CU20150176A7 - Derivados de prodroga de triazolpiridinas sustituídas - Google Patents
Derivados de prodroga de triazolpiridinas sustituídasInfo
- Publication number
- CU20150176A7 CU20150176A7 CUP2015000176A CU20150176A CU20150176A7 CU 20150176 A7 CU20150176 A7 CU 20150176A7 CU P2015000176 A CUP2015000176 A CU P2015000176A CU 20150176 A CU20150176 A CU 20150176A CU 20150176 A7 CU20150176 A7 CU 20150176A7
- Authority
- CU
- Cuba
- Prior art keywords
- derivatives
- triazolpiridines
- substituted
- supply
- mps
- Prior art date
Links
- 229940125502 MPS1 kinase inhibitor Drugs 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 229940002612 prodrug Drugs 0.000 abstract 1
- 239000000651 prodrug Substances 0.000 abstract 1
- 238000011321 prophylaxis Methods 0.000 abstract 1
- 238000011282 treatment Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
- C07K5/06052—Val-amino acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06086—Dipeptides with the first amino acid being basic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Derivados de prodroga de inhibidores de la quinasa Mps-1, procesos para su preparación y su uso en el tratamiento y/o la profilaxis de enfermedades.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP13171508 | 2013-06-11 | ||
PCT/EP2014/061779 WO2014198647A2 (en) | 2013-06-11 | 2014-06-06 | Prodrug derivatives of substituted triazolopyridines |
Publications (1)
Publication Number | Publication Date |
---|---|
CU20150176A7 true CU20150176A7 (es) | 2016-05-30 |
Family
ID=48576905
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CUP2015000176A CU20150176A7 (es) | 2013-06-11 | 2015-12-11 | Derivados de prodroga de triazolpiridinas sustituídas |
Country Status (35)
Country | Link |
---|---|
US (1) | US9586958B2 (es) |
EP (1) | EP3008062B1 (es) |
JP (1) | JP2016526534A (es) |
KR (1) | KR20160019492A (es) |
CN (1) | CN105377848A (es) |
AP (1) | AP2015008898A0 (es) |
AR (1) | AR096585A1 (es) |
AU (1) | AU2014280356A1 (es) |
CA (1) | CA2914745A1 (es) |
CL (1) | CL2015003605A1 (es) |
CR (1) | CR20150659A (es) |
CU (1) | CU20150176A7 (es) |
DK (1) | DK3008062T3 (es) |
DO (1) | DOP2015000299A (es) |
EA (1) | EA201600002A1 (es) |
ES (1) | ES2626790T3 (es) |
HK (1) | HK1221955A1 (es) |
HR (1) | HRP20170717T1 (es) |
HU (1) | HUE033131T2 (es) |
IL (1) | IL242847A0 (es) |
LT (1) | LT3008062T (es) |
MA (1) | MA38654B1 (es) |
MX (1) | MX2015017119A (es) |
NI (1) | NI201500176A (es) |
PE (1) | PE20160156A1 (es) |
PH (1) | PH12015502746A1 (es) |
PL (1) | PL3008062T3 (es) |
PT (1) | PT3008062T (es) |
RS (1) | RS56034B1 (es) |
SG (1) | SG11201509858QA (es) |
SI (1) | SI3008062T1 (es) |
TN (1) | TN2015000545A1 (es) |
UY (1) | UY35610A (es) |
WO (1) | WO2014198647A2 (es) |
ZA (1) | ZA201508868B (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MA41136A (fr) * | 2014-12-09 | 2017-10-17 | Bayer Pharma AG | Composés pour le traitement d'un cancer |
PT3283642T (pt) | 2015-04-17 | 2024-01-02 | Crossfire Oncology Holding B V | Biomarcadores de prognóstico para quimioterapia inibidora de ttk |
MX2018011831A (es) | 2016-04-04 | 2019-02-13 | Chemocentryx Inc | Antagonistas solubles de receptor de c5aa(c5ar). |
CA3241111A1 (en) * | 2021-12-15 | 2023-06-22 | Heidi Lane | Methods of treating neoplastic diseases |
