CS217997B2 - Method of making the new derivatives of the pyrimidine - Google Patents
Method of making the new derivatives of the pyrimidine Download PDFInfo
- Publication number
- CS217997B2 CS217997B2 CS813920A CS392081A CS217997B2 CS 217997 B2 CS217997 B2 CS 217997B2 CS 813920 A CS813920 A CS 813920A CS 392081 A CS392081 A CS 392081A CS 217997 B2 CS217997 B2 CS 217997B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- pyrimidine
- formula
- compounds
- methyl ester
- acetic acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Pulmonology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Immunology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH499580 | 1980-06-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CS217997B2 true CS217997B2 (en) | 1983-02-25 |
Family
ID=4286126
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS813920A CS217997B2 (en) | 1980-06-27 | 1981-05-27 | Method of making the new derivatives of the pyrimidine |
Country Status (25)
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1142924A (en) * | 1980-06-27 | 1983-03-15 | Hoffmann-La Roche Limited | Pyrimidine derivatives |
| US4797486A (en) * | 1986-09-08 | 1989-01-10 | Pfizer Inc. | Heterocyclic ring fused pyrimidine-4(3H)-ones as anticoccidial agents |
| US4725599A (en) * | 1986-09-08 | 1988-02-16 | Pfizer Inc. | Heterocyclic ring fused pyrimidine-4 (3H)-ones as anticoccidial agents |
| DK522187D0 (da) * | 1987-10-06 | 1987-10-06 | Ferrosan As | Imidozothienopyrimidiner, deres fremstilling og anvendelse |
| ATE216999T1 (de) * | 1996-03-11 | 2002-05-15 | Syngenta Participations Ag | Pyrimidin-4-on derivate als pestizidesmittel |
| FR2872165B1 (fr) * | 2004-06-24 | 2006-09-22 | Sod Conseils Rech Applic | Nouveaux derives de pyrimido-benzimidazole |
| US8809346B2 (en) * | 2008-05-30 | 2014-08-19 | Universite De Versailles-Saint-Quentin-En-Yvelines | ANT-ligands molecules and biological applications |
| CN104478851A (zh) * | 2014-12-31 | 2015-04-01 | 济南诚汇双达化工有限公司 | 一种盐酸阿替卡因的制备方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE755404A (fr) * | 1969-08-29 | 1971-03-01 | Sandoz Sa | Nouveau derives de la thiazolo-(3,2-a) pyrrolo (2,3-d) pyrimidine, leurpreparation et medicaments contenant ces derives |
| US3932407A (en) * | 1973-11-19 | 1976-01-13 | Bristol-Myers Company | Optionally substituted 1,2,3,5-tetrahydroimidezo(2,1-b)-quinazolin-2-ones and 6(H)-1,2,3,4-tetrahydropyimido(2,1-b)quinazolin-2-ones |
| DE2411273A1 (de) * | 1974-03-06 | 1975-09-18 | Schering Ag | Neue thieno eckige klammer auf 2,3-d eckige klammer zu pyrimidinone und verfahren zu ihrer herstellung |
| DE2411274A1 (de) * | 1974-03-06 | 1975-09-18 | Schering Ag | Neue 2-nitrothieno eckige klammer auf 2,3-d eckige klammer zu pyrimidinon-derivate und verfahren zu ihrer herstellung |
| US4054656A (en) * | 1975-09-10 | 1977-10-18 | Mead Johnson & Company | Thieno[2,3-d]pyrimidine antiallergic agents |
| JPS5527105A (en) * | 1978-08-11 | 1980-02-27 | Dai Ichi Seiyaku Co Ltd | Imidazothienopyrimidinones compound |
