CY1114628T1 - Θειαζολοπυριδιν-2-υλοξυ-φαινυλ και θειαζολοπυραζιν-2-υλοξυ-φαινυλ αμινες ως ρυθμιστες υδρολασης λευκοτριενιου α4 - Google Patents

Θειαζολοπυριδιν-2-υλοξυ-φαινυλ και θειαζολοπυραζιν-2-υλοξυ-φαινυλ αμινες ως ρυθμιστες υδρολασης λευκοτριενιου α4

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Publication number
CY1114628T1
CY1114628T1 CY20131101029T CY131101029T CY1114628T1 CY 1114628 T1 CY1114628 T1 CY 1114628T1 CY 20131101029 T CY20131101029 T CY 20131101029T CY 131101029 T CY131101029 T CY 131101029T CY 1114628 T1 CY1114628 T1 CY 1114628T1
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CY
Cyprus
Prior art keywords
yloxy
thiazolopyridine
phenyl
leukotriene
regulators
Prior art date
Application number
CY20131101029T
Other languages
English (en)
Inventor
Genesis M Bacani
Diego Broggini
Eugene Y Cheung
Christa C Chrovian
Xiaohu Deng
Anne M Fourine
Laurent Gomez
Cheryl A Grice
Aaron M Kearney
Adrienne M Landry-Bayle
Alice Lee-Dutra
Jimmy T Liang
Susanne Lochner
Neelakandha S Mani
Alejandro Santillan
Kathleen C Sappey
Kia Sepassi
Virginia M Tanis
Alvah T Wickboldt
John J M Wiener
Hartmut Zinser
Original Assignee
Janssen Pharmaceutica N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica N.V. filed Critical Janssen Pharmaceutica N.V.
Publication of CY1114628T1 publication Critical patent/CY1114628T1/el

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    • C07D498/04—Ortho-condensed systems
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    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof

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Abstract

Περιγράφονται θειαζολοπυριδιν-2-υλοξυ-φαινύλ και θειαζολοπυραζιν-2-υλοξυ-φαινυλ αμίνης ενώσεις, οι οποίες είναι χρήσιμες ως ρυθμιστές υδρολάσης LTA4 (LTA4H). Τέτοιες ενώσεις μπορεί να χρησιμοποιηθούν σε φαρμακευτικές συνθέσεις και μεθόδους για τη ρύθμιση LTA4H και για τη θεραπεία καταστάσεων ασθένειας, διαταραχών και παθήσεων που προκαλούνται από δραστικότητα υδρολάσης LTA4.
CY20131101029T 2008-04-11 2013-11-20 Θειαζολοπυριδιν-2-υλοξυ-φαινυλ και θειαζολοπυραζιν-2-υλοξυ-φαινυλ αμινες ως ρυθμιστες υδρολασης λευκοτριενιου α4 CY1114628T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4434908P 2008-04-11 2008-04-11
US14912909P 2009-02-02 2009-02-02
EP09729596.8A EP2268646B9 (en) 2008-04-11 2009-04-09 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene a4 hydrolase

Publications (1)

Publication Number Publication Date
CY1114628T1 true CY1114628T1 (el) 2016-10-05

Family

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CY20131101029T CY1114628T1 (el) 2008-04-11 2013-11-20 Θειαζολοπυριδιν-2-υλοξυ-φαινυλ και θειαζολοπυραζιν-2-υλοξυ-φαινυλ αμινες ως ρυθμιστες υδρολασης λευκοτριενιου α4

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SI (2) SI2336125T1 (el)
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TW (2) TW201420100A (el)
UY (1) UY31760A (el)
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