CS226449B2 - Method of preparing new imidazo(1,2-a)-pyrimidines - Google Patents

Method of preparing new imidazo(1,2-a)-pyrimidines Download PDF

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Publication number
CS226449B2
CS226449B2 CS824664A CS466482A CS226449B2 CS 226449 B2 CS226449 B2 CS 226449B2 CS 824664 A CS824664 A CS 824664A CS 466482 A CS466482 A CS 466482A CS 226449 B2 CS226449 B2 CS 226449B2
Authority
CS
Czechoslovakia
Prior art keywords
acid
formula
pyrimidines
compounds
imidazo
Prior art date
Application number
CS824664A
Other languages
Czech (cs)
English (en)
Inventor
Helmut Dr Ataehle
Herbert Dr Koeppe
Werner Dr Kummer
Klaus Dr Stockhaus
Wolfram Dr Gaida
Wolfgang Dr Hoefke
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Publication of CS226449B2 publication Critical patent/CS226449B2/cs

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CS824664A 1981-06-24 1982-06-23 Method of preparing new imidazo(1,2-a)-pyrimidines CS226449B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19813124718 DE3124718A1 (de) 1981-06-24 1981-06-24 Neue imidazo (1,2-a)pyramidine, deren saeureadditionssalze, diese enthaltende arzneimittel und verfahren zu deren herstellung

Publications (1)

Publication Number Publication Date
CS226449B2 true CS226449B2 (en) 1984-03-19

Family

ID=6135235

Family Applications (1)

Application Number Title Priority Date Filing Date
CS824664A CS226449B2 (en) 1981-06-24 1982-06-23 Method of preparing new imidazo(1,2-a)-pyrimidines

Country Status (18)

Country Link
US (1) US4438118A (el)
EP (1) EP0068302A1 (el)
JP (1) JPS584784A (el)
KR (1) KR840000551A (el)
AU (1) AU8531482A (el)
CS (1) CS226449B2 (el)
DE (1) DE3124718A1 (el)
DK (1) DK281882A (el)
ES (2) ES513377A0 (el)
FI (1) FI822236L (el)
GR (1) GR76833B (el)
HU (1) HU185108B (el)
IL (1) IL66111A0 (el)
NO (1) NO822076L (el)
PL (1) PL237052A1 (el)
PT (1) PT75107B (el)
YU (1) YU135182A (el)
ZA (1) ZA824437B (el)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4636502A (en) * 1982-12-27 1987-01-13 Eli Lilly And Company Methods of producing a positive inotropic effect or vasodilation by administration of 2-phenyl imidazo pyrimidines and pyrazines
JPS60193990A (ja) * 1984-03-12 1985-10-02 Yoshitomi Pharmaceut Ind Ltd 新規なポリアザ複素環誘導体
JPS6152118A (ja) * 1984-08-21 1986-03-14 三菱電機株式会社 電源装置
US5252563A (en) * 1991-12-19 1993-10-12 G. D. Searle & Company 5,6,7,8-tetrahydro-imidazo[1,2-a]pyrimidine compounds for treatment of neurotoxic injury
JP4209165B2 (ja) 2002-09-30 2009-01-14 本田技研工業株式会社 車両用情報表示装置
WO2008060817A2 (en) * 2006-10-19 2008-05-22 Blaise Harrison Llc Exothermic personal lubricant

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2118261A1 (de) 1971-04-15 1972-11-02 C.H. Boehringer Sohn, 6507 Ingelheim Neue N-haltige Bicyclen, deren Säureadditionssalze sowie Verfahren zu deren Herstellung
BE786028A (fr) 1971-07-08 1973-01-08 Boehringer Sohn Ingelheim 2,3-dihydro-oxo-imidazo(1,2-a)-pyrimidines, leurs sels d'addition avec des acides et procedes pour les fabriquer
DE2523103C3 (de) 1975-05-24 1979-11-29 C.H. Boehringer Sohn, 6507 Ingelheim Substituierte 2-[N-Progargyl-N-(2-chlorphenyl)amino] -imidazoline-^), deren Säureadditionssalze, Verfahren zu ihrer Herstellung und deren Verwendung

Also Published As

Publication number Publication date
FI822236L (fi) 1982-12-25
JPS584784A (ja) 1983-01-11
GR76833B (el) 1984-09-04
ES518499A0 (es) 1983-10-01
FI822236A0 (fi) 1982-06-22
DE3124718A1 (de) 1983-01-13
YU135182A (en) 1986-04-30
ZA824437B (en) 1984-02-29
NO822076L (no) 1982-12-27
US4438118A (en) 1984-03-20
ES8307811A1 (es) 1983-07-01
EP0068302A1 (de) 1983-01-05
HU185108B (en) 1984-12-28
PL237052A1 (en) 1983-06-20
IL66111A0 (en) 1982-09-30
KR840000551A (ko) 1984-02-25
AU8531482A (en) 1983-01-06
PT75107B (de) 1985-05-31
DK281882A (da) 1982-12-25
ES8308884A1 (es) 1983-10-01
ES513377A0 (es) 1983-07-01
PT75107A (de) 1982-07-01

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