CY1108275T1 - Χημικες ενωσεις - Google Patents
Χημικες ενωσειςInfo
- Publication number
- CY1108275T1 CY1108275T1 CY20081100887T CY081100887T CY1108275T1 CY 1108275 T1 CY1108275 T1 CY 1108275T1 CY 20081100887 T CY20081100887 T CY 20081100887T CY 081100887 T CY081100887 T CY 081100887T CY 1108275 T1 CY1108275 T1 CY 1108275T1
- Authority
- CY
- Cyprus
- Prior art keywords
- chemical compounds
- novel compounds
- cancer
- formula
- treatment
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Oncology (AREA)
- Pain & Pain Management (AREA)
- Transplantation (AREA)
- Ophthalmology & Optometry (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Hematology (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Αυτή η εφεύρεση αναφέρεται σε νέες ενώσεις του τύπου (Ι)· και στις φαρμακευτικές τους συνθέσεις και τις μεθόδους χρήσης τους. Αυτές οι νέες ενώσεις παρέχουν μία θεραπεία για τον καρκίνο.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US65357505P | 2005-02-16 | 2005-02-16 | |
US74213805P | 2005-12-01 | 2005-12-01 | |
EP06709750A EP1853588B1 (en) | 2005-02-16 | 2006-02-15 | Chemical compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1108275T1 true CY1108275T1 (el) | 2014-02-12 |
Family
ID=36168456
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20081100887T CY1108275T1 (el) | 2005-02-16 | 2008-08-21 | Χημικες ενωσεις |
Country Status (22)
Country | Link |
---|---|
US (2) | US8129403B2 (el) |
EP (1) | EP1853588B1 (el) |
JP (1) | JP5001179B2 (el) |
KR (1) | KR101362621B1 (el) |
AT (1) | ATE398613T1 (el) |
AU (1) | AU2006215386B2 (el) |
BR (1) | BRPI0607455A2 (el) |
CA (1) | CA2597813C (el) |
CY (1) | CY1108275T1 (el) |
DE (1) | DE602006001515D1 (el) |
DK (1) | DK1853588T3 (el) |
ES (1) | ES2308731T3 (el) |
HK (1) | HK1114375A1 (el) |
IL (1) | IL185063A (el) |
MX (1) | MX2007009843A (el) |
NO (1) | NO20073788L (el) |
NZ (1) | NZ561525A (el) |
PL (1) | PL1853588T3 (el) |
PT (1) | PT1853588E (el) |
RU (1) | RU2405780C2 (el) |
SI (1) | SI1853588T1 (el) |
WO (1) | WO2006087530A1 (el) |
Families Citing this family (51)
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PT2383268E (pt) * | 2005-02-04 | 2015-12-21 | Astrazeneca Ab | Derivados de pirazolilaminopiridina úteis como inibidores de quinase |
PT1853588E (pt) | 2005-02-16 | 2008-08-25 | Astrazeneca Ab | Compostos químicos |
KR20080015409A (ko) * | 2005-05-16 | 2008-02-19 | 아스트라제네카 아베 | 티로신 키나제 억제제로서 유용한 피라졸릴아미노피리미딘 유도체 |
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CN101679432B (zh) * | 2006-10-19 | 2015-04-22 | 西格诺药品有限公司 | 杂芳基化合物、其组合物及其作为蛋白激酶抑制剂的用途 |
IN2009CN02154A (el) * | 2006-10-20 | 2015-08-07 | Organon Nv | |
CN101679429A (zh) * | 2007-04-18 | 2010-03-24 | 阿斯利康(瑞典)有限公司 | 5-氨基吡唑-3-基-3h-咪唑并[4,5-b]吡啶衍生物及其治疗癌的用途 |
UA99459C2 (en) * | 2007-05-04 | 2012-08-27 | Астразенека Аб | 9-(pyrazol-3-yl)- 9h-purine-2-amine and 3-(pyraz0l-3-yl)-3h-imidazo[4,5-b]pyridin-5-amine derivatives and their use for the treatment of cancer |