| US4230707A (en) * | 1979-08-27 | 1980-10-28 | Warner-Lambert Company | Oxo-pyrido[1,2-a]thienopyrimidine compounds and methods for their production |
| CA1142924A (en) * | 1980-06-27 | 1983-03-15 | Hoffmann-La Roche Limited | Pyrimidine derivatives |
-
1981
- 1981-05-14 CA CA000377588A patent/CA1142924A/en not_active Expired
- 1981-05-14 ZW ZW117/81A patent/ZW11781A1/xx unknown
- 1981-05-25 FI FI811600A patent/FI811600A7/fi not_active Application Discontinuation
- 1981-05-27 CS CS813920A patent/CS217997B2/cs unknown
- 1981-06-10 DK DK252981A patent/DK252981A/da not_active Application Discontinuation
- 1981-06-19 NZ NZ197476A patent/NZ197476A/en unknown
- 1981-06-19 ZA ZA814162A patent/ZA814162B/xx unknown
- 1981-06-19 US US06/275,271 patent/US4376121A/en not_active Expired - Fee Related
- 1981-06-19 AU AU71967/81A patent/AU7196781A/en not_active Abandoned
- 1981-06-22 DE DE8181104750T patent/DE3166449D1/de not_active Expired
- 1981-06-22 CU CU8135489A patent/CU35489A/es unknown
- 1981-06-22 IL IL63145A patent/IL63145A/xx unknown
- 1981-06-22 AT AT81104750T patent/ATE9698T1/de active
- 1981-06-22 EP EP81104750A patent/EP0043054B1/de not_active Expired
- 1981-06-24 BR BR8103967A patent/BR8103967A/pt unknown
- 1981-06-24 HU HU811851A patent/HU181608B/hu unknown
- 1981-06-24 JP JP56096812A patent/JPS5762282A/ja active Pending
- 1981-06-25 MC MC811524A patent/MC1395A1/xx unknown
- 1981-06-25 GR GR65340A patent/GR74943B/el unknown
- 1981-06-25 PH PH25819A patent/PH16060A/en unknown
- 1981-06-26 ES ES503407A patent/ES503407A0/es active Granted
- 1981-06-26 NO NO812208A patent/NO812208L/no unknown
- 1981-06-26 AR AR285881A patent/AR230748A1/es active
- 1981-06-26 KR KR1019810002316A patent/KR840000705B1/ko not_active Expired
- 1981-06-26 PT PT73270A patent/PT73270B/pt unknown
-
1982
- 1982-12-23 US US06/452,677 patent/US4442289A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| PH16060A (en) | 1983-06-09 |
| ZW11781A1 (en) | 1982-01-20 |
| HU181608B (en) | 1983-10-28 |
| ES8207541A1 (es) | 1982-10-01 |
| ZA814162B (en) | 1982-07-28 |
| DE3166449D1 (en) | 1984-11-08 |
| ES503407A0 (es) | 1982-10-01 |
| JPS5762282A (en) | 1982-04-15 |
| NO812208L (no) | 1981-12-28 |
| ATE9698T1 (de) | 1984-10-15 |
| FI811600L (fi) | 1981-12-28 |
| EP0043054A3 (en) | 1982-03-17 |
| IL63145A0 (en) | 1981-09-13 |
| AR230748A1 (es) | 1984-06-29 |
| CA1142924A (en) | 1983-03-15 |
| BR8103967A (pt) | 1982-03-09 |
| GR74943B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1984-07-12 |
| KR840000705B1 (ko) | 1984-05-21 |
| MC1395A1 (fr) | 1982-04-27 |
| EP0043054B1 (de) | 1984-10-03 |
| IL63145A (en) | 1984-05-31 |
| CU35489A (en) | 1982-12-22 |
| AU7196781A (en) | 1982-01-07 |
| PT73270A (en) | 1981-07-01 |
| NZ197476A (en) | 1984-05-31 |
| EP0043054A2 (de) | 1982-01-06 |
| KR830006302A (ko) | 1983-09-20 |
| DK252981A (da) | 1981-12-28 |
| PT73270B (en) | 1983-05-11 |
| US4376121A (en) | 1983-03-08 |
| US4442289A (en) | 1984-04-10 |
| FI811600A7 (fi) | 1981-12-28 |
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