PT2201002E - Antagonistas de receptores 5-ht7 - Google Patents
Antagonistas de receptores 5-ht7 Download PDFInfo
- Publication number
- PT2201002E PT2201002E PT08836911T PT08836911T PT2201002E PT 2201002 E PT2201002 E PT 2201002E PT 08836911 T PT08836911 T PT 08836911T PT 08836911 T PT08836911 T PT 08836911T PT 2201002 E PT2201002 E PT 2201002E
- Authority
- PT
- Portugal
- Prior art keywords
- methyl
- tetrahydro
- ylmethyl
- pyrazol
- mmol
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US97946407P | 2007-10-12 | 2007-10-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PT2201002E true PT2201002E (pt) | 2012-04-27 |
Family
ID=40134870
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT08836911T PT2201002E (pt) | 2007-10-12 | 2008-09-30 | Antagonistas de receptores 5-ht7 |
Country Status (19)
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI396857B (zh) * | 2009-12-30 | 2013-05-21 | Etron Technology Inc | 晶片測試電路 |
| MX2014004210A (es) | 2011-10-11 | 2014-05-28 | Ucb Pharma Sa | Derivados de 2-oxo-piperidinilo. |
| ES2804545T3 (es) | 2013-03-11 | 2021-02-08 | Univ Temple | Nuevos moduladores de la actividad del receptor de 5-hidroxitriptamina 7 y su método de uso |
| TW201601632A (zh) * | 2013-11-20 | 2016-01-16 | 杜邦股份有限公司 | １－芳基－３－烷基吡唑殺蟲劑 |
| EP3200589A4 (en) | 2014-09-10 | 2018-07-25 | Temple University Of The Commonwealth System Of Higher Education | Novel 5-hydroxytryptamine receptor 7 activity modulators and their method of use |
| KR102900157B1 (ko) | 2016-11-15 | 2025-12-12 | 템플 유니버시티-오브 더 커먼웰쓰 시스템 오브 하이어 에듀케이션 | 5-히드록시트립타민 수용체 7의 신규 조절제 및 이의 사용 방법 |
| JP7365238B2 (ja) | 2017-03-21 | 2023-10-19 | テンプル・ユニバーシティ－オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション | ５－ヒドロキシトリプタミン受容体７調節物質および治療剤としてのその使用 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6465467B1 (en) | 1999-05-21 | 2002-10-15 | Biovitrum Ab | Certain aryl-aliphatic and heteroaryl-aliphatic piperazinyl pyrazines and their use in the treatment of serotonin-related diseases |
| US20030008880A1 (en) | 2001-05-02 | 2003-01-09 | Pfizer Inc. | 4-(2-Pyridyl) piperizines having 5HT7 receptor agonist activity |
| WO2004067703A2 (en) * | 2003-01-31 | 2004-08-12 | Pfizer Products Inc. | 5ht7 antagonists and inverse agonists |
| US7211783B2 (en) | 2004-01-09 | 2007-05-01 | Tamperproof Container Licensing Corp. | Tamper-proof container |
| JP2008501031A (ja) | 2004-05-28 | 2008-01-17 | バーテックス ファーマシューティカルズ インコーポレイテッド | ムスカリン受容体のモジュレーター |
| TW200914020A (en) * | 2007-08-28 | 2009-04-01 | Lilly Co Eli | Substituted piperazinyl pyrazines and pyridines as 5-HT7 receptor antagonists |
-
2008
- 2008-09-30 WO PCT/US2008/078294 patent/WO2009048765A1/en not_active Ceased
- 2008-09-30 HR HR20120257T patent/HRP20120257T1/hr unknown
- 2008-09-30 JP JP2010528941A patent/JP5291716B2/ja not_active Expired - Fee Related
