1223686A (en) 1967-02-24 1967-02-24 Salts of pyrimidine derivatives and the use thereof as fungicides
IE19468A IE31957B1 (en) 1967-02-24 1968-02-15 Salts of pyrimidine derivatives and the use thereof as fungicides
IL2949668A IL29496A (en) 1967-02-24 1968-02-19 Fungicidal compositions containing salts of pyrimidine derivatives and certain novel salts of pyrimidine derivative
US05/207,530 US3980781A (en) 1966-03-31 1971-12-13 Fungicidal composition and method containing 2-amino-pyrimidines
CY68273A CY682A (en) 1967-02-24 1973-05-03 Salts of pyrimidine derivatives and the use thereof as fungicides
MY7300294A MY7300294A (en) 1967-02-24 1973-12-31 Salts of pyrimidine derivatives and the use thereof as fungicides
US05/650,864 US4000138A (en) 1966-03-31 1976-01-21 Organic compounds and compositions containing them

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB3034867A GB1223686A (en) 1967-02-24 1967-02-24 Salts of pyrimidine derivatives and the use thereof as fungicides
GB3035467 1967-06-30

Publications (1)

Publication Number Publication Date
GB1223686A true GB1223686A (en) 1971-03-03

Family

ID=26260398

Family Applications (1)

Application Number Title Priority Date Filing Date
GB3034867A Expired GB1223686A (en) 1966-03-31 1967-02-24 Salts of pyrimidine derivatives and the use thereof as fungicides

Country Status (4)

Country Link
CY (1) CY682A (en)
GB (1) GB1223686A (en)
IE (1) IE31957B1 (en)
IL (1) IL29496A (en)

Cited By (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3932617A (en) * 1974-05-24 1976-01-13 The Upjohn Company Interferon induction
WO1980000966A1 (en) * 1978-11-13 1980-05-15 Smith Kline French Lab New histamine h2-antagonists
EP0019450A1 (en) * 1979-05-15 1980-11-26 Takeda Chemical Industries, Ltd. Pyrimidine derivatives and their production and agricultural uses
US4238493A (en) 1978-05-30 1980-12-09 Smith Kline & French Laboratories Limited 2-(Substituted amino)-3-nitro-2,3-unsaturated nitrogen heterocycles
US4255428A (en) 1979-03-24 1981-03-10 Smith Kline & French Laboratories Limited 5-(Hydroxypyridylalkyl)-4-pyrimidones
US4305945A (en) 1978-07-15 1981-12-15 Smith Kline & French Laboratories Limited Isoureas and isothioureas
US4308272A (en) 1980-10-03 1981-12-29 The Upjohn Company Process for treating hypertension
EP0055692A1 (en) * 1980-12-15 1982-07-07 Sandoz Ag Novel pyrimidinyl ethers, their use as herbicides, herbicidal compositions comprising said pyrimidinyl ethers and processes for the preparation thereof
US4341787A (en) 1973-05-03 1982-07-27 Smith Kline & French Laboratories Limited Pharmacologically active compounds
US4399142A (en) 1973-05-03 1983-08-16 Smith Kline & French Laboratories Limited Pharmacologically active compounds
US4460589A (en) * 1980-10-03 1984-07-17 The Upjohn Company Process for treating hypertension
US4470985A (en) * 1973-05-03 1984-09-11 Smithkline & French Laboratories Limited Pharmacologically active compounds
US4507302A (en) * 1979-03-19 1985-03-26 The Upjohn Company Method for treating arthritis with 6-aryl pyrimidine compounds
US4521418A (en) * 1979-02-21 1985-06-04 Smith Kline & French Laboratories Limited Guanidinothiazolyl derivatives
US4525477A (en) * 1981-12-02 1985-06-25 Smith Kline & French Laboratories Limited 2-Thiazolyl, isothiazolyl, oxazolyl and isoxazolyl alkylamino-3-nitro-heterocyclic compounds
US4537779A (en) * 1973-05-03 1985-08-27 Smith Kline & French Laboratories Limited Pharmacologically active compounds
US4593096A (en) * 1982-06-09 1986-06-03 The Upjohn Company Novel compounds and process for treating hypertension
US4600720A (en) * 1973-05-03 1986-07-15 Smith Kline & French Laboratories Ltd. Pharmacologically active compounds
US4649141A (en) * 1978-02-13 1987-03-10 Smith Kline & French Laboratories Limited Pyrimidine compounds
US5002951A (en) * 1979-03-19 1991-03-26 The Upjohn Company Method for treating bacterial and protozoal infections
US5434157A (en) * 1979-03-19 1995-07-18 The Upjohn Company 6-aryl pyrimidine compounds and method for treating viral infections and inducing interferon production
US5554617A (en) * 1979-09-28 1996-09-10 The Upjohn Company Method for treating cancer with 6-aryl pyrimidine compounds
US6495558B1 (en) 1999-01-22 2002-12-17 Amgen Inc. Kinase inhibitors

