CY2022A - 8-Alkoxyquinolonecarboxylic acid and salts thereof excellent in the selective toxicity and process of preparing the same - Google Patents

8-Alkoxyquinolonecarboxylic acid and salts thereof excellent in the selective toxicity and process of preparing the same

Info

Publication number
CY2022A
CY2022A CY202298A CY202298A CY2022A CY 2022 A CY2022 A CY 2022A CY 202298 A CY202298 A CY 202298A CY 202298 A CY202298 A CY 202298A CY 2022 A CY2022 A CY 2022A
Authority
CY
Cyprus
Prior art keywords
salts
preparing
same
selective toxicity
alkoxyquinolonecarboxylic
Prior art date
Application number
CY202298A
Other languages
English (en)
Original Assignee
Kyorin Seiyaku Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26346239&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY2022(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Kyorin Seiyaku Kk filed Critical Kyorin Seiyaku Kk
Publication of CY2022A publication Critical patent/CY2022A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/22Oxygen atoms attached in position 2 or 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CY202298A 1986-01-21 1998-02-20 8-Alkoxyquinolonecarboxylic acid and salts thereof excellent in the selective toxicity and process of preparing the same CY2022A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP1088086 1986-01-21
JP61220149A JPH089597B2 (ja) 1986-01-21 1986-09-18 選択毒性に優れた8‐アルコキシキノロンカルボン酸およびその塩並びにその製造方法

Publications (1)

Publication Number Publication Date
CY2022A true CY2022A (en) 1998-02-20

Family

ID=26346239

Family Applications (1)

Application Number Title Priority Date Filing Date
CY202298A CY2022A (en) 1986-01-21 1998-02-20 8-Alkoxyquinolonecarboxylic acid and salts thereof excellent in the selective toxicity and process of preparing the same

Country Status (11)

Country Link
US (2) US4980470A (de)
EP (1) EP0230295B1 (de)
JP (1) JPH089597B2 (de)
KR (1) KR940007308B1 (de)
CN (1) CN1021052C (de)
CA (1) CA1340316C (de)
CY (1) CY2022A (de)
DE (2) DE3789878T2 (de)
HK (1) HK79797A (de)
HU (1) HU203339B (de)
NL (1) NL300110I2 (de)

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US5233091A (en) * 1988-06-21 1993-08-03 Pfizer Inc. 6-fluoro-1,4-dihydroquinol-4-one-3-carboxylic acid derivatives and intermediates therefor
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WO1990002123A1 (en) * 1988-08-23 1990-03-08 Pfizer Inc. Amino-substituted bridged azabicyclic quinolone carboxylic acids and esters
US5385913A (en) * 1989-10-06 1995-01-31 Pfizer Inc. 1,4-dihydro-4-oxo-3-quinoline derivatives as selectively toxic mammalian antibacterial agents
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CN110122493B (zh) * 2019-06-14 2022-04-12 山东省联合农药工业有限公司 喹诺酮类化合物用于防治有用植物中细菌性有害生物的用途
CN114716373B (zh) * 2022-04-14 2023-01-10 内蒙古源宏精细化工有限公司 一种加替沙星环合酯的制备方法
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Also Published As

Publication number Publication date
KR940007308B1 (ko) 1994-08-12
EP0230295A3 (en) 1987-11-04
NL300110I2 (nl) 2003-05-01
DE10299006I2 (de) 2002-11-07
EP0230295B1 (de) 1994-05-25
CN87100580A (zh) 1987-08-19
EP0230295A2 (de) 1987-07-29
DE10299006I1 (de) 2002-07-04
CN1021052C (zh) 1993-06-02
JPS62252772A (ja) 1987-11-04
HUT43583A (en) 1987-11-30
US5043450A (en) 1991-08-27
DE3789878T2 (de) 1995-01-05
AU6769087A (en) 1987-07-23
HU203339B (en) 1991-07-29
US4980470A (en) 1990-12-25
DE3789878D1 (de) 1994-06-30
NL300110I1 (nl) 2003-02-03
AU610491B2 (en) 1991-05-23
HK79797A (en) 1997-06-20
JPH089597B2 (ja) 1996-01-31
CA1340316C (en) 1999-01-12
KR870007128A (ko) 1987-08-17

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