CS244405B2 - 3-aminovinyl cephalosporines' new derivatives production method - Google Patents

3-aminovinyl cephalosporines' new derivatives production method Download PDF

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Publication number
CS244405B2
CS244405B2 CS803543A CS354380A CS244405B2 CS 244405 B2 CS244405 B2 CS 244405B2 CS 803543 A CS803543 A CS 803543A CS 354380 A CS354380 A CS 354380A CS 244405 B2 CS244405 B2 CS 244405B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
mixture
radical
group
solution
Prior art date
Application number
CS803543A
Other languages
Czech (cs)
English (en)
Other versions
CS354380A2 (it
Inventor
Daniel Farge
Roy Pierre Le
Claude Moutonnier
Jean-Francois Peyronel
Original Assignee
Rhone Poulenc Ind
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Ind filed Critical Rhone Poulenc Ind
Publication of CS354380A2 publication Critical patent/CS354380A2/cs
Publication of CS244405B2 publication Critical patent/CS244405B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/02—Nutrients, e.g. vitamins, minerals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
CS803543A 1979-05-23 1980-05-21 3-aminovinyl cephalosporines' new derivatives production method CS244405B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7913096A FR2457296A1 (fr) 1979-05-23 1979-05-23 Nouveaux derives de vinyl-3 cephalosporines et leur preparation

Publications (2)

Publication Number Publication Date
CS354380A2 CS354380A2 (it) 1985-09-17
CS244405B2 true CS244405B2 (en) 1986-07-17

Family

ID=9225762

Family Applications (1)

Application Number Title Priority Date Filing Date
CS803543A CS244405B2 (en) 1979-05-23 1980-05-21 3-aminovinyl cephalosporines' new derivatives production method

Country Status (31)

Country Link
US (1) US4307233A (it)
JP (1) JPS55154981A (it)
AT (1) AT369375B (it)
AU (1) AU534806B2 (it)
BE (1) BE883416A (it)
CA (1) CA1144919A (it)
CH (1) CH645379A5 (it)
CS (1) CS244405B2 (it)
DD (1) DD150899A5 (it)
DE (1) DE3019462A1 (it)
DK (1) DK222080A (it)
ES (1) ES491687A0 (it)
FI (1) FI801641A (it)
FR (1) FR2457296A1 (it)
GB (1) GB2051062B (it)
GR (1) GR68426B (it)
HU (1) HU185890B (it)
IE (1) IE49814B1 (it)
IL (1) IL60139A (it)
IT (1) IT1140974B (it)
LU (1) LU82477A1 (it)
NL (1) NL8003023A (it)
NO (1) NO801502L (it)
NZ (1) NZ193799A (it)
PH (1) PH15946A (it)
PL (1) PL126481B1 (it)
PT (1) PT71276A (it)
SE (1) SE451072B (it)
SU (1) SU1031409A3 (it)
YU (1) YU136880A (it)
ZA (1) ZA803038B (it)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI793566A (fi) * 1978-11-15 1980-05-16 Glaxo Group Ltd Kefalosporinantibioter
FR2494279A1 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouvelles oxacephalosporines, leur preparation et les medicaments qui les contiennent
FR2494275A2 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouveaux derives de vinyl-3 cephalosporines et leur preparation
FR2494280A1 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouveaux derives de la cephalosporine et leur preparation
FR2505334A1 (fr) * 1981-05-11 1982-11-12 Rhone Poulenc Sante Nouvelles oxacephalosporines et leur preparation
FR2511372A1 (fr) * 1981-08-17 1983-02-18 Rhone Poulenc Sante Nouveaux derives de la cephalosporine et leur preparation
US4486586A (en) * 1983-02-10 1984-12-04 Bristol-Myers Company Cephalosporin derivatives
US4560749A (en) * 1983-11-18 1985-12-24 Eli Lilly And Company Cephem-3-imidates and 3-amidines
US4708955A (en) * 1985-06-24 1987-11-24 Bristol-Myers Company 3-(substituted)propenyl-7-aminothiazol-ylcephalosporanic acids and esters thereof
US4874856A (en) * 1985-06-24 1989-10-17 Bristol-Myers Company 3-(substituted)propenyl-7-(aminothiazolylacetamido) ceph-3-em-4-carboxylic acids and esters thereof
DE3787030T2 (de) * 1986-04-14 1994-04-07 Banyu Pharma Co Ltd 1-carboxy-1-vinyloxyiminoaminothiazol-cephalosporin-derivate und deren herstellung.
ATE354577T1 (de) 1996-11-06 2007-03-15 Basilea Pharmaceutica Ag Vinylpyrrolidinon-cephalosporin-derivate
CA2702257C (en) * 2007-10-09 2016-07-12 Sopharmia, Inc. Broad spectrum beta-lactamase inhibitors
DK2968352T3 (da) 2013-03-12 2019-01-02 Gladius Pharmaceuticals Corp Derivatiserede 3-styryl-cephalosporiner

