ES8207541A1 - Procedimiento para la preparacion de derivados de pirimidina - Google Patents
Procedimiento para la preparacion de derivados de pirimidinaInfo
- Publication number
- ES8207541A1 ES8207541A1 ES503407A ES503407A ES8207541A1 ES 8207541 A1 ES8207541 A1 ES 8207541A1 ES 503407 A ES503407 A ES 503407A ES 503407 A ES503407 A ES 503407A ES 8207541 A1 ES8207541 A1 ES 8207541A1
- Authority
- ES
- Spain
- Prior art keywords
- pyrimidine derivatives
- preparation
- medicaments containing
- hydrogen
- antiallergically
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pulmonology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Immunology (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DE PIRIMIDINA. CONSISTE EN HACER REACCIONAR DE FORMULA GENERAL (I) CON AMONIACO O CON UNA SOLUCION DE AMONIACO EN AGUA O EN ALCHOL (TAL COMO EL METANO) A UNA TEMPERATURA DE 0 A 150 GRADOS CENTIGRADOS-PREFERENTEMENTE PROXIMA A 120 GRADOS CENTIGRADOS- Y BAJO PRESION. TAMBIEN PUEDE EMPLEARSE COMO REACTIVO EL AMONIACO LIQUIDO. SE OBTIENE EL COMPUESTO (III) EN QUE R'' ES HIDROGENO, CLORO, BROMO O ALLQUILO C1-4 Y R2 ES HIDROGENO O METILO. PUEDEN OBTENERSE LAS FORMAS TAUTOMERAS DE COMPUESTO (II).
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH499580 | 1980-06-27 |
Publications (2)
Publication Number | Publication Date |
---|---|
ES503407A0 ES503407A0 (es) | 1982-10-01 |
ES8207541A1 true ES8207541A1 (es) | 1982-10-01 |
Family
ID=4286126
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES503407A Expired ES8207541A1 (es) | 1980-06-27 | 1981-06-26 | Procedimiento para la preparacion de derivados de pirimidina |
Country Status (25)
Country | Link |
---|---|
US (2) | US4376121A (es) |
EP (1) | EP0043054B1 (es) |
JP (1) | JPS5762282A (es) |
KR (1) | KR840000705B1 (es) |
AR (1) | AR230748A1 (es) |
AT (1) | ATE9698T1 (es) |
AU (1) | AU7196781A (es) |
BR (1) | BR8103967A (es) |
CA (1) | CA1142924A (es) |
CS (1) | CS217997B2 (es) |
CU (1) | CU35489A (es) |
DE (1) | DE3166449D1 (es) |
DK (1) | DK252981A (es) |
ES (1) | ES8207541A1 (es) |
FI (1) | FI811600L (es) |
GR (1) | GR74943B (es) |
HU (1) | HU181608B (es) |
IL (1) | IL63145A (es) |
MC (1) | MC1395A1 (es) |
NO (1) | NO812208L (es) |
NZ (1) | NZ197476A (es) |
PH (1) | PH16060A (es) |
PT (1) | PT73270B (es) |
ZA (1) | ZA814162B (es) |
ZW (1) | ZW11781A1 (es) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ZW11781A1 (en) * | 1980-06-27 | 1982-01-20 | Hoffmann La Roche | Pyrimidine derivatives |
US4797486A (en) * | 1986-09-08 | 1989-01-10 | Pfizer Inc. | Heterocyclic ring fused pyrimidine-4(3H)-ones as anticoccidial agents |
US4725599A (en) * | 1986-09-08 | 1988-02-16 | Pfizer Inc. | Heterocyclic ring fused pyrimidine-4 (3H)-ones as anticoccidial agents |
DK522187D0 (da) * | 1987-10-06 | 1987-10-06 | Ferrosan As | Imidozothienopyrimidiner, deres fremstilling og anvendelse |
DK0888359T3 (da) | 1996-03-11 | 2002-08-12 | Syngenta Participations Ag | Pyrimidin-4-on-derivat som pesticid |
FR2872165B1 (fr) | 2004-06-24 | 2006-09-22 | Sod Conseils Rech Applic | Nouveaux derives de pyrimido-benzimidazole |
US8809346B2 (en) * | 2008-05-30 | 2014-08-19 | Universite De Versailles-Saint-Quentin-En-Yvelines | ANT-ligands molecules and biological applications |
CN104478851A (zh) * | 2014-12-31 | 2015-04-01 | 济南诚汇双达化工有限公司 | 一种盐酸阿替卡因的制备方法 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE755404A (fr) * | 1969-08-29 | 1971-03-01 | Sandoz Sa | Nouveau derives de la thiazolo-(3,2-a) pyrrolo (2,3-d) pyrimidine, leurpreparation et medicaments contenant ces derives |
