HK79797A - 8-alkoxyquinolonecarboxylic acid and salts thereof excellent in the selective toxicity and process of preparing the same - Google Patents

8-alkoxyquinolonecarboxylic acid and salts thereof excellent in the selective toxicity and process of preparing the same

Info

Publication number
HK79797A
HK79797A HK79797A HK79797A HK79797A HK 79797 A HK79797 A HK 79797A HK 79797 A HK79797 A HK 79797A HK 79797 A HK79797 A HK 79797A HK 79797 A HK79797 A HK 79797A
Authority
HK
Hong Kong
Prior art keywords
salts
preparing
same
selective toxicity
alkoxyquinolonecarboxylic
Prior art date
Application number
HK79797A
Other languages
English (en)
Inventor
Kuniyoshi Masuzawa
Seigo Suzue
Keiji Hirai
Takayoshi Ishizaki
Original Assignee
Kyorin Seiyaku Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26346239&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK79797(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Kyorin Seiyaku Kk filed Critical Kyorin Seiyaku Kk
Publication of HK79797A publication Critical patent/HK79797A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/22—Oxygen atoms attached in position 2 or 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
HK79797A 1986-01-21 1997-06-12 8-alkoxyquinolonecarboxylic acid and salts thereof excellent in the selective toxicity and process of preparing the same HK79797A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP1088086 1986-01-21
JP61220149A JPH089597B2 (ja) 1986-01-21 1986-09-18 選択毒性に優れた８‐アルコキシキノロンカルボン酸およびその塩並びにその製造方法

Publications (1)

Publication Number Publication Date
HK79797A true HK79797A (en) 1997-06-20

Family

ID=26346239

Family Applications (1)

Application Number Title Priority Date Filing Date
HK79797A HK79797A (en) 1986-01-21 1997-06-12 8-alkoxyquinolonecarboxylic acid and salts thereof excellent in the selective toxicity and process of preparing the same

Country Status (11)

Country Link
US (2) US4980470A (xx)
EP (1) EP0230295B1 (xx)
JP (1) JPH089597B2 (xx)
KR (1) KR940007308B1 (xx)
CN (1) CN1021052C (xx)
CA (1) CA1340316C (xx)
CY (1) CY2022A (xx)
DE (2) DE3789878T2 (xx)
HK (1) HK79797A (xx)
HU (1) HU203339B (xx)
NL (1) NL300110I2 (xx)

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US5233091A (en) * 1988-06-21 1993-08-03 Pfizer Inc. 6-fluoro-1,4-dihydroquinol-4-one-3-carboxylic acid derivatives and intermediates therefor
JPH0674261B2 (ja) * 1988-06-21 1994-09-21 塩野義製薬株式会社 キノロンカルボン酸誘導体
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JP2016510750A (ja) 2013-03-08 2016-04-11 アラーガン、インコーポレイテッドＡｌｌｅｒｇａｎ，Ｉｎｃｏｒｐｏｒａｔｅｄ ステロイド薬と直接結合した抗生物質共役体
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KR101537911B1 (ko) * 2014-11-11 2015-07-23 한서대학교 산학협력단 제어 방출형 가티플록사신 제제 및 이의 제조방법
CN110122493B (zh) * 2019-06-14 2022-04-12 山东省联合农药工业有限公司 喹诺酮类化合物用于防治有用植物中细菌性有害生物的用途
CN114716373B (zh) * 2022-04-14 2023-01-10 内蒙古源宏精细化工有限公司 一种加替沙星环合酯的制备方法
CN114989165A (zh) * 2022-05-30 2022-09-02 青岛大学附属医院 一种抗持留菌和生物膜菌的化合物或组合物及其用途

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Also Published As

Publication number Publication date
NL300110I1 (nl) 2003-02-03
JPS62252772A (ja) 1987-11-04
US5043450A (en) 1991-08-27
NL300110I2 (nl) 2003-05-01
KR870007128A (ko) 1987-08-17
DE3789878T2 (de) 1995-01-05
HU203339B (en) 1991-07-29
EP0230295A3 (en) 1987-11-04
AU6769087A (en) 1987-07-23
HUT43583A (en) 1987-11-30
DE10299006I2 (de) 2002-11-07
CY2022A (en) 1998-02-20
AU610491B2 (en) 1991-05-23
US4980470A (en) 1990-12-25
CN87100580A (zh) 1987-08-19
EP0230295B1 (en) 1994-05-25
KR940007308B1 (ko) 1994-08-12
JPH089597B2 (ja) 1996-01-31
DE3789878D1 (de) 1994-06-30
CA1340316C (en) 1999-01-12
CN1021052C (zh) 1993-06-02
EP0230295A2 (en) 1987-07-29
DE10299006I1 (de) 2002-07-04

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