Family Cites Families (42)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE69736711T2 (de) | 1996-08-28 | 2007-09-20 | Pfizer Inc. | Substituierte 6,5-heterobicyclische-derivate |
IL133007A (en) | 1997-05-28 | 2005-06-19 | Aventis Pharma Inc | Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases |
US6514989B1 (en) | 2001-07-20 | 2003-02-04 | Hoffmann-La Roche Inc. | Aromatic and heteroaromatic substituted 1,2,4-triazolo pyridine derivatives |
JP2004346016A (ja) | 2003-05-22 | 2004-12-09 | Otsuka Chemical Co Ltd | トリフルオロメチルキノキサリン化合物、その製造方法、及び有害生物防除剤 |
JP4499721B2 (ja) | 2003-06-30 | 2010-07-07 | ヒフ バイオ,インク. | 化合物、組成物および方法 |
EP1799680A2 (en) | 2004-10-07 | 2007-06-27 | Warner-Lambert Company LLC | Triazolopyridine derivatives as antibacterial agents |
US20070049591A1 (en) | 2005-08-25 | 2007-03-01 | Kalypsys, Inc. | Inhibitors of MAPK/Erk Kinase |
US20070078136A1 (en) | 2005-09-22 | 2007-04-05 | Bristol-Myers Squibb Company | Fused heterocyclic compounds useful as kinase modulators |
US7723336B2 (en) | 2005-09-22 | 2010-05-25 | Bristol-Myers Squibb Company | Fused heterocyclic compounds useful as kinase modulators |
WO2007065010A2 (en) | 2005-12-02 | 2007-06-07 | Hif Bio, Inc. | Anti-angiogenesis compounds |
EA200870592A1 (ru) | 2006-05-31 | 2009-08-28 | Галапагос Н.В. | Триазолопиразиновые соединения, пригодные для лечения дегенеративных и воспалительных заболеваний |
US20100075947A1 (en) | 2006-08-16 | 2010-03-25 | Exelixis, Inc. | Methods of Using PI3K and MEK Modulators |
CN103641829A (zh) | 2006-08-30 | 2014-03-19 | 塞尔佐姆有限公司 | 作为激酶抑制剂的三唑衍生物 |
PE20090288A1 (es) | 2007-05-10 | 2009-04-03 | Smithkline Beecham Corp | Derivados de quinoxalina como inhibidores de la pi3 quinasa |
CN101801966A (zh) | 2007-07-18 | 2010-08-11 | 诺瓦提斯公司 | 双环杂芳基化合物和它们作为激酶抑制剂的用途 |
JP2010535804A (ja) | 2007-08-09 | 2010-11-25 | グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー | Pi3キナーゼ阻害薬としてのキノキサリン誘導体 |
MX2010002115A (es) | 2007-08-23 | 2010-06-01 | Aztrazeneca Ab | 2-anilinopurin-8-onas como inhibidores de ttk/mps1 para el tratamiento de trastornos .proliferativos. |
KR20100075881A (ko) | 2007-08-31 | 2010-07-05 | 메르크 세로노 에스. 에이. | 트리아졸로피리딘 화합물 및 ask 저해제로서 이의 용도 |
GB0719803D0 (en) | 2007-10-10 | 2007-11-21 | Cancer Rec Tech Ltd | Therapeutic compounds and their use |
EP2222674B8 (en) | 2007-11-27 | 2016-01-06 | Cellzome Limited | Amino triazoles as pi3k inhibitors |
US8415376B2 (en) | 2008-05-30 | 2013-04-09 | Amgen Inc. | Inhibitors of PI3 kinase |
TWI491610B (zh) | 2008-10-09 | 2015-07-11 | 必治妥美雅史谷比公司 | 作為激酶抑制劑之咪唑并嗒腈 |
WO2010092015A1 (en) | 2009-02-10 | 2010-08-19 | Cellzome Limited | Urea triazololo [1, 5-a] pyridine derivatives as pi3k inhibitors |
EA201101188A1 (ru) | 2009-02-13 | 2012-04-30 | Фовеа Фармасьютикалз | [1,2,4]триазоло[1,5-а]пиридины в качестве ингибиторов киназы |
CN102413831B (zh) | 2009-04-29 | 2014-06-04 | 拜耳知识产权有限责任公司 | 取代的咪唑并喹喔啉 |
TW201107329A (en) | 2009-07-30 | 2011-03-01 | Oncotherapy Science Inc | Fused imidazole derivative having ttk inhibitory action |
CN102596932A (zh) | 2009-09-04 | 2012-07-18 | 拜耳医药股份有限公司 | 作为酪氨酸苏氨酸激酶抑制剂的取代氨基喹喔啉 |
EP2343295A1 (en) * | 2009-11-30 | 2011-07-13 | Bayer Schering Pharma AG | Triazolopyridine derivates |
EP2343294A1 (en) | 2009-11-30 | 2011-07-13 | Bayer Schering Pharma AG | Substituted triazolopyridines |