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4065620A (en) * 1971-06-14 1977-12-27 Eli Lilly And Company 3-(Substituted) vinyl cephalosporins
GB1463077A (en) * 1973-04-19 1977-02-02 Glaxo Lab Ltd 7-substituted-ethyl-cephalosporin derivatives
HU172234B (hu) * 1973-12-21 1978-07-28 Glaxo Lab Ltd Sposob poluchenija novykh proizvodnykh 7-beta-acilamido-cef-3-em-4-karbonovojj kisloty
US4144393A (en) * 1973-12-21 1979-03-13 Glaxo Laboratories Limited 3-Acetoxymethyl cephalosporins having at position-7 a carboxy substituted α-etherified hydroxyiminoarylacetamido group
JPS5129492A (en) * 1974-09-04 1976-03-12 Sankyo Co Sefuarosuhorinjudotai no seiho
DK154939C (da) * 1974-12-19 1989-06-12 Takeda Chemical Industries Ltd Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
JPS5253890A (en) * 1975-10-14 1977-04-30 Syntex Inc Production of cephalosporin type compound
PT71651B (en) * 1979-08-15 1982-01-21 Merck & Co Inc Process for preparing allysulfoxide enzyme inhibitors

Also Published As

Publication number Publication date
DK222080A (da) 1980-11-24
NL8003023A (nl) 1980-11-25
ZA803038B (en) 1981-05-27
AU5859580A (en) 1980-11-27
IL60139A0 (en) 1980-07-31
GB2051062A (en) 1981-01-14
SE8003821L (sv) 1980-11-24
ES8102136A1 (es) 1980-12-16
PL224391A1 (it) 1981-02-13
LU82477A1 (fr) 1980-12-16
AT369375B (de) 1982-12-27
PT71276A (fr) 1980-06-01
FI801641A (fi) 1980-11-24
GB2051062B (en) 1983-10-12
IE801062L (en) 1980-11-23
ATA270980A (de) 1982-05-15
FR2457296A1 (fr) 1980-12-19
CA1144919A (fr) 1983-04-19
YU136880A (en) 1983-04-30
CH645379A5 (fr) 1984-09-28
NO801502L (no) 1980-11-24
PL126481B1 (en) 1983-08-31
PH15946A (en) 1983-04-29
IT1140974B (it) 1986-10-10
FR2457296B1 (it) 1982-02-05
US4307233A (en) 1981-12-22
SU1031409A3 (ru) 1983-07-23
IL60139A (en) 1984-04-30
AU534806B2 (en) 1984-02-16
BE883416A (fr) 1980-11-21
GR68426B (it) 1981-12-30
SE451072B (sv) 1987-08-31
DD150899A5 (de) 1981-09-23
IT8022243A0 (it) 1980-05-21
HU185890B (en) 1985-04-28
DE3019462A1 (de) 1980-12-04
IE49814B1 (en) 1985-12-25
CS354380A2 (it) 1985-09-17
NZ193799A (en) 1983-03-15
ES491687A0 (es) 1980-12-16
JPS55154981A (en) 1980-12-02
JPH0246595B2 (it) 1990-10-16

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