CS221802B2 - Method of preparation of the 4-deoxy-4-aminoerythromycine a - Google Patents

Method of preparation of the 4-deoxy-4-aminoerythromycine a Download PDF

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Publication number
CS221802B2
CS221802B2 CS814590A CS459081A CS221802B2 CS 221802 B2 CS221802 B2 CS 221802B2 CS 814590 A CS814590 A CS 814590A CS 459081 A CS459081 A CS 459081A CS 221802 B2 CS221802 B2 CS 221802B2
Authority
CS
Czechoslovakia
Prior art keywords
hydrogen
deoxy
product
water
compounds
Prior art date
Application number
CS814590A
Other languages
Czech (cs)
English (en)
Inventor
Frank Ch Sciavolino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CS221802B2 publication Critical patent/CS221802B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CS814590A 1977-02-04 1978-02-02 Method of preparation of the 4-deoxy-4-aminoerythromycine a CS221802B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US76548077A 1977-02-04 1977-02-04

Publications (1)

Publication Number Publication Date
CS221802B2 true CS221802B2 (en) 1983-04-29

Family

ID=25073668

Family Applications (2)

Application Number Title Priority Date Filing Date
CS814591A CS221803B2 (en) 1977-02-04 1978-02-02 Method of preparation of the derivative of the 4-deoxy-4-oxoerythromycine a
CS814590A CS221802B2 (en) 1977-02-04 1978-02-02 Method of preparation of the 4-deoxy-4-aminoerythromycine a

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CS814591A CS221803B2 (en) 1977-02-04 1978-02-02 Method of preparation of the derivative of the 4-deoxy-4-oxoerythromycine a

Country Status (10)

Country Link
US (1) US4150220A (hu)
JP (3) JPS597718B2 (hu)
AT (1) AT359643B (hu)
BE (1) BE863621A (hu)
CS (2) CS221803B2 (hu)
DD (1) DD143779A5 (hu)
HU (1) HU184999B (hu)
PL (1) PL115793B1 (hu)
SU (3) SU837326A3 (hu)
ZA (1) ZA78676B (hu)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4283527A (en) * 1980-04-01 1981-08-11 Pfizer Inc. Erythromycylamine 11,12-carbonate and derivatives thereof
US4413119A (en) * 1982-03-01 1983-11-01 Pfizer Inc. Semi-synthetic macrolides
US4382085A (en) * 1982-03-01 1983-05-03 Pfizer Inc. 4"-Epi erythromycin A and derivatives thereof as useful antibacterial agents
US4363803A (en) * 1982-03-01 1982-12-14 Pfizer Inc. 3",4"-Oxyallylene erythromycin and oleandomycin, composition and method of use
US4382086A (en) * 1982-03-01 1983-05-03 Pfizer Inc. 9-Dihydro-11,12-ketal derivatives of erythromycin A and epi-erythromycin A
DK149776C (da) * 1984-01-06 1987-04-21 Orion Yhtymae Oy Antibiotisk virksom erytromycinforbindelse og praeparat indeholdende forbindelsen
US4512982A (en) * 1984-04-13 1985-04-23 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical composition and therapeutic method
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
ES552858A1 (es) 1985-03-12 1987-11-01 Beecham Group Plc Un procedimiento para la preparacion de derivados de eritromicina.
US5175150A (en) * 1985-08-31 1992-12-29 Kitasato, Kenkyusho Erythromycin derivative
US4672056A (en) * 1985-11-12 1987-06-09 Abbott Laboratories Erythromycin A derivatives and method of use
FR2639945B1 (fr) * 1988-12-07 1994-03-25 Oreal Ethers et/ou esters lipophiles de d-desosamine, leur procede de preparation et leur utilisation en tant qu'agents antibacteriens et antifongiques
US5808017A (en) * 1996-04-10 1998-09-15 Abbott Laboratories Process for preparing erythromycin A oxime
HN1998000074A (es) * 1997-06-11 1999-01-08 Pfizer Prod Inc Derivados de macrolidos c-4 sustituidos

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3842069A (en) * 1973-06-21 1974-10-15 Abbott Lab 4"-deoxy-4"-oxoerythromycin b derivatives
US3884903A (en) * 1973-06-21 1975-05-20 Abbott Lab 4{41 -Deoxy-4{41 -oxoerythromycin B derivatives

Also Published As

Publication number Publication date
ZA78676B (en) 1978-12-27
JPS57154198A (en) 1982-09-22
SU886749A3 (ru) 1981-11-30
ATA75378A (de) 1980-04-15
AT359643B (de) 1980-11-25
SU1172451A3 (ru) 1985-08-07
CS221803B2 (en) 1983-04-29
US4150220A (en) 1979-04-17
DD143779A5 (de) 1980-09-10
PL115793B1 (en) 1981-04-30
JPS597718B2 (ja) 1984-02-20
SU837326A3 (ru) 1981-06-07
JPS5853000B2 (ja) 1983-11-26
JPS57154199A (en) 1982-09-22
HU184999B (en) 1984-11-28
JPS57158799A (en) 1982-09-30
BE863621A (fr) 1978-08-03
JPS5827800B2 (ja) 1983-06-11

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