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-
2006
- 2006-02-15 PT PT06709750T patent/PT1853588E/pt unknown
- 2006-02-15 MX MX2007009843A patent/MX2007009843A/es active IP Right Grant
- 2006-02-15 PL PL06709750T patent/PL1853588T3/pl unknown
- 2006-02-15 AU AU2006215386A patent/AU2006215386B2/en not_active Ceased
- 2006-02-15 DK DK06709750T patent/DK1853588T3/da active
- 2006-02-15 AT AT06709750T patent/ATE398613T1/de active
- 2006-02-15 EP EP06709750A patent/EP1853588B1/en not_active Not-in-force
- 2006-02-15 CA CA2597813A patent/CA2597813C/en not_active Expired - Fee Related
- 2006-02-15 ES ES06709750T patent/ES2308731T3/es active Active
- 2006-02-15 DE DE602006001515T patent/DE602006001515D1/de active Active
- 2006-02-15 US US11/816,374 patent/US8129403B2/en not_active Expired - Fee Related
- 2006-02-15 WO PCT/GB2006/000513 patent/WO2006087530A1/en active IP Right Grant
- 2006-02-15 KR KR1020077020887A patent/KR101362621B1/ko not_active IP Right Cessation
- 2006-02-15 JP JP2007555688A patent/JP5001179B2/ja not_active Expired - Fee Related
- 2006-02-15 BR BRPI0607455-3A patent/BRPI0607455A2/pt not_active IP Right Cessation
- 2006-02-15 RU RU2007134396/04A patent/RU2405780C2/ru not_active IP Right Cessation
- 2006-02-15 NZ NZ561525A patent/NZ561525A/en not_active IP Right Cessation
- 2006-02-15 SI SI200630060T patent/SI1853588T1/sl unknown
-
2007
- 2007-07-20 NO NO20073788A patent/NO20073788L/no not_active Application Discontinuation
- 2007-08-06 IL IL185063A patent/IL185063A/en not_active IP Right Cessation
-
2008
- 2008-03-07 HK HK08102715.2A patent/HK1114375A1/xx not_active IP Right Cessation
- 2008-08-21 CY CY20081100887T patent/CY1108275T1/el unknown
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- 2012-01-25 US US13/357,848 patent/US20120122892A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
NO20073788L (no) | 2007-09-03 |
CA2597813C (en) | 2014-04-22 |
PL1853588T3 (pl) | 2008-11-28 |
RU2007134396A (ru) | 2009-03-27 |
KR20070103773A (ko) | 2007-10-24 |
IL185063A (en) | 2012-01-31 |
IL185063A0 (en) | 2007-12-03 |
ES2308731T3 (es) | 2008-12-01 |
AU2006215386A1 (en) | 2006-08-24 |
DE602006001515D1 (de) | 2008-07-31 |
MX2007009843A (es) | 2007-08-23 |
EP1853588B1 (en) | 2008-06-18 |
EP1853588A1 (en) | 2007-11-14 |
BRPI0607455A2 (pt) | 2009-09-01 |
US20120122892A1 (en) | 2012-05-17 |
PT1853588E (pt) | 2008-08-25 |
ATE398613T1 (de) | 2008-07-15 |
US20080176872A1 (en) | 2008-07-24 |
HK1114375A1 (en) | 2008-10-31 |
RU2405780C2 (ru) | 2010-12-10 |
CA2597813A1 (en) | 2006-08-24 |
DK1853588T3 (da) | 2008-09-15 |
WO2006087530A1 (en) | 2006-08-24 |
US8129403B2 (en) | 2012-03-06 |
AU2006215386B2 (en) | 2009-06-11 |
JP5001179B2 (ja) | 2012-08-15 |
JP2008530190A (ja) | 2008-08-07 |
KR101362621B1 (ko) | 2014-02-13 |
SI1853588T1 (sl) | 2008-10-31 |
NZ561525A (en) | 2010-11-26 |
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