CY1119721T1 - Ετεροδιλειτουργικοι αναστολεις παν-σελεκτινης - Google Patents

Ετεροδιλειτουργικοι αναστολεις παν-σελεκτινης

Info

Publication number
CY1119721T1
CY1119721T1 CY20171101350T CY171101350T CY1119721T1 CY 1119721 T1 CY1119721 T1 CY 1119721T1 CY 20171101350 T CY20171101350 T CY 20171101350T CY 171101350 T CY171101350 T CY 171101350T CY 1119721 T1 CY1119721 T1 CY 1119721T1
Authority
CY
Cyprus
Prior art keywords
selectin
hydroderutical
suspensions
pan
class
Prior art date
Application number
CY20171101350T
Other languages
Greek (el)
English (en)
Inventor
John L. Magnani
John T. PATTON, Jr
Arun K. Sarkar
Sergei A. Svarovsky
Beat Ernst
Original Assignee
Glycomimetics, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glycomimetics, Inc. filed Critical Glycomimetics, Inc.
Publication of CY1119721T1 publication Critical patent/CY1119721T1/el

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    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/549—Sugars, nucleosides, nucleotides or nucleic acids
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
CY20171101350T 2005-09-02 2017-12-27 Ετεροδιλειτουργικοι αναστολεις παν-σελεκτινης CY1119721T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US71399405P 2005-09-02 2005-09-02
EP06814078A EP1934236B1 (en) 2005-09-02 2006-09-01 Heterobifunctional pan-selectin inhibitors

Publications (1)

Publication Number Publication Date
CY1119721T1 true CY1119721T1 (el) 2018-06-27

Family

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CY20171101350T CY1119721T1 (el) 2005-09-02 2017-12-27 Ετεροδιλειτουργικοι αναστολεις παν-σελεκτινης

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US (6) US7728117B2 (US07728117-20100601-C00004.png)
EP (2) EP2264043B1 (US07728117-20100601-C00004.png)
JP (2) JP5209476B2 (US07728117-20100601-C00004.png)
CN (2) CN101287741B (US07728117-20100601-C00004.png)
AU (1) AU2006284578B2 (US07728117-20100601-C00004.png)
CA (1) CA2670130A1 (US07728117-20100601-C00004.png)
CY (1) CY1119721T1 (US07728117-20100601-C00004.png)
DK (2) DK2264043T3 (US07728117-20100601-C00004.png)
ES (2) ES2397850T3 (US07728117-20100601-C00004.png)
HK (1) HK1122041A1 (US07728117-20100601-C00004.png)
HU (1) HUE038246T2 (US07728117-20100601-C00004.png)
LT (1) LT2264043T (US07728117-20100601-C00004.png)
PL (2) PL2264043T3 (US07728117-20100601-C00004.png)
PT (2) PT1934236E (US07728117-20100601-C00004.png)
SI (2) SI1934236T1 (US07728117-20100601-C00004.png)
WO (1) WO2007028050A1 (US07728117-20100601-C00004.png)

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