CZ35494A3 - Process for preparing derivatives of beta-phenylisoserine and their utilization - Google Patents

Process for preparing derivatives of beta-phenylisoserine and their utilization Download PDF

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Publication number
CZ35494A3
CZ35494A3 CS94354A CS3549492A CZ35494A3 CZ 35494 A3 CZ35494 A3 CZ 35494A3 CS 94354 A CS94354 A CS 94354A CS 3549492 A CS3549492 A CS 3549492A CZ 35494 A3 CZ35494 A3 CZ 35494A3
Authority
CZ
Czechia
Prior art keywords
groups
mmol
group
added
phenyl
Prior art date
Application number
CS94354A
Other languages
Czech (cs)
English (en)
Inventor
Jean-No'el Denis
Andrew Greene
Alice Kanazawa
Original Assignee
Rhone Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa
Publication of CZ35494A3 publication Critical patent/CZ35494A3/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
CS94354A 1991-08-19 1992-08-17 Process for preparing derivatives of beta-phenylisoserine and their utilization CZ35494A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR919110398A FR2680506B1 (fr) 1991-08-19 1991-08-19 Procede de preparation de derives de la beta-phenylisoserine et leur utilisation.
PCT/FR1992/000795 WO1993004038A1 (fr) 1991-08-19 1992-08-17 PROCEDE DE PREPARATION DE DERIVES DE LA β-PHENYLISOSERINE ET LEUR UTILISATION

Publications (1)

Publication Number Publication Date
CZ35494A3 true CZ35494A3 (en) 1994-07-13

Family

ID=9416254

Family Applications (1)

Application Number Title Priority Date Filing Date
CS94354A CZ35494A3 (en) 1991-08-19 1992-08-17 Process for preparing derivatives of beta-phenylisoserine and their utilization

Country Status (16)

Country Link
EP (2) EP0528729A1 (cg-RX-API-DMAC10.html)
JP (1) JPH06510033A (cg-RX-API-DMAC10.html)
AU (1) AU2490492A (cg-RX-API-DMAC10.html)
CA (1) CA2113827A1 (cg-RX-API-DMAC10.html)
CZ (1) CZ35494A3 (cg-RX-API-DMAC10.html)
FI (1) FI940775A7 (cg-RX-API-DMAC10.html)
FR (1) FR2680506B1 (cg-RX-API-DMAC10.html)
HU (1) HUT68255A (cg-RX-API-DMAC10.html)
MX (1) MX9204635A (cg-RX-API-DMAC10.html)
NO (1) NO940027L (cg-RX-API-DMAC10.html)
NZ (1) NZ243972A (cg-RX-API-DMAC10.html)
SK (1) SK19094A3 (cg-RX-API-DMAC10.html)
TW (1) TW222620B (cg-RX-API-DMAC10.html)
WO (1) WO1993004038A1 (cg-RX-API-DMAC10.html)
YU (1) YU78092A (cg-RX-API-DMAC10.html)
ZA (1) ZA926189B (cg-RX-API-DMAC10.html)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5646176A (en) * 1992-12-24 1997-07-08 Bristol-Myers Squibb Company Phosphonooxymethyl ethers of taxane derivatives
CA2155304C (en) * 1993-02-05 2010-07-20 Charles Swindell Syntheses of paclitaxel, analogs and intermediates with variable a-ring side chains
US5684175A (en) * 1993-02-05 1997-11-04 Napro Biotherapeutics, Inc. C-2' hydroxyl-benzyl protected, N-carbamate protected (2R, 3S)- 3-phenylisoserine and production process therefor
US5580899A (en) * 1995-01-09 1996-12-03 The Liposome Company, Inc. Hydrophobic taxane derivatives
US5675025A (en) * 1995-06-07 1997-10-07 Napro Biotherapeutics, Inc. Paclitaxel synthesis from precursor compounds and methods of producing the same
US6107332A (en) 1995-09-12 2000-08-22 The Liposome Company, Inc. Hydrolysis-promoting hydrophobic taxane derivatives
US6051600A (en) * 1995-09-12 2000-04-18 Mayhew; Eric Liposomal hydrolysis-promoting hydrophobic taxane derivatives
US6107497A (en) * 1996-02-29 2000-08-22 Napro Biotherapeutics, Inc. Intermediate for use in docetaxel synthesis and production method therefor
US5688977A (en) * 1996-02-29 1997-11-18 Napro Biotherapeutics, Inc. Method for docetaxel synthesis
US5750737A (en) * 1996-09-25 1998-05-12 Sisti; Nicholas J. Method for paclitaxel synthesis
US6025516A (en) * 1998-10-14 2000-02-15 Chiragene, Inc. Resolution of 2-hydroxy-3-amino-3-phenylpropionamide and its conversion to C-13 sidechain of taxanes
US6452025B1 (en) 2001-04-25 2002-09-17 Napro Biotherapeutics, Inc. Three-step conversion of protected taxane ester to paclitaxel
ATE346084T1 (de) * 2002-02-27 2006-12-15 Ferring Bv Zwischenprodukte und verfahren zur herstellung von heptapeptid-oxytocinanaloga
BR112014031421A2 (pt) 2012-06-15 2017-06-27 Brigham & Womens Hospital Inc composições para tratamento de câncer e métodos para produção das mesmas
KR20160132496A (ko) 2014-04-03 2016-11-18 인빅터스 온콜로지 피비티. 엘티디. 초분자 조합 치료제

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2629818B1 (fr) * 1988-04-06 1990-11-16 Centre Nat Rech Scient Procede de preparation du taxol
FR2629819B1 (fr) * 1988-04-06 1990-11-16 Rhone Poulenc Sante Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii
FR2662441B1 (fr) * 1990-05-22 1992-10-23 Rhone Poulenc Sante Procede de preparation enantioselective de derives de la phenylisoserine.
FR2662440B1 (fr) * 1990-05-22 1992-07-31 Rhone Poulenc Sante Procede de preparation stereoselective de derives de la phenylisoserine.

Also Published As

Publication number Publication date
EP0599973A1 (fr) 1994-06-08
MX9204635A (es) 1993-02-01
AU2490492A (en) 1993-03-16
FR2680506A1 (fr) 1993-02-26
CA2113827A1 (fr) 1993-03-04
WO1993004038A1 (fr) 1993-03-04
FI940775A0 (fi) 1994-02-18
FR2680506B1 (fr) 1994-09-02
EP0528729A1 (fr) 1993-02-24
ZA926189B (en) 1993-03-01
FI940775L (fi) 1994-02-18
TW222620B (cg-RX-API-DMAC10.html) 1994-04-21
NO940027D0 (no) 1994-01-04
YU78092A (sh) 1995-10-03
SK19094A3 (en) 1994-09-07
HUT68255A (en) 1995-06-28
FI940775A7 (fi) 1994-02-18
HU9400478D0 (en) 1994-06-28
NZ243972A (en) 1994-11-25
NO940027L (no) 1994-01-04
JPH06510033A (ja) 1994-11-10

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