EP2343297A1 (en) * | 2009-11-30 | 2011-07-13 | Bayer Schering Pharma AG | Triazolopyridines |
EP2523949B1 (en) | 2010-01-15 | 2014-08-20 | Janssen Pharmaceuticals Inc. | Novel substituted triazole derivatives as gamma secretase modulators |
US20110190269A1 (en) | 2010-02-01 | 2011-08-04 | Karlheinz Baumann | Gamma secretase modulators |
UY33452A (es) * | 2010-06-16 | 2012-01-31 | Bayer Schering Pharma Ag | Triazolopiridinas sustituidas |
TWI541243B (zh) | 2010-09-10 | 2016-07-11 | 拜耳知識產權公司 | 經取代咪唑并嗒 |
AU2012244859B2 (en) | 2011-04-21 | 2017-06-08 | Bayer Intellectual Property Gmbh | Triazolopyridines |
UA112096C2 (uk) * | 2011-12-12 | 2016-07-25 | Байєр Інтеллектуал Проперті Гмбх | Заміщені триазолопіридини та їх застосування як інгібіторів ttk |
ES2605946T3 (es) | 2012-03-14 | 2017-03-17 | Bayer Intellectual Property Gmbh | Imidazopiridazinas sustituidas |
EP2872506A1 (en) * | 2012-07-10 | 2015-05-20 | Bayer Pharma Aktiengesellschaft | Method for preparing substituted triazolopyridines |
AR096469A1 (es) * | 2013-06-06 | 2015-12-30 | Bayer Pharma AG | Composiciones farmacéuticas que comprenden compuestos del tipo triazolpiridinas |
CN105431435A (zh) * | 2013-06-07 | 2016-03-23 | 拜耳制药股份公司 | 具有作为mps-1抑制剂的活性的取代的三唑并吡啶类 |
BR112015030774A2 (pt) * | 2013-06-10 | 2017-07-25 | Bayer Pharma AG | novos compostos para o tratamento de câncer |
CA2914742A1 (en) * | 2013-06-11 | 2014-12-18 | Bayer Pharma Aktiengesellschaft | Handovers with co-operating cells configured to provide coordinated multi-point transmission/reception |
-
2014
- 2014-06-06 SG SG11201509858QA patent/SG11201509858QA/en unknown
- 2014-06-06 RS RS20170534A patent/RS56034B1/sr unknown
- 2014-06-06 US US14/897,951 patent/US9586958B2/en not_active Expired - Fee Related
- 2014-06-06 MA MA38654A patent/MA38654B1/fr unknown
- 2014-06-06 WO PCT/EP2014/061779 patent/WO2014198647A2/en active Application Filing
- 2014-06-06 CA CA2914745A patent/CA2914745A1/en not_active Abandoned
- 2014-06-06 DK DK14728949.0T patent/DK3008062T3/en active
- 2014-06-06 EA EA201600002A patent/EA201600002A1/ru unknown
- 2014-06-06 PL PL14728949T patent/PL3008062T3/pl unknown
- 2014-06-06 CN CN201480040729.XA patent/CN105377848A/zh active Pending
- 2014-06-06 HU HUE14728949A patent/HUE033131T2/en unknown
- 2014-06-06 AU AU2014280356A patent/AU2014280356A1/en not_active Abandoned
- 2014-06-06 AP AP2015008898A patent/AP2015008898A0/xx unknown
- 2014-06-06 LT LTEP14728949.0T patent/LT3008062T/lt unknown
- 2014-06-06 JP JP2016518941A patent/JP2016526534A/ja active Pending
- 2014-06-06 KR KR1020167000270A patent/KR20160019492A/ko not_active Application Discontinuation
- 2014-06-06 TN TN2015000545A patent/TN2015000545A1/en unknown
- 2014-06-06 EP EP14728949.0A patent/EP3008062B1/en active Active
- 2014-06-06 PT PT147289490T patent/PT3008062T/pt unknown
- 2014-06-06 PE PE2015002605A patent/PE20160156A1/es not_active Application Discontinuation
- 2014-06-06 SI SI201430219A patent/SI3008062T1/sl unknown
- 2014-06-06 MX MX2015017119A patent/MX2015017119A/es unknown
- 2014-06-06 ES ES14728949.0T patent/ES2626790T3/es active Active
- 2014-06-11 AR ARP140102239A patent/AR096585A1/es unknown
- 2014-06-11 UY UY0001035610A patent/UY35610A/es not_active Application Discontinuation
-
2015