- 2008-09-30 EP EP08836911A patent/EP2201002B1/en not_active Not-in-force
- 2008-09-30 CN CN2008801107600A patent/CN101821257B/zh not_active Expired - Fee Related
- 2008-09-30 BR BRPI0818450 patent/BRPI0818450A2/pt active Search and Examination
- 2008-09-30 EA EA201070462A patent/EA016787B1/ru not_active IP Right Cessation
- 2008-09-30 AU AU2008311154A patent/AU2008311154B2/en not_active Ceased
- 2008-09-30 KR KR1020107007725A patent/KR101161070B1/ko not_active Expired - Fee Related
- 2008-09-30 US US12/678,345 patent/US7910588B2/en not_active Expired - Fee Related
- 2008-09-30 PT PT08836911T patent/PT2201002E/pt unknown
- 2008-09-30 DK DK08836911.1T patent/DK2201002T3/da active
- 2008-09-30 SI SI200830580T patent/SI2201002T1/sl unknown
- 2008-09-30 ES ES08836911T patent/ES2380756T3/es active Active
- 2008-09-30 AT AT08836911T patent/ATE548365T1/de active
- 2008-09-30 PL PL08836911T patent/PL2201002T3/pl unknown
- 2008-09-30 MX MX2010003986A patent/MX2010003986A/es active IP Right Grant
- 2008-09-30 CA CA2699674A patent/CA2699674C/en not_active Expired - Fee Related
-
2012
- 2012-04-26 CY CY20121100400T patent/CY1112709T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR20100054853A (ko) | 2010-05-25 |
| EA201070462A1 (ru) | 2010-10-29 |
| CN101821257A (zh) | 2010-09-01 |
| JP5291716B2 (ja) | 2013-09-18 |
| CA2699674A1 (en) | 2009-04-16 |
| AU2008311154B2 (en) | 2013-09-26 |
| EA016787B1 (ru) | 2012-07-30 |
| AU2008311154A1 (en) | 2009-04-16 |
| CN101821257B (zh) | 2013-05-22 |
| BRPI0818450A2 (pt) | 2015-05-12 |
| JP2011500575A (ja) | 2011-01-06 |
| SI2201002T1 (sl) | 2012-04-30 |
| US20100197700A1 (en) | 2010-08-05 |
| ATE548365T1 (de) | 2012-03-15 |
| DK2201002T3 (da) | 2012-04-10 |
| CY1112709T1 (el) | 2016-02-10 |
| EP2201002B1 (en) | 2012-03-07 |
| US7910588B2 (en) | 2011-03-22 |
| HRP20120257T1 (hr) | 2012-04-30 |
| CA2699674C (en) | 2013-07-16 |
| EP2201002A1 (en) | 2010-06-30 |
| ES2380756T3 (es) | 2012-05-18 |
| WO2009048765A1 (en) | 2009-04-16 |
| KR101161070B1 (ko) | 2012-07-13 |
| PL2201002T3 (pl) | 2012-07-31 |
| MX2010003986A (es) | 2010-04-27 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ES2395872T3 (es) | 2-[4-(Pirazol-4-ilalquil)piperazin-1-il]-3-fenil pirazinas y piridinas y 3-[4-(pirazol-4-ilalquil)piperazin-1-il]-2-fenil piridinas como antagonistas del receptor de 5-HT7 | |
| PT2201002E (pt) | Antagonistas de receptores 5-ht7 | |
| WO2015152367A1 (ja) | オキソ複素環誘導体 | |
| JPWO2013187466A1 (ja) | 分岐鎖アルキルヘテロ芳香環誘導体 | |
| EP1265870A1 (en) | New ccr5 modulators: benzimidazoles or benzotriazoles | |
| JP5685440B2 (ja) | ３位において二置換されているインドール−２−オン誘導体、これらの調製およびこれらの治療上の使用 | |
| AU2008293715B2 (en) | Substituted piperazinyl pyrazines and pyridines as 5-HT7 receptor antagonists | |
| CN101124216A (zh) | 杂环MCHr1拮抗剂及其在治疗中的用途 |