CY1112709T1 - Ανταγωνιστες υποδοχεα 5-ητ7 - Google Patents

Ανταγωνιστες υποδοχεα 5-ητ7

Info

Publication number
CY1112709T1
CY1112709T1 CY20121100400T CY121100400T CY1112709T1 CY 1112709 T1 CY1112709 T1 CY 1112709T1 CY 20121100400 T CY20121100400 T CY 20121100400T CY 121100400 T CY121100400 T CY 121100400T CY 1112709 T1 CY1112709 T1 CY 1112709T1
Authority
CY
Cyprus
Prior art keywords
competitive
receptors
competitive receptors
migraine
formula
Prior art date
Application number
CY20121100400T
Other languages
Greek (el)
English (en)
Inventor
Valentina O Badescu
Sandra Ann Filla
Peter Thaddeus Gallagher
Maria Ann Whatton
Original Assignee
Eli Lilly And Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly And Company filed Critical Eli Lilly And Company
Publication of CY1112709T1 publication Critical patent/CY1112709T1/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CY20121100400T 2007-10-12 2012-04-26 Ανταγωνιστες υποδοχεα 5-ητ7 CY1112709T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US97946407P 2007-10-12 2007-10-12
EP08836911A EP2201002B1 (en) 2007-10-12 2008-09-30 5-ht7 receptor antagonists

Publications (1)

Publication Number Publication Date
CY1112709T1 true CY1112709T1 (el) 2016-02-10

Family

ID=40134870

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20121100400T CY1112709T1 (el) 2007-10-12 2012-04-26 Ανταγωνιστες υποδοχεα 5-ητ7

Country Status (19)

Country Link
US (1) US7910588B2 (cg-RX-API-DMAC7.html)
EP (1) EP2201002B1 (cg-RX-API-DMAC7.html)
JP (1) JP5291716B2 (cg-RX-API-DMAC7.html)
KR (1) KR101161070B1 (cg-RX-API-DMAC7.html)
CN (1) CN101821257B (cg-RX-API-DMAC7.html)
AT (1) ATE548365T1 (cg-RX-API-DMAC7.html)
AU (1) AU2008311154B2 (cg-RX-API-DMAC7.html)
BR (1) BRPI0818450A2 (cg-RX-API-DMAC7.html)
CA (1) CA2699674C (cg-RX-API-DMAC7.html)
CY (1) CY1112709T1 (cg-RX-API-DMAC7.html)
DK (1) DK2201002T3 (cg-RX-API-DMAC7.html)
EA (1) EA016787B1 (cg-RX-API-DMAC7.html)
ES (1) ES2380756T3 (cg-RX-API-DMAC7.html)
HR (1) HRP20120257T1 (cg-RX-API-DMAC7.html)
MX (1) MX2010003986A (cg-RX-API-DMAC7.html)
PL (1) PL2201002T3 (cg-RX-API-DMAC7.html)
PT (1) PT2201002E (cg-RX-API-DMAC7.html)
SI (1) SI2201002T1 (cg-RX-API-DMAC7.html)
WO (1) WO2009048765A1 (cg-RX-API-DMAC7.html)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI396857B (zh) * 2009-12-30 2013-05-21 Etron Technology Inc 晶片測試電路
MX2014004210A (es) 2011-10-11 2014-05-28 Ucb Pharma Sa Derivados de 2-oxo-piperidinilo.
ES2804545T3 (es) 2013-03-11 2021-02-08 Univ Temple Nuevos moduladores de la actividad del receptor de 5-hidroxitriptamina 7 y su método de uso
TW201601632A (zh) * 2013-11-20 2016-01-16 杜邦股份有限公司 1-芳基-3-烷基吡唑殺蟲劑
EP3200589A4 (en) 2014-09-10 2018-07-25 Temple University Of The Commonwealth System Of Higher Education Novel 5-hydroxytryptamine receptor 7 activity modulators and their method of use
KR102900157B1 (ko) 2016-11-15 2025-12-12 템플 유니버시티-오브 더 커먼웰쓰 시스템 오브 하이어 에듀케이션 5-히드록시트립타민 수용체 7의 신규 조절제 및 이의 사용 방법
JP7365238B2 (ja) 2017-03-21 2023-10-19 テンプル・ユニバーシティ-オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション 5-ヒドロキシトリプタミン受容体7調節物質および治療剤としてのその使用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6465467B1 (en) 1999-05-21 2002-10-15 Biovitrum Ab Certain aryl-aliphatic and heteroaryl-aliphatic piperazinyl pyrazines and their use in the treatment of serotonin-related diseases
US20030008880A1 (en) 2001-05-02 2003-01-09 Pfizer Inc. 4-(2-Pyridyl) piperizines having 5HT7 receptor agonist activity
WO2004067703A2 (en) * 2003-01-31 2004-08-12 Pfizer Products Inc. 5ht7 antagonists and inverse agonists
US7211783B2 (en) 2004-01-09 2007-05-01 Tamperproof Container Licensing Corp. Tamper-proof container
JP2008501031A (ja) 2004-05-28 2008-01-17 バーテックス ファーマシューティカルズ インコーポレイテッド ムスカリン受容体のモジュレーター
TW200914020A (en) * 2007-08-28 2009-04-01 Lilly Co Eli Substituted piperazinyl pyrazines and pyridines as 5-HT7 receptor antagonists

Also Published As

Publication number Publication date
KR20100054853A (ko) 2010-05-25
EA201070462A1 (ru) 2010-10-29
CN101821257A (zh) 2010-09-01
JP5291716B2 (ja) 2013-09-18
CA2699674A1 (en) 2009-04-16
AU2008311154B2 (en) 2013-09-26
EA016787B1 (ru) 2012-07-30
AU2008311154A1 (en) 2009-04-16
CN101821257B (zh) 2013-05-22
BRPI0818450A2 (pt) 2015-05-12
JP2011500575A (ja) 2011-01-06
SI2201002T1 (sl) 2012-04-30
US20100197700A1 (en) 2010-08-05
ATE548365T1 (de) 2012-03-15
DK2201002T3 (da) 2012-04-10
EP2201002B1 (en) 2012-03-07
US7910588B2 (en) 2011-03-22
HRP20120257T1 (hr) 2012-04-30
CA2699674C (en) 2013-07-16
EP2201002A1 (en) 2010-06-30
PT2201002E (pt) 2012-04-27
ES2380756T3 (es) 2012-05-18
WO2009048765A1 (en) 2009-04-16
KR101161070B1 (ko) 2012-07-13
PL2201002T3 (pl) 2012-07-31
MX2010003986A (es) 2010-04-27

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