- 2015-11-30 IL IL242847A patent/IL242847A0/en unknown
- 2015-12-03 ZA ZA2015/08868A patent/ZA201508868B/en unknown
- 2015-12-09 PH PH12015502746A patent/PH12015502746A1/en unknown
- 2015-12-11 CR CR20150659A patent/CR20150659A/es unknown
- 2015-12-11 NI NI201500176A patent/NI201500176A/es unknown
- 2015-12-11 CU CUP2015000176A patent/CU20150176A7/es unknown
- 2015-12-11 DO DO2015000299A patent/DOP2015000299A/es unknown
- 2015-12-11 CL CL2015003605A patent/CL2015003605A1/es unknown
-
2016
- 2016-08-29 HK HK16110219.6A patent/HK1221955A1/zh unknown
-
2017
- 2017-05-12 HR HRP20170717TT patent/HRP20170717T1/hr unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
SV2018005610A (es) | Derivados de oxopiridina sustituidos | |
CL2016002735A1 (es) | Compuestos de imidazo[4,5-c]quinolin-2-ona y su uso para tratar cáncer | |
CL2016002027A1 (es) | Ciclopropilamina como inhibidor de la lsd1 | |
CL2015001985A1 (es) | Compuestos de tiazolcarboxamidas y piridinacarboxamida, inhibidores de quinasa pim. | |
DOP2015000274A (es) | Compuestos químicos | |
CL2015003686A1 (es) | Derivados de pirrolo[3,2-d]pirimidina para el tratamiento de infecciones víricas y otras enfermedades | |
CL2016000153A1 (es) | Derivados de pirrolamida sustituidos con glioxamida y su uso como medicamentos para el tratamiento de la hepatitis b | |
CR20150472A (es) | USO DE DERIVADOS DE PIRAZOLOPIRIMIDINA PARA EL TRATAMIENTO DE TRANSTORNOS RELACIONADOS CON LA PI3Kd | |
CL2015002335A1 (es) | Derivados de 2-aminopirimidina para el tratamiento de infecciones víricas. | |
CL2018003444A1 (es) | Derivados de adenosina para uso en el tratamiento del cancer. | |
CL2016001895A1 (es) | Compuestos | |
CL2014001793A1 (es) | Compuestos derivados de 1,3,5-triazinas sustituidas y sus sales, como inhibidores de la idh2 mutante; composicion farmaceutica que los comprende; y su uso para el tratamiento del cancer. | |
CL2016003214A1 (es) | Derivados de la indolizina como inhibidores de las fosfoinositido-3 quinasas | |
CL2016001151A1 (es) | Derivados de purina 2,6-sustituidos y su uso en el tratamiento de trastorno proliferativos. | |
NI201500115A (es) | Estra-1,3,5(10), 16-tetraeno-3-carboxamidas para la inhibición de la 17b-hidroxiesteroide deshidrogenasa (akr1 c3) | |
CL2016003074A1 (es) | Compuestos derivados de 2-oxi-2-fenil-n-5-pirrolidin-3-ilamino-1,3,4-tiadiazol-2-ilacetamida, inhibidores gls1 composición farmacéutica y su uso para tratar el cáncer. | |
NI201500175A (es) | Compuestos nuevos para el tratamiento del cáncer | |
CL2016002151A1 (es) | Derivados de piridazina para uso en la prevención o el tratamiento de un trastorno atáxico | |
DOP2016000297A (es) | Composiciones farmacéuticas útiles para tratar enfermedades infecciosas | |
CU20150176A7 (es) | Derivados de prodroga de triazolpiridinas sustituídas | |
CR20160494A (es) | Compuestos heteroaromáticos y su uso como ligandos de dopamina d1 | |
CL2015003460A1 (es) | Composiciones oftálmicas acuosas tópicas que contienen un derivado de 1h-indol-1-carboxamida y uso de estas para el tratamiento de una enfermedad oftálmica | |
CL2016001054A1 (es) | Compuestos para el tratamiento de diabetes y complicaciones de enfermedades derivadas de la misma | |
NI201700072A (es) | Compuestos para tratar el cáncer. | |
DOP2015000290A (es) | Benzoxazoles sustituidos |