US3932407A (en) * | 1973-11-19 | 1976-01-13 | Bristol-Myers Company | Optionally substituted 1,2,3,5-tetrahydroimidezo(2,1-b)-quinazolin-2-ones and 6(H)-1,2,3,4-tetrahydropyimido(2,1-b)quinazolin-2-ones |
DE2411274A1 (de) * | 1974-03-06 | 1975-09-18 | Schering Ag | Neue 2-nitrothieno eckige klammer auf 2,3-d eckige klammer zu pyrimidinon-derivate und verfahren zu ihrer herstellung |
DE2411273A1 (de) * | 1974-03-06 | 1975-09-18 | Schering Ag | Neue thieno eckige klammer auf 2,3-d eckige klammer zu pyrimidinone und verfahren zu ihrer herstellung |
US4054656A (en) * | 1975-09-10 | 1977-10-18 | Mead Johnson & Company | Thieno[2,3-d]pyrimidine antiallergic agents |
JPS5527105A (en) * | 1978-08-11 | 1980-02-27 | Dai Ichi Seiyaku Co Ltd | Imidazothienopyrimidinones compound |
US4230707A (en) * | 1979-08-27 | 1980-10-28 | Warner-Lambert Company | Oxo-pyrido[1,2-a]thienopyrimidine compounds and methods for their production |
ZW11781A1 (en) * | 1980-06-27 | 1982-01-20 | Hoffmann La Roche | Pyrimidine derivatives |
-
1981
- 1981-05-14 ZW ZW117/81A patent/ZW11781A1/xx unknown
- 1981-05-14 CA CA000377588A patent/CA1142924A/en not_active Expired
- 1981-05-25 FI FI811600A patent/FI811600L/fi not_active Application Discontinuation
- 1981-05-27 CS CS813920A patent/CS217997B2/cs unknown
- 1981-06-10 DK DK252981A patent/DK252981A/da not_active Application Discontinuation
- 1981-06-19 AU AU71967/81A patent/AU7196781A/en not_active Abandoned
- 1981-06-19 ZA ZA814162A patent/ZA814162B/xx unknown
- 1981-06-19 US US06/275,271 patent/US4376121A/en not_active Expired - Fee Related
- 1981-06-19 NZ NZ197476A patent/NZ197476A/en unknown
- 1981-06-22 IL IL63145A patent/IL63145A/xx unknown
- 1981-06-22 EP EP81104750A patent/EP0043054B1/de not_active Expired
- 1981-06-22 DE DE8181104750T patent/DE3166449D1/de not_active Expired
- 1981-06-22 CU CU8135489A patent/CU35489A/es unknown
- 1981-06-22 AT AT81104750T patent/ATE9698T1/de active
- 1981-06-24 BR BR8103967A patent/BR8103967A/pt unknown
- 1981-06-24 HU HU811851A patent/HU181608B/hu unknown
- 1981-06-24 JP JP56096812A patent/JPS5762282A/ja active Pending
- 1981-06-25 PH PH25819A patent/PH16060A/en unknown
- 1981-06-25 GR GR65340A patent/GR74943B/el unknown
- 1981-06-25 MC MC811524A patent/MC1395A1/xx unknown
- 1981-06-26 ES ES503407A patent/ES8207541A1/es not_active Expired
- 1981-06-26 AR AR285881A patent/AR230748A1/es active
- 1981-06-26 PT PT73270A patent/PT73270B/pt unknown
- 1981-06-26 NO NO812208A patent/NO812208L/no unknown
- 1981-06-26 KR KR1019810002316A patent/KR840000705B1/ko active
-
1982
- 1982-12-23 US US06/452,677 patent/US4442289A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
HU181608B (en) | 1983-10-28 |
KR830006302A (ko) | 1983-09-20 |
ZW11781A1 (en) | 1982-01-20 |
PH16060A (en) | 1983-06-09 |
ES503407A0 (es) | 1982-10-01 |
US4442289A (en) | 1984-04-10 |
CS217997B2 (en) | 1983-02-25 |
ZA814162B (en) | 1982-07-28 |
PT73270A (en) | 1981-07-01 |
AR230748A1 (es) | 1984-06-29 |
CU35489A (en) | 1982-12-22 |
FI811600L (fi) | 1981-12-28 |
JPS5762282A (en) | 1982-04-15 |
NZ197476A (en) | 1984-05-31 |
ATE9698T1 (de) | 1984-10-15 |
EP0043054B1 (de) | 1984-10-03 |
BR8103967A (pt) | 1982-03-09 |
EP0043054A3 (en) | 1982-03-17 |
CA1142924A (en) | 1983-03-15 |
EP0043054A2 (de) | 1982-01-06 |
PT73270B (en) | 1983-05-11 |
DE3166449D1 (en) | 1984-11-08 |
MC1395A1 (fr) | 1982-04-27 |
KR840000705B1 (ko) | 1984-05-21 |
AU7196781A (en) | 1982-01-07 |
US4376121A (en) | 1983-03-08 |
IL63145A0 (en) | 1981-09-13 |
IL63145A (en) | 1984-05-31 |
GR74943B (es) | 1984-07-12 |
NO812208L (no) | 1981-12-28 |
DK252981A (da) | 1981-12-28 |
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