ATE474574T1 - Imidazoazephinonverbindungen - Google Patents
ImidazoazephinonverbindungenInfo
- Publication number
- ATE474574T1 ATE474574T1 AT07795237T AT07795237T ATE474574T1 AT E474574 T1 ATE474574 T1 AT E474574T1 AT 07795237 T AT07795237 T AT 07795237T AT 07795237 T AT07795237 T AT 07795237T AT E474574 T1 ATE474574 T1 AT E474574T1
- Authority
- AT
- Austria
- Prior art keywords
- compounds
- imidazoazephinone
- formula
- treatment
- methods
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 208000023275 Autoimmune disease Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Immunology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Transplantation (AREA)
- Cardiology (AREA)
- Endocrinology (AREA)
- Vascular Medicine (AREA)
- Emergency Medicine (AREA)
- Urology & Nephrology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Dermatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US80877006P | 2006-05-26 | 2006-05-26 | |
| PCT/US2007/012298 WO2007139833A2 (en) | 2006-05-26 | 2007-05-24 | Imidazoazephinone compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE474574T1 true ATE474574T1 (de) | 2010-08-15 |
Family
ID=38668997
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT07795237T ATE474574T1 (de) | 2006-05-26 | 2007-05-24 | Imidazoazephinonverbindungen |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US7985746B2 (de) |
| EP (1) | EP2021003B1 (de) |
| JP (1) | JP2009538312A (de) |
| AT (1) | ATE474574T1 (de) |
| DE (1) | DE602007007934D1 (de) |
| ES (1) | ES2347837T3 (de) |
| WO (1) | WO2007139833A2 (de) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG158091A1 (en) * | 2006-05-26 | 2010-01-29 | Eisai R&D Man Co Ltd | Imidazoazepinone compounds |
| KR20100088695A (ko) * | 2007-11-15 | 2010-08-10 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 거울상 이성질체가 강화된 이미다조아제피논 화합물 |
| US20090197867A1 (en) * | 2007-11-15 | 2009-08-06 | Mark Spyvee | Enantiomerically enriched imidazoazepinone compounds |
| EP2217242A1 (de) * | 2007-11-15 | 2010-08-18 | Eisai R&D Management Co., Ltd. | Anwendungsverfahren |
| JP2011504878A (ja) * | 2007-11-26 | 2011-02-17 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | イミダゾアゼピノン化合物の製造方法 |
| KR20110086769A (ko) * | 2008-11-23 | 2011-07-29 | 화이자 인코포레이티드 | 베타 세크레타제 억제제로서의 락탐 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2010742A1 (en) * | 1989-03-03 | 1990-09-03 | Kenji Koga | Azacyclooctadiene compound and pharmaceutical use |
| JPH04266886A (ja) | 1991-02-20 | 1992-09-22 | Eisai Co Ltd | アザシクロオクタジエン誘導体 |
| EP1619193A4 (de) | 2003-04-18 | 2010-08-11 | Ono Pharmaceutical Co | Spiropiperidinverbindung und deren medizinische verwendung |
| WO2006079119A2 (en) * | 2005-01-20 | 2006-07-27 | President And Fellows Of Harvard College | Modulation of th2 lineage commitment by t-bet |
| TW200724140A (en) * | 2005-05-27 | 2007-07-01 | Eisai Co Ltd | Hydantoin compounds |
| SG158091A1 (en) * | 2006-05-26 | 2010-01-29 | Eisai R&D Man Co Ltd | Imidazoazepinone compounds |
-
2007
- 2007-05-24 JP JP2009512128A patent/JP2009538312A/ja active Pending
- 2007-05-24 WO PCT/US2007/012298 patent/WO2007139833A2/en not_active Ceased
- 2007-05-24 AT AT07795237T patent/ATE474574T1/de not_active IP Right Cessation
- 2007-05-24 US US12/299,864 patent/US7985746B2/en not_active Expired - Fee Related
- 2007-05-24 EP EP07795237A patent/EP2021003B1/de active Active
- 2007-05-24 DE DE602007007934T patent/DE602007007934D1/de active Active
- 2007-05-24 ES ES07795237T patent/ES2347837T3/es active Active
Also Published As
| Publication number | Publication date |
|---|---|
| ES2347837T3 (es) | 2010-11-04 |
| WO2007139833A2 (en) | 2007-12-06 |
| WO2007139833A3 (en) | 2008-01-31 |
| DE602007007934D1 (en) | 2010-09-02 |
| US20090131405A1 (en) | 2009-05-21 |
| US7985746B2 (en) | 2011-07-26 |
| EP2021003A2 (de) | 2009-02-11 |
| JP2009538312A (ja) | 2009-11-05 |
| EP2021003B1 (de) | 2010-07-21 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |