CS382091A3 - 1-(2-aryl-2-halogen-1-ethenyl)-1h-azoles, process of their preparation and pharmaceuticals based thereon - Google Patents

1-(2-aryl-2-halogen-1-ethenyl)-1h-azoles, process of their preparation and pharmaceuticals based thereon Download PDF

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Publication number
CS382091A3
CS382091A3 CS913820A CS382091A CS382091A3 CS 382091 A3 CS382091 A3 CS 382091A3 CS 913820 A CS913820 A CS 913820A CS 382091 A CS382091 A CS 382091A CS 382091 A3 CS382091 A3 CS 382091A3
Authority
CS
Czechoslovakia
Prior art keywords
substituted
phenyl
lower alkyl
halogen
aryl
Prior art date
Application number
CS913820A
Other languages
Czech (cs)
English (en)
Inventor
Jan Heeres
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of CS382091A3 publication Critical patent/CS382091A3/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CS913820A 1983-11-07 1991-12-16 1-(2-aryl-2-halogen-1-ethenyl)-1h-azoles, process of their preparation and pharmaceuticals based thereon CS382091A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US54912783A 1983-11-07 1983-11-07
US06/630,158 US4539325A (en) 1983-11-07 1984-07-12 1-(2-Aryl-2-halo-1-ethenyl)-1H-azoles, and anticonvulsant use thereof

Publications (1)

Publication Number Publication Date
CS382091A3 true CS382091A3 (en) 1992-04-15

Family

ID=27069019

Family Applications (1)

Application Number Title Priority Date Filing Date
CS913820A CS382091A3 (en) 1983-11-07 1991-12-16 1-(2-aryl-2-halogen-1-ethenyl)-1h-azoles, process of their preparation and pharmaceuticals based thereon

Country Status (17)

Country Link
US (1) US4539325A (da)
EP (1) EP0142190B1 (da)
JP (1) JPH0613480B2 (da)
AU (1) AU566022B2 (da)
CA (1) CA1241657A (da)
CS (1) CS382091A3 (da)
CY (1) CY1606A (da)
DE (1) DE3478743D1 (da)
DK (1) DK162984C (da)
FI (1) FI85854C (da)
HK (1) HK52591A (da)
IE (1) IE57826B1 (da)
IL (1) IL73425A (da)
NO (1) NO161800C (da)
NZ (1) NZ210014A (da)
SG (1) SG46991G (da)
SU (1) SU1322978A3 (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3470881D1 (de) * 1983-12-20 1988-06-09 Ciba Geigy Ag Microbizides
JPS62149666A (ja) * 1985-12-25 1987-07-03 Shionogi & Co Ltd Ｎ−ビニルアゾ−ル類
JP2792694B2 (ja) * 1989-12-12 1998-09-03 エスケ−化研株式会社 塗布装置
US5196446A (en) * 1990-04-16 1993-03-23 Yissum Research Development Company Of The Hebrew University Of Jerusalem Certain indole compounds which inhibit EGF receptor tyrosine kinase
US5418245A (en) * 1990-04-16 1995-05-23 Rhone-Poulenc Rorer International (Holdings) Inc. Styryl-substituted monocyclic and bicyclic heteroaryl compounds which inhibit EGF receptor tyrosine kinase
US5302606A (en) * 1990-04-16 1994-04-12 Rhone-Poulenc Rorer Pharmaceuticals Inc. Styryl-substituted pyridyl compounds which inhibit EGF receptor tyrosine kinase
AU2002221222A1 (en) * 2000-12-04 2002-06-18 Biovitrum Ab Novel method and use
SE0004462D0 (sv) 2000-12-04 2000-12-04 Pharmacia Ab Novel method and use
RU2632682C1 (ru) * 2016-09-30 2017-10-09 Федеральное государственное автономное образовательное учреждение высшего образования Первый Московский государственный медицинский университет им. И.М. Сеченова Министерства здравоохранения Российской Федерации (Сеченовский университет) Комплекс ацетата цинка с 1-пропаргилимидазолом, обладающий антигипоксической активностью

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3679697A (en) * 1970-10-08 1972-07-25 Searle & Co 1-({62 -halophenethyl)imidazoles
GB1533705A (en) * 1975-03-10 1978-11-29 Ici Ltd Method of combating fungal infections in plants using imidazoles and 1,2,4-triazoles
DE2839388A1 (de) * 1978-09-11 1980-03-27 Siegfried Ag Imidazolylvinylaether und deren verwendung
NL8005204A (nl) * 1980-09-17 1982-04-16 Gist Brocades Nv Ethenyl-imidazool-derivaten met antimycotische werkzaamheid.
GR78234B (da) * 1981-03-10 1984-09-26 Ciba Geigy Ag
CA1189857A (en) * 1981-03-27 1985-07-02 Janssen Pharmaceutica Naamloze Vennootschap Antimicrobial triazole derivatives
CA1206970A (en) * 1981-10-01 1986-07-02 Hak-Foon Chan Substituted ethylenic imidazoles and triazoles

Also Published As

Publication number Publication date
SG46991G (en) 1991-07-26
IL73425A (en) 1987-09-16
DE3478743D1 (de) 1989-07-27
FI844349L (fi) 1985-05-08
NZ210014A (en) 1987-03-06
DK528284D0 (da) 1984-11-06
SU1322978A3 (ru) 1987-07-07
FI85854B (fi) 1992-02-28
NO844420L (no) 1985-05-08
IE842852L (en) 1985-05-07
JPH0613480B2 (ja) 1994-02-23
DK162984B (da) 1992-01-06
EP0142190A3 (en) 1986-12-03
DK162984C (da) 1992-06-01
FI844349A0 (fi) 1984-11-06
DK528284A (da) 1985-05-08
IL73425A0 (en) 1985-02-28
CA1241657A (en) 1988-09-06
US4539325A (en) 1985-09-03
HK52591A (en) 1991-07-19
NO161800B (no) 1989-06-19
CY1606A (en) 1992-04-03
AU566022B2 (en) 1987-10-08
EP0142190A2 (en) 1985-05-22
NO161800C (no) 1989-09-27
EP0142190B1 (en) 1989-06-21
IE57826B1 (en) 1993-04-21
FI85854C (fi) 1992-06-10
JPS60166666A (ja) 1985-08-29
AU3513784A (en) 1985-05-16

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Legal Events

Date Code Title Description
PD00 Pending as of 2000-06-30 in czech republic