Cited By (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4341787A (en) 1973-05-03 1982-07-27 Smith Kline & French Laboratories Limited Pharmacologically active compounds
US4600720A (en) * 1973-05-03 1986-07-15 Smith Kline & French Laboratories Ltd. Pharmacologically active compounds
US4537779A (en) * 1973-05-03 1985-08-27 Smith Kline & French Laboratories Limited Pharmacologically active compounds
US4470985A (en) * 1973-05-03 1984-09-11 Smithkline & French Laboratories Limited Pharmacologically active compounds
US4399142A (en) 1973-05-03 1983-08-16 Smith Kline & French Laboratories Limited Pharmacologically active compounds
US3932617A (en) * 1974-05-24 1976-01-13 The Upjohn Company Interferon induction
US4649141A (en) * 1978-02-13 1987-03-10 Smith Kline & French Laboratories Limited Pyrimidine compounds
US4656176A (en) * 1978-05-30 1987-04-07 Smithkline & French Laboratories Limited 2-thiazolyl, oxazolyl, triazolyl and thiadiazolyl alkylamino-3-nitro-heterocyclic compounds
US4238493A (en) 1978-05-30 1980-12-09 Smith Kline & French Laboratories Limited 2-(Substituted amino)-3-nitro-2,3-unsaturated nitrogen heterocycles
US4305945A (en) 1978-07-15 1981-12-15 Smith Kline & French Laboratories Limited Isoureas and isothioureas
US4439435A (en) * 1978-07-15 1984-03-27 Smith Kline & French Laboratories Ltd. Isoureas and isothioureas
WO1980000966A1 (en) * 1978-11-13 1980-05-15 Smith Kline French Lab New histamine h2-antagonists
US4496567A (en) * 1978-11-13 1985-01-29 Smith Kline & French Laboratories Limited Phenyl alkylaminopyrimidones
EP0013071A1 (en) * 1978-11-13 1980-07-09 Smith Kline & French Laboratories Limited Pyrimidinone derivatives, processes for preparing them and pharmaceutical compositions containing them
US4521418A (en) * 1979-02-21 1985-06-04 Smith Kline & French Laboratories Limited Guanidinothiazolyl derivatives
US5434157A (en) * 1979-03-19 1995-07-18 The Upjohn Company 6-aryl pyrimidine compounds and method for treating viral infections and inducing interferon production
US4507302A (en) * 1979-03-19 1985-03-26 The Upjohn Company Method for treating arthritis with 6-aryl pyrimidine compounds
US5002951A (en) * 1979-03-19 1991-03-26 The Upjohn Company Method for treating bacterial and protozoal infections
US4255428A (en) 1979-03-24 1981-03-10 Smith Kline & French Laboratories Limited 5-(Hydroxypyridylalkyl)-4-pyrimidones
EP0019450A1 (en) * 1979-05-15 1980-11-26 Takeda Chemical Industries, Ltd. Pyrimidine derivatives and their production and agricultural uses
US5554617A (en) * 1979-09-28 1996-09-10 The Upjohn Company Method for treating cancer with 6-aryl pyrimidine compounds
US4308272A (en) 1980-10-03 1981-12-29 The Upjohn Company Process for treating hypertension
US4460589A (en) * 1980-10-03 1984-07-17 The Upjohn Company Process for treating hypertension
EP0055692A1 (en) * 1980-12-15 1982-07-07 Sandoz Ag Novel pyrimidinyl ethers, their use as herbicides, herbicidal compositions comprising said pyrimidinyl ethers and processes for the preparation thereof
US4525477A (en) * 1981-12-02 1985-06-25 Smith Kline & French Laboratories Limited 2-Thiazolyl, isothiazolyl, oxazolyl and isoxazolyl alkylamino-3-nitro-heterocyclic compounds
US4593096A (en) * 1982-06-09 1986-06-03 The Upjohn Company Novel compounds and process for treating hypertension
US6495558B1 (en) 1999-01-22 2002-12-17 Amgen Inc. Kinase inhibitors

Also Published As

Publication number Publication date
IE31957B1 (en) 1973-02-21
CY682A (en) 1973-05-03
IE31957L (en) 1968-08-24
IL29496A (en) 1976-01-30

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Legal Events

Date Code Title Description
PS Patent sealed
PE20 Patent expired after termination of 20 years